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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T6174 | R406 | R-406 besylate | Apoptosis , FLT , Syk |
R406 (R-406 besylate) is an effective Syk inhibitor (IC50: 41 nM) and shows no effects on Lyn. | |||
T2467 | R406 free base | R406 (free base) | Apoptosis , FLT , Syk |
R406 free base (R406 (free base)) is a potent Syk inhibitor. | |||
T6115 | Fostamatinib | R788 | FLT , Syk , Monoamine Transporter , Adenosine Receptor |
Fostamatinib (R788)(IC50 of 41 nM), which is a prodrug of the active metabolite R406, is a Syk inhibitor. It does not work on Lyn. | |||
T2605 | Fostamatinib Disodium | Tamatinib Fosdium,R788(Disodium),R788 Disodium,R788 (Fostamatinib) Disodium | FLT , Syk |
Fostamatinib Disodium (R788 Disodium) is an orally available Syk kinase inhibitor with potential anti-inflammatory and immunomodulating activities. |