Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in uniform time-resolved fluorescence (htf) measurements using CHO cells expressing the human receptor (ECso-12.9 nM).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 11,000 | |||
5 mg | 在庫あり | ¥ 26,000 | |||
10 mg | 在庫あり | ¥ 41,000 | |||
25 mg | 在庫あり | ¥ 68,000 | |||
50 mg | 在庫あり | ¥ 95,500 | |||
100 mg | 在庫あり | ¥ 142,000 |
説明 | MK 1903 is a potent and selective complete agonist for the hydroxy-carboxylic acid receptor 2 (HCA2). HCA2 is also known as G protein-coupled receptor 109A(GPR109A). MK 1903 reduced Foschlin-induced cAMP production in uniform time-resolved fluorescence (htf) measurements using CHO cells expressing the human receptor (ECso-12.9 nM). |
In vivo | MK-1903 (Compound R, R-19a ) was well tolerated and produced a robust decrease in plasma-free fatty acids.[1] |
分子量 | 164.16 |
分子式 | C8H8N2O2 |
CAS No. | 1268882-43-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: < 8.21 mg/mL
DMSO: 112.5 mg/mL (685.3 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
MK 1903 1268882-43-4 Endocrinology/Hormones GPCR/G Protein GPR MK-1903 MK1903 Inhibitor inhibitor inhibit