Powder: -20°C for 3 years | In solvent: -80°C for 1 year
UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 11,000 | |||
10 mg | 在庫あり | ¥ 18,500 | |||
25 mg | 在庫あり | ¥ 33,500 | |||
50 mg | 在庫あり | ¥ 57,000 | |||
100 mg | 在庫あり | ¥ 85,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 12,000 |
説明 | UNC0379 is a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8. |
ターゲット&IC50 | SETD8:7.3 μM |
In vitro | UNC0379 is competitive with the peptide substrate and noncompetitive with the cofactor SAM. [1] |
分子量 | 413.56 |
分子式 | C23H35N5O2 |
CAS No. | 1620401-82-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 76 mg/mL (183.8 mM)
H2O: < 1 mg/mL (insoluble or slightly soluble)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
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