Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Upacicalcet (AJT-240) is an intraventricular calcium mimetic, a SHPT available for human hemodialysis, that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on parathyroid cell membrane calcium-sensitive receptors, thereby lowering blood levels of PTH.Upacicalcet is an orthosteric modulator of calcium-sensitive receptors and prevents adenine-induced secondary vascular calcification and bone disease in a rat model of adenine-induced secondary hyperparathyroidism.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 25,500 | |||
5 mg | 在庫あり | ¥ 62,000 | |||
10 mg | 在庫あり | ¥ 92,000 | |||
25 mg | 在庫あり | ¥ 153,500 | |||
50 mg | 在庫あり | ¥ 218,000 | |||
100 mg | 在庫あり | ¥ 296,000 | |||
500 mg | 在庫あり | ¥ 592,500 |
説明 | Upacicalcet (AJT-240) is an intraventricular calcium mimetic, a SHPT available for human hemodialysis, that inhibits excessive parathyroid hormone (PTH) secretion by directly acting on parathyroid cell membrane calcium-sensitive receptors, thereby lowering blood levels of PTH.Upacicalcet is an orthosteric modulator of calcium-sensitive receptors and prevents adenine-induced secondary vascular calcification and bone disease in a rat model of adenine-induced secondary hyperparathyroidism. |
別名 | PLS-240, SK-1403, AJT-240 |
分子量 | 351.76 |
分子式 | C11H14ClN3O6S |
CAS No. | 1333218-50-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (142.14 mM)
You can also refer to dose conversion for different animals. 詳細
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Upacicalcet 1333218-50-0 Membrane transporter/Ion channel Metabolism Calcium Channel PLS-240 AJT240 SK1403 PLS 240 SK-1403 SK 1403 AJT 240 AJT-240 PLS240 Inhibitor inhibitor inhibit