Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Naphthol AS-E (nAS-E) is an the KIX-KID interaction and CREB-mediated gene transcription inhibitor.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
50 mg | 在庫あり | ¥ 7,500 | |||
100 mg | 在庫あり | ¥ 11,000 | |||
200 mg | 在庫あり | ¥ 16,000 | |||
500 mg | 在庫あり | ¥ 26,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 12,000 |
説明 | Naphthol AS-E (nAS-E) is an the KIX-KID interaction and CREB-mediated gene transcription inhibitor. |
ターゲット&IC50 | c-Kit:2.26 μM (IC50) |
In vivo | nAS-E could reverse bone loss induced by MDA-MB-231 tumour.?These results suggest that small molecules targeting CREB-CBP interaction to inhibit CREB-mediated gene transcription might be a potential approach for the treatment of breast cancer bone metastasis[1]. |
別名 | nAS-E |
分子量 | 297.74 |
分子式 | C17H12ClNO2 |
CAS No. | 92-78-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 2.98 mg/mL (10 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Naphthol AS-E 92-78-4 Chromatin/Epigenetic Epigenetic Reader Domain Histone Acetyltransferase Naphthol AS E inhibit CBP KIX-KID A549 Inhibitor nAS-E MCF-7 HAT Naphthol ASE CREB cancer HATs inhibitor