keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Prosaptide TX14(A) acetate is a potent GPR37L1 and GPR37 agonist. Prosaptide Tx14(A) TFA increases both ERK1 and ERK2 phosphorylation in Schwann cells.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 34,000 | |||
5 mg | 在庫あり | ¥ 84,000 | |||
10 mg | 在庫あり | ¥ 125,000 | |||
25 mg | 在庫あり | ¥ 201,500 | |||
50 mg | 在庫あり | ¥ 273,500 | |||
100 mg | 在庫あり | ¥ 374,000 |
説明 | Prosaptide TX14(A) acetate is a potent GPR37L1 and GPR37 agonist. Prosaptide Tx14(A) TFA increases both ERK1 and ERK2 phosphorylation in Schwann cells. |
ターゲット&IC50 | GPR37:7 nM(EC50), GPR37L1:5 nM(EC50) |
In vitro | Prosaptide Tx14(A) is a potent GPR37L1(EC50: 5 nM) and GPR37(EC50: 7 nM) agonist, bound to both receptors and activated signaling in a GPR37- and GPR37L1-dependent manner[1]. |
別名 | Prosaptide TX14(A) acetate(196391-82-9 free base) |
分子量 | 1639.76 |
分子式 | C71H114N16O28 |
CAS No. | TP1970L |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. 詳細
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Prosaptide TX14(A) acetate TP1970L Endocrinology/Hormones GPCR/G Protein MAPK GPR ERK Prosaptide TX14(A) acetate(196391-82-9 free base) Prosaptide TX-14(A) acetate Prosaptide TX14(A) Acetate Inhibitor inhibitor inhibit