Powder: -20°C for 3 years | In solvent: -80°C for 1 year
VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.
ターゲット&IC50 | KCC2:560 nM |
別名 | N-(4-Methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide, VU0240551-2-D4 |
分子量 | 342.44 |
分子式 | C16H14N4OS2 |
CAS No. | 893990-34-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: Insoluble
DMSO: 45 mg/mL (131.4 mM)
You can also refer to dose conversion for different animals. 詳細
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VU 0240551 893990-34-6 Angiogenesis JAK/STAT signaling Membrane transporter/Ion channel Metabolism Tyrosine Kinase/Adaptors Potassium Channel Calcium Channel HER VU0240551 N-(4-Methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide VU0240551-2-D4 VU-0240551 Inhibitor inhibitor inhibit