Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against δPI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, β, and γ).
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 53,500 |
2 mg | 在庫あり | ¥ 79,500 |
5 mg | 在庫あり | ¥ 134,000 |
10 mg | 在庫あり | ¥ 192,000 |
25 mg | 在庫あり | ¥ 291,500 |
50 mg | 在庫あり | ¥ 388,000 |
100 mg | 在庫あり | ¥ 525,500 |
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 189,500 |
説明 | Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against δPI3 kinase is at least 20 times lower than that of the inhibitors against other PI3K isoforms (A, β, and γ). |
別名 | TGR-1202 R-enantiomer, RP5264 R-enantiomer |
分子量 | 571.55 |
分子式 | C31H24F3N5O3 |
CAS No. | 1532533-69-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 9 mg/mL (15.75 mM)
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Umbralisib R-enantiomer 1532533-69-9 PI3K/Akt/mTOR signaling PI3K TGR-1202 R-enantiomer RP5264 R-enantiomer Inhibitor inhibitor inhibit