ホーム 計算ツール
代理店ログイン

BCRP

The breast cancer resistance protein (BCRP), this protein functions as a xenobiotic transporter which may play a role in multi-drug resistance to chemotherapeutic agents including mitoxantrone and camptothecin analogues.
Cat. No. 製品名 CAS No. Purity Chemical Structure
T38400 Triclabendazole sulfoxide 100648-13-3 98%
Triclabendazole sulfoxide is a main plasma metabolite of Triclabendazole. Triclabendazole sulfoxide inhibits membrane transporter ABCG2/BCRP and exhibits anti-pa...
T4595 YHO-13177 912287-56-0 98%
YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells and no effect on P-glycoprotein–mediated paclitaxel r...
T13365 YHO-13351 free base 912288-64-3 98%
YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .
T3208 Brevianamide F 38136-70-8 98%
Brevianamide F, also known as cyclo-(L-Trp-L-Pro), belongs to a class of naturally occurring 2,5-diketopiperazines. Brevianamide F possess interesting breast can...
T13383 Zamicastat 1080028-80-3 98%
Zamicastat is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0...
TQ0186 Ko 143 461054-93-3 98%
Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).
T2657 Elacridar 143664-11-3 98%
Elacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.
T3581 KS176 1253452-78-6 98%
KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter, showing no inhibitory activity against P-gp or MR...
T4337 PCI 29732 330786-25-9 98%
PCI 29732 is a selective and irreversible Btk inhibitor with IC50 of 8.2 nM in a FRET based biochemical enzymology assay.
T15355 Fumitremorgin C 118974-02-0 98%
Fumitremorgin C is a potent and selective inhibitor of ABCG2/BRCP.
TN3150 6,8-Diprenylnaringenin 68236-11-3 98%
6,8-Diprenylnaringenin is a natural product from hop Humulus lupulus. 6,8-Diprenylnaringenin is a breast cancer resistance protein(BCRP) inhibitor with some estr...
T67821 GS-9191 PM 98%
GS-9191 PM is a novel antitumorviral compound, a bis-amide prodrug of the nucleotide analog 9-(2-phosphonomethoxyethyl)-N6-cyclopropyl-2,6-diaminopurine (cPrPMED...
Triclabendazole sulfoxide
T38400
Triclabendazole sulfoxide is a main plasma metabolite of Triclabendazole. Triclabendazole sulfoxide inhibits membrane transporter ABCG2/BCRP and exhibits anti-pa...
YHO-13177
T4595
YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells and no effect on P-glycoprotein–mediated paclitaxel r...
YHO-13351 free base
T13365
YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .
Brevianamide F
T3208
Brevianamide F, also known as cyclo-(L-Trp-L-Pro), belongs to a class of naturally occurring 2,5-diketopiperazines. Brevianamide F possess interesting breast can...
Zamicastat
T13383
Zamicastat is an inhibitor of dopamine β-hydroxylase (DBH), and is also a concentration-dependent dual inhibitor of P-gp and BCRP(IC50 values of 73.8 μM and 17.0...
Ko 143
TQ0186
Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).
Elacridar
T2657
Elacridar (GF120918) is an effective BCRP and P-gp (MDR-1) inhibitor.
KS176
T3581
KS176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter, showing no inhibitory activity against P-gp or MR...
PCI 29732
T4337
PCI 29732 is a selective and irreversible Btk inhibitor with IC50 of 8.2 nM in a FRET based biochemical enzymology assay.
Fumitremorgin C
T15355
Fumitremorgin C is a potent and selective inhibitor of ABCG2/BRCP.
6,8-Diprenylnaringenin
TN3150
6,8-Diprenylnaringenin is a natural product from hop Humulus lupulus. 6,8-Diprenylnaringenin is a breast cancer resistance protein(BCRP) inhibitor with some estr...
GS-9191 PM
T67821
GS-9191 PM is a novel antitumorviral compound, a bis-amide prodrug of the nucleotide analog 9-(2-phosphonomethoxyethyl)-N6-cyclopropyl-2,6-diaminopurine (cPrPMED...