Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Bictegravir Sodium (GS-9883 Sodium) is a potent inhibitor of HIV-1 integrase, with an IC50 of 7.5 nM. Bictegravir Sodium exhibits potent and selective anti-HIV activity and low cytotoxicity
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 9,500 | |||
5 mg | 在庫あり | ¥ 14,000 | |||
10 mg | 在庫あり | ¥ 22,500 | |||
25 mg | 在庫あり | ¥ 45,500 | |||
50 mg | 在庫あり | ¥ 88,000 | |||
100 mg | 在庫あり | ¥ 130,500 | |||
500 mg | 在庫あり | ¥ 287,000 |
説明 | Bictegravir Sodium (GS-9883 Sodium) is a potent inhibitor of HIV-1 integrase, with an IC50 of 7.5 nM. Bictegravir Sodium exhibits potent and selective anti-HIV activity and low cytotoxicity |
ターゲット&IC50 | HIV-1 integrase:7.5 nM |
In vitro | Bictegravir Sodium potently inhibits HIV-1 replication in both MT-2 and MT-4 cells with EC50s of 1.5 and 2.4 nM, respectively, and selectivity indices (50% cytotoxic concentration [CC50]/EC50) of ∼6,800 in MT-2 cells and ∼1,500 in MT-4 cells[1]. |
別名 | GS-9883 Sodium |
分子量 | 471.36 |
分子式 | C21H17F3N3NaO5 |
CAS No. | 1807988-02-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 15.3 mg/mL (32.5 mM), Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. 詳細
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Bictegravir Sodium 1807988-02-8 Microbiology/Virology Proteases/Proteasome HIV Protease GS-9883 Sodium Inhibitor inhibitor inhibit