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T24840 |
STS-E412
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STS E412,STSE412 |
Others
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STS-E412 is a tissue-protective and selective EPOR/CD131 receptor activator for the study of neurological disorders. |
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T2577 |
Dienogest
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STS 557 |
Apoptosis
,
Estrogen/progestogen Receptor
,
Progesterone Receptor
,
Autophagy
|
|
Dienogest (STS 557) is an orally-active, semisynthetic, fourth generation, nonethinylated progestogen with antiproliferative, antiandrogenic, anti-inflammatory and antiangiogenic activities that is used in hormone therap... |
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T11416 |
Glucagon receptor antagonists-5
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Others
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Glucagon receptor antagonists-5 is an orally bioavailable indazole-based glucagon receptor antagonist (Ki: 32 nM). It has potential for the treatment of type 2 diabetes mellitus (T2DM). |
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T126527 |
Poststerone
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Poststerone is a useful organic compound for research related to life sciences and the catalog number is T126527. |
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TP2421 |
Ysdspstst peptide
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Ysdspstst peptide is a biochemical. |
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T11415 |
Glucagon receptor antagonists-3
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Others
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|
Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist. |
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T11414 |
Glucagon receptor antagonists-2
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Others
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|
Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist. |
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T11413 |
Glucagon receptor antagonists-1
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Others
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Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist. |
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T25973 |
Poststatin
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Poststatin is a prolyl endopeptidase inhibitor produced by Streptomyces viridochromogenes MH534-30F3. |
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T15584 |
Integrin Antagonists 27
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Others
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Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist. It has a binding affinity of 18 nM and as a novel anticancer agent. |
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T10665 |
Calcium-Sensing Receptor Antagonists I
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Others
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Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium. |
|
T72470 |
Estrone O-sulfamate
|
Estrone 3-O-sulfamate |
Others
|
|
Estrone O-sulfamate (Estrone 3-O-sulfamate) is a potent inhibitor of steroid sulfatase (STS). Estrone O-sulfamate is a placental microsomal inhibitor (P.M.) with IC50 values of 18 nM. Estrone O-sulfamate showed inhibitor... |
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T81089 |
Steroid sulfatase-IN-7
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Steroid sulfatase-IN-7 is an irreversible inhibitor of steroid sulfatase (STS), demonstrating potent activity with an IC50 of 0.05 nM against human placental STS, rendering it suitable for application in cancer research ... |
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T81090 |
Steroid sulfatase-IN-6
|
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Steroid Sulfatase-IN-6 (Compound 10c) serves as an irreversible steroid sulfatase (STS) inhibitor, exhibiting a K i value of 0.4 nM against human placenta STS, and is applicable in tumor disease research [1]. |
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T62237 |
Steroid sulfatase-IN-4
|
|
|
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Steroid sulfatase-IN-4 (Compound 16) is an irreversible inhibitor of steroid sulfatase (STS) that acts on human STS (IC50: 25 nM). steroid sulfatase-IN-4 can be used to study endometriosis. |
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T62236 |
Steroid sulfatase/17β-HSD1-IN-3
|
|
|
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Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1). Steroid sulfatase/17β-HSD1-IN-3 can be used to study endometriosis and ... |
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T61979 |
Steroid sulfatase/17β-HSD1-IN-4
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Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ). Steroid sulfatase/17β-HSD1-IN-4 irreversibly inhibits hSTS a... |
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T81092 |
Steroid sulfatase/17β-HSD1-IN-5
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Steroid sulfatase/17β-HSD1-IN-5 serves as an irreversible inhibitor of steroid sulfatase (STS) and a reversible, selective inhibitor of 7β-hydroxysteroid dehydrogenase type1 (17β-HSD1), exhibiting IC50 values of 43 nM fo... |
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T61212 |
Steroid sulfatase-IN-2
|
|
|
|
Steroid sulfatase-IN-2 is an active inhibitor of steroid sulfatase (STS), demonstrating an IC50 value of 109.5 nM. Its potential application lies in hormone-dependent cancer research, specifically estrogen-dependent brea... |
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T61686 |
Steroid sulfatase-IN-3
|
|
|
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Steroid sulfatase-IN-3 (compound 1q) is a highly effective Steroid sulfatase (STS) inhibitor, exhibiting an IC 50 value of 25.8 nM. This compound also demonstrates antiproliferative properties against T-47D estrogen-depe... |
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T81091 |
Steroid sulfatase-IN-5
|
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|
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Steroid sulfatase-IN-5 (compound 10b), an inhibitor of steroid sulfatase (STS) with an IC50 of 0.32 nM, effectively suppresses T-47D breast cancer cell proliferation, demonstrating an IC50 value of 35.7 μM. This compound... |
