store at low temperature,keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
HS-276 is a highly selective, orally active inhibitor of TAK1 (Ki: 2.5 nM). HS-276 significantly inhibits TAK1 (IC50: 8.25 nM), CLK2 (IC50: 29 nM), GCK (IC50: 22 nM), ULK2 (IC50: 63 nM), MAP4K5 (IC50. HS-276 can be used to study rheumatoid arthritis (RA).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 21,000 | |||
5 mg | 在庫あり | ¥ 49,000 | |||
10 mg | 在庫あり | ¥ 76,500 | |||
25 mg | 在庫あり | ¥ 135,000 | |||
50 mg | 在庫あり | ¥ 196,500 | |||
100 mg | 在庫あり | ¥ 271,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 54,000 |
説明 | HS-276 is a highly selective, orally active inhibitor of TAK1 (Ki: 2.5 nM). HS-276 significantly inhibits TAK1 (IC50: 8.25 nM), CLK2 (IC50: 29 nM), GCK (IC50: 22 nM), ULK2 (IC50: 63 nM), MAP4K5 (IC50. HS-276 can be used to study rheumatoid arthritis (RA). |
ターゲット&IC50 | NUAK:270 nM, CaMKK β1:1280 nM, MAP4K5:125 nM, TAK1:8.25 nM, TAK1:2.5 nM (Ki), ULK2:63 nM, GCK:33 nM, CLK2:29 nM, CSNK1G2:810 nM, MLK1:5585 nM, IRAK1:264 nM |
分子量 | 419.52 |
分子式 | C24H29N5O2 |
CAS No. | 2767422-72-8 |
store at low temperature,keep away from direct sunlight
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45.0 mg/mL (107.3 mM), when pH is adjusted to 2 with HCl. Sonication and heating to 80℃ are recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
HS-276 2767422-72-8 MAPK Inhibitor inhibitor inhibit