Powder: -20°C for 3 years | In solvent: -80°C for 1 year
TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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5 mg | 在庫あり | ¥ 9,000 | |||
10 mg | 在庫あり | ¥ 14,000 | |||
25 mg | 在庫あり | ¥ 30,500 | |||
50 mg | 在庫あり | ¥ 52,000 | |||
100 mg | 在庫あり | ¥ 83,500 | |||
200 mg | 在庫あり | ¥ 121,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 15,500 |
説明 | TRPM4-IN-1 (4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid) is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM. |
ターゲット&IC50 | TRPM4:1.5 μM |
In vitro | TRPM4-IN-1 selectively inhibits TRPM4 overexpressed in HEK293 cells. TRPM4-IN-1 inhibits endogenous TRPM4 currents in LNCaP cells. TRPM4-IN-1 restores functional expression of A432T, a loss‐of‐expression TRPM4 variant. |
別名 | CBA, 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid |
分子量 | 340.16 |
分子式 | C15H11Cl2NO4 |
CAS No. | 351424-20-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 80 mg/mL(235.18 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
TRPM4-IN-1 351424-20-9 Membrane transporter/Ion channel TRP/TRPV Channel TRP Channel Transient receptor potential channels non-selective TRPM4IN1 diseases TRPM4 CBA inhibit Inhibitor TRPM-4-IN-1 TRPM4 IN 1 cancer cation cardiac 4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid channel prostate calcium-activated inhibitor