Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 22,000 | |||
2 mg | 在庫あり | ¥ 33,000 | |||
5 mg | 在庫あり | ¥ 50,500 | |||
10 mg | 在庫あり | ¥ 75,500 | |||
25 mg | 在庫あり | ¥ 129,000 | |||
50 mg | 在庫あり | ¥ 181,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 51,000 |
説明 | Atherosperminine shows cholinesterase inhibitory activity against acetylcholinesterase (AChE) and butyrylcholinesterase (BChE). Atherosperminine exerts a non-specific relaxant effect on the trachealis, its major mechanism of action appears to be inhibition of cAMP phosphodiesterase. |
ターゲット&IC50 | DPPH:54.53 ug/mL, Anti-plasmodial:5.80 μM |
In vitro | Atherosperminine shows strong anti-plasmodial activity against Plasmodium falciparum, with the IC50 value of 5.80 μM. Atherosperminine also shows antioxidant activity in a DPPH assay with the IC50 value of 54.53 ug/mL[3]. |
植物由来 |
分子量 | 309.4 |
分子式 | C20H23NO2 |
CAS No. | 5531-98-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (161.6 mM)
You can also refer to dose conversion for different animals. 詳細
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Atherosperminine 5531-98-6 GPCR/G Protein Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience Calcium Channel cAMP AChR Parasite inhibit antiplasmodial Inhibitor pro-oxidant reductants Atherospermine trachealis inhibitor