Powder: -20°C for 3 years | In solvent: -80°C for 1 year
S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of 0.5 and 112 nM respectively.
説明 | S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of 0.5 and 112 nM respectively. |
ターゲット&IC50 | MT1:0.5 nM(Ki), MT2:112 nM(Ki) |
In vitro | S26131 is an effective and selective antagonist of MT1 and MT2 with KBs of 5.32 and 143 nM, respectively[1]. |
別名 | N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide |
分子量 | 498.61 |
分子式 | C31H34N2O4 |
CAS No. | 296280-56-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (50.14 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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S26131 296280-56-3 Neuroscience MT Receptor inhibit melatoninergic ligand MT2 antagonist selectively Melatonin Receptor N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide Inhibitor S 26131 S-26131 inhibitor