Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Penfluridol (TLP-607) is a highly potent antipsychotic.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
25 mg | 在庫あり | ¥ 11,000 | |||
50 mg | 在庫あり | ¥ 14,000 | |||
100 mg | 在庫あり | ¥ 17,500 | |||
200 mg | 在庫あり | ¥ 27,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,000 |
説明 | Penfluridol (TLP-607) is a highly potent antipsychotic. |
ターゲット&IC50 | Dopamine receptor:1.6 μM(Ki) |
In vivo | Penfluridol inhibits the binding of dopamine to its receptors with a Ki value of 1.6 μM. At a concentration of 10 μM, Penfluridol suppresses the contractile response of isolated rabbit thoracic aortic rings to NE and KCl, as well as the calcium influx stimulated by NE or KCl. Additionally, Penfluridol selectively inhibits the binding of [3H]Nitrendipine to rat cerebral cortex membranes and competitively antagonizes potassium-induced, calcium-dependent contractions in the rat vas deferens. |
別名 | R-16341, TLP-607 |
分子量 | 523.97 |
分子式 | C28H27ClF5NO |
CAS No. | 26864-56-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: < 1 mg/mL (insoluble or slightly soluble)
Ethanol: 93 mg/mL (177.5 mM)
DMSO: 93 mg/mL (177.5 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Penfluridol 26864-56-2 Autophagy GPCR/G Protein Membrane transporter/Ion channel Metabolism Neuroscience Calcium Channel Dopamine Receptor Inhibitor Ca2+ channels R-16341 Ca channels R16341 R 16341 TLP607 inhibit TLP 607 TLP-607 inhibitor