Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a reactive conformation.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 30,500 | |||
5 mg | 在庫あり | ¥ 69,500 | |||
10 mg | 在庫あり | ¥ 104,000 | |||
25 mg | 在庫あり | ¥ 171,500 | |||
50 mg | 在庫あり | ¥ 241,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 86,000 |
説明 | SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a reactive conformation. |
ターゲット&IC50 | EGFR:429 nM, HER2:11 nM, HER4: > 10000 nM |
In vitro | IC50 data: HER2 = 11 nM; EGFR = 429 nM; HER4 > 10000 nM |
別名 | SYR-127063, BDBM 92454, SYR 127063, BDBM-92454, BDBM92454 |
分子量 | 492.88 |
分子式 | C23H20ClF3N4O3 |
CAS No. | 871026-18-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (111.59 mM)
H2O: Insoluble
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
SYR127063 871026-18-5 Angiogenesis JAK/STAT signaling Tyrosine Kinase/Adaptors EGFR HER SYR-127063 BDBM 92454 SYR 127063 BDBM-92454 BDBM92454 Inhibitor inhibitor inhibit