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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T29112 | VPC171 | VPC 171,VPC-171 | Adenosine Receptor |
VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM). | |||
T15623 | JNJ-61432059 | iGluR | |
JNJ-61432059 is an oral active and selective negative modulator of AMPAR associated with trans-membrane AMPAR regulatory protein (TARP) γ-8 (pIC50: 9.7 for GluA1/γ-8). | |||
T10774 | CFM-2 | iGluR | |
CFM-2, a potent and selective non-competitive antagonist of AMPAR (AMPAR), exhibits anticonvulsant activity across various seizure models. | |||
T16524 | Philanthotoxin 74 dihydrochloride | PhTx-74 HCl,PhTx 74 dihydrochloride | GluR , iGluR |
Philanthotoxin 74 dihydrochloride is an antagonist of AMPAR with IC50s of 263 and 296 nM for GluR3 and GluR1. | |||
T17179 | Tulrampator | CX-1632,S-47445 | iGluR |
Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects. | |||
T12187L | Naspm trihydrochloride | 1-Naphthylacetyl spermine trihydrochloride | iGluR |
T23267 | (RS)-AMPA hydrobromide | Others | |
AMPAR agonist | |||
T13480L | (S)-(-)-5-Fluorowillardiine hydrochloride | (S)-5-Fluorowillardiine hydrochloride,(5S)-Fluorowillardiine hydrochloride | Others |
(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR. | |||
T31979 | GNE-3476 | GNE 3476 | |
GNE-3476 is an NMDA receptor PAM. Ge-3476 has different degrees of activity on different receptors.GNE-3476 has relatively low efficacy on GluN2A, some activity as an AMPAR PAM, and weak activity at GluN2B-containing rec... | |||
T78971 | AMPA receptor modulator-4 | iGluR | |
AMPA Receptor Modulator-4, a 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide (BTD), serves as an orally active positive allosteric modulator of the AMPA receptors (AMPAR PAMs). This compound is capable of crossing the ... | |||
T16505 | PF-4778574 | Others | |
PF-4778574 is a positive AMPA receptor allosteric modulation (EC50: 45 to 919 nM in different cells). |