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T0168 |
Estradiol (cypionate)
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Depofemin,Estradiol cypionate |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor. |
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T2231 |
Estradiol dipropionate
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17-Beta-Estradiol-3,17-Dipropionate |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Progesterone Receptor
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Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol. |
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T0384 |
Estradiol benzoate
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Benzoestrofol,Benzhormovarine,Benovocylin |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility and secondary sexual characteristics in females. |
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T11235 |
Estradiol 3-sulfamate
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E2MATE,BLE 00084,ES-J 995 |
Estrogen Receptor/ERR
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Estradiol 3-sulfamate (BLE 00084) is an orally active and highly potent steroidal estrone sulfatase (ES) inhibitor.Estradiol 3-sulfamate has a K(i) value of 73 nM for ES in human placental microsomes and can be used in t... |
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T9604 |
Beta-Estradiol 17-hemisuccinate
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Estrogen Receptor/ERR
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beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells. |
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T72390 |
Estradiol hemihydrate
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17β-Oestradiol hemihydrate,β-Estradiol hemihydrate ; 17β-Estradiol hemihydrate ; 17β-Oestradiol hemihydrate,17β-Estradiol hemihydrate,β-Estradiol hemihydrate |
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Estradiol (β-Estradiol) hemihydrate, a key female sex hormone and steroid, plays a significant role in up-regulating neural markers in human endometrial stem cells (hEnSCs) and facilitating their neural differentiation. ... |
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T40580 |
17β-Estradiol sulfate sodium
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17β-Estradiol 3-sulfate sodium |
Antibiotic
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17β-Estradiol sulfate sodium (17β-Estradiol 3-sulfate sodium) is a neuroactive estrogen with vasoprotective properties that inhibits the growth of Neisseria brasiliensis and disrupts aquatic ecosystems. |
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T1536 |
Promestriene
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3-propyl ethyl,17B-methyl estradiol,Promestriano |
Estrogen/progestogen Receptor
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Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation. It is described as a tropic agent and antiseborrheic. |
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T37004 |
Estradiol 3-sulfate 17β-Glucuronide (potassium salt)
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Estradiol 3-sulfate is a sulfated form of the steroid hormone 17β-estradiol , and is common in fetal plasma and in the breast tissues of patients with mammary carcinoma. Sulfated estrogens, including estradiol 3-sulfate,... |
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T36917 |
Ethynyl Estradiol 3-β-D-Glucuronide (hydrate)
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Ethynyl estradiol 3-β-D-glucuronide is a metabolite of ethynyl estradiol that can be detected in urine.1,2It is used as a marker of estrogen contamination in fresh and saltwater.2
1.Hadd, H.E., Slikker, W., Jr., and Helt... |
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T31681 |
Estradiol undecylate
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AI352642,AI3-52642,AI3 52642 |
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Estradiol undecylate can be used in the treatment of prostatic cancer. |
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T36807 |
Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate)
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Estradiol 17-(β-D-glucuronide) (E217G) is an estrogen metabolite formed in the liver and subsequently excreted in bile.1It acts as a substrate of the multidrug resistance protein 2 (MRP2; Km= 75 μM), and through MRP2-med... |
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T18876 |
β-Estradiol-6-CMO-PEG3-biotin
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Others
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β-Estradiol-6-CMO-PEG3-biotin serves as a cleavable 3-unit PEG ADC linker for the synthesis of antibody-drug conjugates (ADCs)[1]. |
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T18877 |
β-Estradiol-6-one 6-(O-carboxymethyloxime)
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Others
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β-Estradiol-6-one 6-(O-carboxymethyloxime) is an alkyl chain-based PROTAC linker utilized for PROTAC synthesis[1]. |
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T65147 |
Estradiol enanthate
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Estradiol enanthate is a useful organic compound for research related to life sciences. The catalog number is T65147 and the CAS number is 4956-37-0. |
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T1579 |
Mestranol
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Devocin,Norquen,Menophase |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active. |
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T2569 |
Chlorotrianisene
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tris(p-methoxyphenyl)chloroethylene,CTA,tri-p-anisylchloroethylene,TACE |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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COX
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Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen receptor modulator (SERM), with predominantly estrogenic but... |
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T31699 |
Ethinylestradiol mixture with Levonorgestrel
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Ethinylestradiol mixture with Levonorgestrel is formulated with increasing dosages of levonorgestrel and ethinyl estradiol. |
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T31578 |
Drospirenone mixture with Ethinylestradiol
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Yaz 28,Nikki,Ocella,Yaz-28,Yasmin 28,Syeda |
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Drospirenone mixture with Ethinylestradiol is a female oral combined contraceptive containing 30 mcg (0.030 mg) Ethinyl Estradiol and 3 mg drospirenone (Androstenes). |
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T31715 |
Ethynylestradiol mixture with lynestrenol
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Ethynylestradiol mixture with lynestrenol is a drug/ therapeutic agent with reproductive effect. |
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T24973 |
2-Iodoestradiol
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2 Iodoestradiol,NSC671618,NSC 671618,NSC-671618 |
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2-Iodoestradiol is an effective human sex hormone-binding globulin (SHBG) ligand. |
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T131627 |
Oestradiol
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Oestradiol is a useful organic compound for research related to life sciences and the catalog number is T131627. |
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T14577 |
Biotin-DADOO
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EZ-Link Amine-PEO2-Biotin,Biotinyl-3,6-dioxaoctanediamine |
Others
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Biotin-DADOO (Biotinyl-3,6-dioxaoctanediamine) is a biotinylation reagent that can be used to synthesize a biotin-estradiol conjugate(i.e., biotin-DADOO-estradiol) to develop a direct, broad-range enzyme immunoassay to m... |
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T11399 |
Giredestrant
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GDC-9545 |
Estrogen Receptor/ERR
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Estrogen/progestogen Receptor
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Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has anti-tumor activity. Giredestrant, a non-steroidal ER ligand,... |
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T7537 |
Norgestimate
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Progesterone Receptor
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Norgestimate is an acetylated progestinused in combination with ethinyl estradiol as an oral contraceptive. |
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T10239 |
Acolbifene
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EM-652,SCH 57068 |
Estrogen Receptor/ERR
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Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifene shows an anticarcinogenic property. |
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T25048 |
Algestone acetophenide
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Neolutin |
Others
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Algestone acetophenide (Neolutin) is progesterone that used in estrus synchronization and has been evaluated as an injectable contraceptive in combination with estradiol enanthate. It is also used therapeutically as a to... |
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T20681 |
Estramustine
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NSC-89201,NSC 89201,LEO 275,LEO275,NSC89201,LEO-275 |
Microtubule Associated
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Estramustine (LEO-275) is a nitrogen mustard linked to estradiol, usually as phosphate. Estramustine has been used to treat prostatic neoplasms; also has radiation protective properties. Estramustine is selectively taken... |
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T22794 |
G36
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G-36 |
Estrogen Receptor/ERR
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G36 is a cell-permeable non-steroidal antagonist of GPER. G36 inhibits activation by either 17β-estradiol or the GPER-selective agonist G-1 (IC50 = 112 and 165 nM, respectively). G36 has no detectable binding activity to... |
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T14344 |
Atrimustine
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KM2210,Bestrabucil |
Others
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T26154 |
RU 45144
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RU45144,RU-45144 |
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RU 45144 is an estradiol derivative with antiestrogenic activity. |
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T10036 |
10β,17β-dihydroxyestra-1,4-dien-3-one
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DHED |
Others
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TP2010 |
Kisspeptin 10 (dog)
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Endogenous ligand for the canine KISS1 receptor (Kisspeptin receptor or GPR54). Stimulates section of luteinizing hormone, follicle stimulating hormone and estradiol in vivo. |
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T73765 |
Estrone 3-glucuronide
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Estrone 3-glucuronide, a deuterium-labeled version, is recognized as the primary metabolite of estradiol and serves as a urinary marker for predicting the fertile window [1]. |
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T36916 |
Estrone-3-Glucuronide (sodium salt hydrate)
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Estrone-3-Glucuronide is a metabolite of the primary premenopausal estrogen 17β-estradiol .1,2Urinary levels of estrone-3-Glucuronide peak approximately 36 hours prior to ovulation and have been used as a marker of ferti... |
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T36913 |
17-Epiestriol
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17-Epiestriol is a metabolite of estrone .1It is formed from estroneviaa 16α-hydroxy estrone intermediate by reduction of the C-17 ketone. 17-Epiestriol binds to estrogen receptor α (ERα) and ERβ with relative binding af... |
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T70399 |
TTC-352
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TTC-352 is an orally bioavailable selective human estrogen receptor alpha (ERalpha; ESR1; ERa) partial agonist (ShERPA), with potential antineoplastic activity. Upon administration, TTC-352 mimics the naturally-occurring... |
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T74335 |
PSDalpha
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PSDalpha, an ERα degrader consisting of a photosensitizer (PS), triphenylamine benzothiadiazole (TB), and 17β-estradiol connected via an acetylene bond, demonstrates superior anti-proliferative effects on MCF-7 cells. It... |
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T76222 |
HFSH-β-(33-53) (TFA)
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hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist. It prevents FSH from binding to its receptor and partially p... |
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T60827 |
TPBM
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TPBM is a potent inhibitor of estrogen receptor α (ERα). The IC 50 value of TPBM for 17β-estradiol (E2)-ERα is 9 μM. TPBM is not toxic to cells and reduces E2·ERα recruitment to an endogenous estrogen-responsive gene. TP... |
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T36039 |
16α-Hydroxyestrone
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The naturally-occurring estrogens are estrone , estradiol , and estriol . 16α-hydroxy Estrone (16α-OHE1) is a hydroxylated metabolite of E1 as well as an interconversion product with E2. E1 is 16α-hydroxylated by cytochr... |
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T70309 |
Dicetrorelix pamoate
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Dicetrorelix pamoate is a synthetic decapeptide with gonadotropin-releasing hormone (GnRH) antagonistic activity. GnRH induces the production and release of luteinizing hormone (LH) and follicle stimulating hormone (FSH)... |
