Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Dehydroaripiprazole (DM-14857) is the active metabolite of aripiprazole. Aripiprazole is an antipsychotic drug, which is metabolized by CYP3A4 and CYP2D6 and mainly forms dehydroaripiprazole. Dehydroaripiprazole has antipsychotic activity equivalent to aripiprazole.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 7,500 | |||
5 mg | 在庫あり | ¥ 16,500 | |||
10 mg | 在庫あり | ¥ 28,000 | |||
25 mg | 在庫あり | ¥ 57,000 | |||
50 mg | 在庫あり | ¥ 84,500 | |||
100 mg | 在庫あり | ¥ 125,000 | |||
500 mg | 在庫あり | ¥ 266,500 |
説明 | Dehydroaripiprazole (DM-14857) is the active metabolite of aripiprazole. Aripiprazole is an antipsychotic drug, which is metabolized by CYP3A4 and CYP2D6 and mainly forms dehydroaripiprazole. Dehydroaripiprazole has antipsychotic activity equivalent to aripiprazole. |
ターゲット&IC50 | 5-HT1A:4.2 nM (ki) |
別名 | OPC-14857, DM-14857 |
分子量 | 446.37 |
分子式 | C23H25Cl2N3O2 |
CAS No. | 129722-25-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 11 mg/mL (24.65 mM)
You can also refer to dose conversion for different animals. 詳細
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Dehydroaripiprazole 129722-25-4 GPCR/G Protein Neuroscience 5-HT Receptor inhibit antipsychotic CYP3A4 Inhibitor OPC-14857 Metabolite Serotonin Receptor DM14857 DM 14857 OPC14857 OPC 14857 5-hydroxytryptamine Receptor CYP2D6 DM-14857 inhibitor