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TP1271L |
Calmodulin-Dependent Protein Kinase II 290-309 acetate
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Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base) |
CaMK
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Calmodulin-Dependent Protein Kinase II 290-309 acetate is an effective antagonist of Ca2+/calmodulin-dependent protein kinase II (IC50 = 52 nM). |
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T75959 |
Calmodulin-Dependent Protein Kinase II(290-309) acetate
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Calmodulin-Dependent Protein Kinase II (290-309) acetate is a potent antagonist of CaMK, exhibiting an IC50 of 52 nM for the inhibition of Ca2+/calmodulin-dependent protein kinase II [1]. |
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T4380 |
Ac-CoA Synthase Inhibitor1
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ACSS2 inhibitor |
RSV
,
Fatty Acid Synthase
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Ac-CoA Synthase Inhibitor1 (ACSS2 inhibitor) is the most potent and specific inhibitor of acetate-dependent acetyl-CoA synthetase 2 (ACSS2). |
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TP1485L |
Calcineurin substrate acetate
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Autophagy
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Calcineurin substrate acetate is from the regulatory RII subunit of cAMP-dependent protein kinase. |
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T40437L |
Caloxin 2A1 acetate
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Proton pump
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Caloxin 2A1 acetate is an inhibitor of extracellular plasma membrane Ca2+-ATPase (PMCA) peptide. Caloxin 2A1 acetate inhibits Ca2+-dependent formation of the 140-kDa acid-stable acylphosphate. |
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T21470L |
Davunetide acetate
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Davunetide acetate(211439-12-2 Free base) |
Beta Amyloid
,
Microtubule Associated
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Davunetide acetate is derived from activity-dependent neuroprotective protein existing in the mammalian CNS. Davunetide acetate is a microtubule-stabilizing peptide and inhibits Aβ aggregation and Aβ-induced neurotoxicit... |
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T37422L |
Ras Inhibitory Peptide acetate
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Ras Inhibitory Peptide acetate(159088-48-9 Free base) |
Ras
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Ras Inhibitory Peptide acetate is a peptide involved in the Ras-dependent signaling pathway that plays an important role in human cancers initiated by oncogenic receptors. |
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TP1403L |
Syntide 2 acetate(108334-68-5 free base)
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CaMK
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Syntide-2 acetate is a synthetic peptide recognized as a substrate by Ca2+/calmodulin-dependent protein kinase II (CaMKII; Km = 12 μM). |
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TP2018L |
GIP (human) acetate
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GIP (human) acetate(100040-31-1 Free base) |
IGF-1R
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GIP (human) acetate is a stimulator of glucose-dependent insulin secretion and a weak inhibitor of gastric acid secretion. GIP (human) acetate plays a vital role in lipid metabolism and the development of obesity. |
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TP1914L1 |
BAM (8-22) acetate
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BAM (8-22) acetate(412961-36-5 free base) |
Others
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BAM (8-22) acetate is a proteolytically cleaved product of proenkephalin A. BAM (8-22) acetate activates Mas-related G-protein-coupled receptors (Mrgprs), MrgprC11 and hMrgprX1, and induces scratching in mice in an Mrgpr... |
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T37588L |
GIP (1-30) amide, porcine acetate
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IGF-1R
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GIP (1-30) amide, porcine acetate is an agonist of fully glucose-dependent insulinotropic polypeptide (GIP) receptor. GIP (1-30) amide, porcine acetate can weakly inhibit gastric acid secretion and strongly stimulate ins... |
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TP1220L |
Carperitide acetate
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Carperitide acetate (89213-87-6 Free base),Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate |
Endothelin Receptor
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Carperitide acetate (Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate), a 28-amino acid hormone, is naturally produced and released by the human heart upon cardiac injury or mechanical stretch. This compou... |
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T21983L |
PKI 14-22 amide, myristoylated Acetate
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PKI 14-22 amide, myristoylated Acetate(201422-03-9 Free base) |
PKA
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PKI 14-22 amide, myristoylated Acetate inhibit cAMP-dependent protein kinase (PKA) and blocks hyperalgesia produced by spinal administration of 8-bromo-cAMP. |
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TP1909L1 |
CALP2 acetate(261969-04-4 free base)
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CaMK
,
PDE
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CALP2 acetate is an antagonist of calmodulin showing high affinity for binding to the CaM EF-hand/Ca2+-binding site with a Kd of 7.9 µM. CALP2 acetate potently inhibits of adhesion and degranulation. CALP2 acetate is als... |
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T21309 |
Nafarelin acetate(76932-56-4 free base)
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RS-94991-298,Nafarelin acetate,Nafarelin acetate hydrate,Synarel |
GNRH Receptor
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Nafarelin acetate(76932-56-4 free base) (RS-94991-298) is a GnRH agonist that acts as an analog of GnRH. Nafarelin acetate(76932-56-4 free base) causes a decrease in the pituitary secretion of gonadotropins luteinizing h... |
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T3650 |
STO-609 acetate
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CaMK
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STO-609 acetate is selective, cell-permeable inhibitor of Ca2+-calmodulin-dependent protein kinase kinase (Ki: 80/15 ng/ml, for CaM-KKα/KKβ); competes for the ATP-binding site. It displays > 80-fold selectivity over CaMK... |
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TP1789L |
Malantide acetate(86555-35-3 free base)
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PKA
,
PKC
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Malantide acetate is a dodecapeptide phosphorylated by cyclic AMP-dependent protein kinase (PKA), and increases PKA activity.Malantide is a synthetic peptide that is phosphorylated by PKA and is used to measure PKA activ... |
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TP1787L |
PKG Substrate acetate（81187-14-6 free base)
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PKA
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PKG Substrate acetate is a selective substrate for cGMP-dependent protein kinase (PKG).PKG Substrate is a selective substrate for protein kinase G (PKG) with a strong preference for PKG Iα (Km = 59 μM) over PKG II (Km = ... |
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TP1051L |
Protein Kinase C Peptide Substrate acetate
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Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) |
Others
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Protein Kinase C Peptide Substrate acetate targets specific cell spacers ina manner that is dependent on second messengers and specific adaptor proteins in response to extracellular signals that activate g protein-couple... |
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T21410 |
Triptorelin acetate(57773-63-4 free base)
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Wy 42422,Triptorelin Acetate,CL 118532,AY 25650,CL 118,532,Wy 42462,BIM 21003 |
GNRH Receptor
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Triptorelin acetate(57773-63-4 free base) (CL 118,532) is used as a GnRH agonist. It decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle-stimulating hormone (FSH) by causing constant stim... |
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T37207L |
Cdk5 Substrate acetate
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CDK
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Cyclin-dependent kinase 5 (Cdk5) is a serine/threonine kinase that is predominantly active in neuronal tissues. With p25 or p35, Cdk5 phosphorylates a range of proteins, including histone H1 and tau. Cdk5 Substrate aceta... |
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TP1910L1 |
CALP1 acetate
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CALP1 acetate(145224-99-3 free base) |
CaMK
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CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site. CALP1 blocks calcium influx and apoptosis (IC50 of 44.78 µM) by inhibiting the open of calcium channel. CALP1 blo... |
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T37589L |
GIP (3-42), human acetate
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GIP (3-42), human acetate(1802086-25-4 Free base) |
IGF-1R
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GIP (3-42), human acetate is an antagonist of a glucose-dependent insulinotropic polypeptide (GIP) receptor and regulates insulin secretion and GIP metabolism in vivo. |
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T38063L |
N-Acetyl lysyltyrosylcysteine amide acetate
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N-Acetyl lysyltyrosylcysteine amide acetate(1287585-40-3 Free base) |
Glutathione Peroxidase
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N-Acetyl lysyltyrosylcysteine amide acetate is an effective and selective tripeptide inhibitor of myeloperoxidase (MPO). N-Acetyl lysyltyrosylcysteine amide acetate inhibits MPO-dependent hypochlorous acid (HOCl) genera... |
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T76262L |
Cagrilintide acetate
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Cagrilintide acetate, a long-acting acylated amylase analogue and non-selective AMYR/CTR agonist, effectively reduces food intake and induces significant weight loss in a dose-dependent manner, making it a valuable compo... |
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T76041 |
GIP (1-30) amide,human acetate
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GIP (1-30) amide, human acetate is a fragment of glucose-dependent insulinotropic polypeptide (GIP), an incretin hormone that plays a crucial role in stimulating insulin secretion and mitigating postprandial glycemic exc... |
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T36412 |
Multiflorenol
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Multiflorenol is a triterpene that has been found in T. kirilowii seeds.1 It inhibits in vitro activation of Epstein-Barr virus early antigen (EBV-EA) induced by the tumor promoter phorbol 12-myristate 13-acetate in a co... |
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T61358 |
AKN-028 acetate
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AKN-028 acetate, a novel tyrosine kinase (TK) inhibitor, is a potent, orally active FMS-like receptor tyrosine kinase 3 (FLT3) inhibitor with an IC 50 value of 6 nM. AKN-028 acetate inhibits FLT3 autophosphorylation. AKN... |
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T74072 |
R-BC154 acetate
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R-BC154 acetate, a selective fluorescent antagonist of α9β1 integrin, serves as a high-affinity, activation-dependent probe for investigating α9β1 and α4β1 integrin binding activity. This compound is particularly useful ... |
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T73658 |
Orexin A (human, rat, mouse) (acetate)
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Orexin A (Hypocretin-1) (human, rat, mouse) acetate, a hypothalamic neuropeptide with analgesic abilities that penetrates the blood-brain barrier, acts as an OX1R agonist. It promotes the expression of BDNF and TH protei... |
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T76048 |
TAK-683 acetate
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TAK-683 acetate is a nonapeptide metastin analog and a potent full agonist of the KISS1 receptor (KISS1R), exhibiting IC 50 =170 pM and enhanced metabolic stability. This compound shows agonistic activities towards KISS1... |
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TD0048 |
5-(and-6)-Carboxy SNARF-1, Acetoxymethyl Ester, Acetate
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The cell-permeant pH indicator, carboxy SNARF-1, acetoxymethyl ester, acetate (CAS #126208-13-7) has a pKa of ~7.5 after de-esterification, thus is useful for measuring pH changes between pH 7 and pH 8. Carboxy-SNARF-1 e... |
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T80084 |
Retatrutide acetate
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LY3437943 acetate |
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Retatrutide acetate (LY3437943) is a peptide that serves as a triple agonist for the glucagon receptor (GCGR), glucose-dependent insulinotropic polypeptide receptor (GIPR), and glucagon-like peptide-1 receptor (GLP-1R). ... |
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T71149 |
Triptorelin pamoate
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Triptorelin, a decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2), is a gonadotropin-releasing hormone agonist (GnRH agonist) used as the acetate or pamoate salts. By causing constant stimulation of the pituita... |
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T36998 |
7β,27-dihydroxy Cholesterol
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7β,27-DHC,7β,27-dihydroxy Cholesterol |
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7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt. [1] It activates RORγ- or RORγt-dependent signaling with EC50 values of 691 and 1,045 nM, res... |
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T36221 |
2-chloro Palmitic Acid
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2-chloro Palmitic acid is a monochlorinated form of palmitic acid . It is produced in a myeloperoxidase (MPO) and time-dependent manner in neutrophils stimulated by phorbol 12-myristate 13-acetate . 2-chloro Palmitic aci... |
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T68525 |
Nafarelin acetate hydrate
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Nafarelin is a gonadotropin-releasing hormone agonist (GnRH agonist) which acts as an analog of GnRH. Nafarelin increases the release of FSH and LH by the anterior pituitary, which in turn leads to an increase of estroge... |
