Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel and elicited TrpA1-mediated nocifensive behaviour in mouse, with EC50 of 97 nM and 23 nM for rTrpA1 and hTrpA1, respectively.
説明 | PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel and elicited TrpA1-mediated nocifensive behaviour in mouse, with EC50 of 97 nM and 23 nM for rTrpA1 and hTrpA1, respectively. |
ターゲット&IC50 | TRPA1 (human):23 nM, TRPA1 (rat):97 nM |
分子量 | 466.62 |
分子式 | C26H38N6O2 |
CAS No. | 1332708-14-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.66 mg/mL (10 mM)
You can also refer to dose conversion for different animals. 詳細
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PF-4840154 1332708-14-1 Membrane transporter/Ion channel TRP/TRPV Channel licking nocifensive Inhibitor PF4840154 PF 4840154 non-electrophilic inhibit Transient receptor potential channels behavior TRP Channel inhibitor