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T1312 |
Nafcillin sodium monohydrate
|
CL 8491,nafcillin sodium |
Antibacterial
,
Antibiotic
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Nafcillin sodium monohydrate (CL 8491) is the sodium salt form of nafcillin, a semi-synthetic naphthalene, penicillin-related Nafcillin inhibits bacterial wall synthesis by a mechanism of action similar to penicillin. Pe... |
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T0234 |
Methicillin sodium salt
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Methicillin sodium,Meticillin sodium |
Antibacterial
,
Antibiotic
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Methicillin sodium salt is the sodium salt form of methicillin, a semisynthetic beta-lactam penicillin antibiotic with beta-lactamase resistant activity. |
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T21358 |
Dalbavancin
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BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl |
Antibacterial
,
Antibiotic
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Dalbavancin (BI-397), a novel second-generation lipoglycopeptide antibiotic, possesses in vitro activity against a variety of Gram-positive pathogens including methicillin-resistant Staphylococcus aureus (MRSA) and methi... |
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T64316 |
VP-4604
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1-((4-Nitrophenyl)sulfonyl)piperidine |
Others
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VP-4604 is a potent anti-methicillin-resistant Staphylococcus aureus (MRSA) compound. VP-4604 exhibited significant microbial growth inhibition against S. aureus with an MIC of 4-8 μg/mL. VP-4604 inhibited the growth of ... |
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T22269 |
Benzyldodecyldimethylammonium Chloride Dihydrate
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Antibacterial
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Benzyldodecyldimethylammonium chloride dihydrate can be used as an insecticide reagent. It can target drug-resistant bacteria, such as methicillin-resistant Staphylococcus aureus, multidrug-resistant Pseudomonas aerugino... |
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T40475 |
Ceftobiprole medocaril
|
BAL5788 |
Antibacterial
|
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Ceftobiprole medocaril (BAL5788) is the parenteral prodrug of Ceftobiprole. Ceftobiprole is a broad-spectrum cephalosporin with activity against Methicillin-resistant staphylococcus aureus (MRSA). |
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TQ0077 |
Ceftobiprole
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Ro 63-9141,BAL 9141 |
Antibacterial
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Ceftobiprole (Ro 63-9141) is a broad-spectrum cephalosporin with activity against Methicillin-resistant staphylococcus aureus (MRSA; MIC90: 2 μg/mL). |
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T4208 |
Targocil
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Antibacterial
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Targocil is used as a bacteriostatic inhibitor of wall teichoic acid (WTA) biosynthesis which can inhibit the growth of methicillin-susceptible S. aureus (MSSA) and methicillin-resistant S. aureus (MRSA) (MIC90s: 2 μg/ m... |
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T0391 |
Linezolid
|
PNU-100766 |
MAO
,
Antibacterial
,
Antibiotic
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Linezolid (PNU-100766), the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistant bacteria including methicillin-resistant Staphylococcus aureus (MRS... |
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TN6672 |
Cyclo(L-Phe-L-Pro)
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Free radical scavengers
,
COX
,
Antibacterial
,
Antifungal
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Cyclo(L-Phe-L-Pro) shows broad-spectrum antibacterial and antifungal activities. Cyclo(L-Phe-L-Pro) exhibits activity against methicillin-resistant S. aureus and Enterococcus raffinosus. |
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T10579 |
BO3482
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Others
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BO3482 is an antimicrobial compound and can inhibit the growth of methicillin-resistant Staphylococci (MIC90: 6.25 mg/mL). |
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T30509 |
BMS-247243
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BMS247243,UNII-KG8365V22L |
Others
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BMS-247243 is a novel cephalosporin inhibitor that is mainly active against Gram-positive bacteria and also against methicillin-resistant Staphylococcus. |
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T1747L |
Tedizolid phosphate disodium salt
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Torezolid phosphate sodium salt,DA 7218,TR-701,TR 701 |
Others
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Tedizolid phosphate is a novel antibacterial prodrug. Tedizolid phosphate is a next-generation oxazolidinone with activity against both methicillin-resistant Staphylococcus aureus and vancomycin-resistant Enterococcus sp... |
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T26162 |
Rubradirin
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Others
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Rubradirin is an antibiotic with a complex chemical structure that is active vs. methicillin resistant staphylococci. It is a selective enzymatic peptide initiation inhibitor. |
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T26256 |
Teicoplanin aglycone
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TD-A3 |
Others
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Teicoplanin aglycone is an antibacterial glycopeptide antibiotic used in the prophylaxis and treatment of serious infections caused by Gram-positive bacteria, including Enterococcus faecalis and methicillin-resistant Sta... |
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T60525 |
VP-4556
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Others
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VP-4556 is a potent anti-methicillin-resistant Staphylococcus aureus ( MRSA ) agent that exhibits significant microbial growth inhibition against Staphylococcus aureus (ATCC 43300) (MIC = 8 μg/mL). VP-4556 inhibits methi... |
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T36032 |
Desotamide
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Others
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Desotamide is a cyclic hexapeptide antibiotic originally isolated from Streptomyces. It is active against S. aureus, S. pneumoniae, and methicillin-resistant S. epidermidis (MRSE; MICs = 16, 12.5, and 32 μg/ml, respectiv... |
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T61624 |
Antibacterial agent 106
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Others
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Antibacterial agent 106 (compound 8) is a highly effective orally active antibacterial compound with antibiofilm activity. It demonstrates potent antibacterial effects against multi-drug resistant (MDR)-Gram-positive pat... |
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T27964 |
Voxvoganan
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LTX109,Lytixar,LTX-109,LTX 109 |
Others
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Lytixar is a Synthetic Antimicrobial Peptide, it shows activity against Daptomycin-Nonsusceptible, Methicillin-Resistant, Vancomycin-Intermediate, Vancomycin-Resistant, and Linezolid-Nonsusceptible Staphylococcus aureus.... |
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T39816 |
Ceftaroline fosamil inner salt
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TAK-599 free acid,PPI0903freeacid |
Others
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Ceftaroline fosamil (TAK-599) inner salt, a cephalosporin derivative, is an N-phosphono prodrug of anti-methicillin-resistant Staphylococcus aureus (MRSA) T-91825. Ceftaroline fosamil inner salt can be used for the resea... |
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T83098 |
Antibacterial agent 163
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Others
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Antibacterial agent 163 (compound 1), a hydroxyquinoline derivative, potently inhibits methicillin-resistant Staphylococcus aureus (MRSA) [1]. |
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T39319 |
Actinomycin X2
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Actinomycin V |
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Actinomycin X2 (Actinomycin V) is a compound synthesized by various species of Streptomyces. It displays potent inhibition against methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentrati... |
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T37729 |
IMP-1700
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Others
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IMP-1700 is an inhibitor of bacterial DNA repair.1It potentiates the activity of the quinolone antibiotic ciprofloxacin against methicillin-resistantS. aureus(MRSA) with a combination index value of 0.7. IMP-1700 inhibit... |
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T37546 |
TPU-0037C
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Others
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TPU-0037C is a metabolite of the marine actinomycete S. platensis that is structurally similar to lydicamycin . It is active against Gram-positive bacteria (MICs = 0.39-3.13 μg/ml), including methicillin-resistant S. aur... |
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T74715 |
Antibacterial agent 136
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Others
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Antibacterial Agent 136 (Compound 3), an oxadiazolone antibiotic, exhibits high antibacterial potency against Methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) 50 value of ... |
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T37731 |
TPU-0037A
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Others
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TPU-0037A is an antibiotic and a congener of lydicamycin . It inhibits the growth of Gram-positive bacteria, including methicillin-resistant S. aureus (MRSA), B. subtilis, and M. luteus (MICs = 1.56-12.5 μg/ml), but not ... |
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T83097 |
Antibacterial agent 165
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Others
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Antibacterial agent 165 (compound 3), a hydroxyquinoline derivative, effectively inhibits methicillin-resistant Staphylococcus aureus (MRSA) [1], demonstrating its potent antibacterial properties. |
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T60546 |
Anti-MRSA agent 6
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Others
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Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1]. |
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T80276 |
Lynronne-3
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Lynronne-3, an antimicrobial peptide, demonstrates activity against Gram-positive bacteria, including multi-drug resistant (MDR) strains, with a minimum inhibitory concentration (MIC) ranging from 32-128 μg/mL for methic... |
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T37465 |
CAY10742
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Others
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CAY10742 is an orally bioavailable oxadiazole antibiotic.1It is active against the Gram-positive bacteriaS. aureus,S. epidermidis,S. haemolyticus,B. cereus,B. licheniformis,E. faecalis, andE. faecium(MICs = 1-4 μg/ml), i... |
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T28314 |
PD 117588
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PD117588,PD-117588 |
Others
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PD 117588 is a quinolone against bacterial isolates from cancer patients. PD 117558 has a broad antimicrobial spectrum with excellent activity against all Gram-positive isolates (including methicillin-resistant Staphyloc... |
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T38125 |
Platencin
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Others
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Platencin is a natural, broad spectrum Gram-positive antibiotic isolated from S. platensis, which is also the source of platensimycin . Platencin inhibits two key enzymes in bacterial fatty acid synthesis, β-ketoacyl-ACP... |
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T74803 |
Levonadifloxacin
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Others
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Levonadifloxacin ((S)-(-)-Nadifloxacin; WCK 771), a broad-spectrum anti-staphylococcal agent, exhibits antibacterial activity against both Methicillin-susceptible Staphylococcus aureus (MSSA) and Methicillin-resistant S.... |
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T61274 |
PC190723
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Others
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PC190723 (Compound 2), an inhibitor of the FtsZ bacterial cell division protein, demonstrates potent efficacy with an IC50 value of 55 ng/ml. Additionally, it showcases notable anti-staphylococcal activity, characterized... |
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T64315 |
VP-4509
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Others
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VP-4509 is an anti-methicillin-resistant Staphylococcus aureus (MRSA) agent (MIC: 49.3 μM). VP-4509 exhibits high antibacterial activity against the gram-negative bacterium Pseudomonas aeruginosa (ATCC9027). |
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T38102 |
Decatromicin B
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Others
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Decatromicin B is a bacterial metabolite that has been found in Actinomadura. It is active against Gram-positive bacteria, including several strains of S. aureus (MICs = 0.39-0.78 μg/ml), two strains of methicillin-resis... |
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T36892 |
4'-Acetyl Chrysomycin A
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Others
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4'-Acetyl chrysomycin A is a bacterial metabolite and derivative of chrysomycin A that has been found inStreptomycesand has antibacterial and anticancer activities.1It is active against strains of methicillin-resistantS.... |
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T80275 |
Lynronne-2
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Lynronne-2, an antimicrobial peptide, exhibits activity against Gram-positive bacteria, including methicillin-resistant MRSA strains (MIC: 32-256 μg/mL), and demonstrates effectiveness in combating P. aeruginosa infectio... |
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T79778 |
Anti-MRSA agent 8
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Others
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Anti-MRSA Agent 8 (Compound 7g), a derivative of DAPG, exhibits potent antibacterial properties by interacting with bacterial cell membranes and is useful for studying methicillin-resistant Staphylococcus aureus (MRSA) [... |
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T72141 |
Ceftobiprole medocaril sodium
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BAL5788 sodium |
Others
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Ceftobiprole medocaril sodium (BAL5788) is a parenteral prodrug of Ceftobiprole, a pyrrolidinone cephalosporin administered intravenously. As a broad-spectrum cephalosporin, Ceftobiprole exhibits high in vitro activity a... |
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T38009 |
Kocurin
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Others
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Kocurin is a thiazolyl peptide originally isolated fromK. palustrisand has antibiotic activity.1It is active against methicillin-resistantS. aureus(MRSA; MIC = 0.25 μg/ml), as well asB. subtilisandE. faeciumin a solid ag... |
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T60302 |
4,4'-Dicyanostilbene
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Others
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4,4'-Dicyanostilbene (compound 43) demonstrates potent antimalarial activity against the Dd2 strain, exhibiting an EC50 value of 27 nM, and exhibits in vivo efficacy against methicillin-resistant Staphylococcus aureus (M... |
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T83758 |
SAAP 148 TFA
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Synthetic Antimicrobial and Antibiofilm Peptide 148 |
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SAAP 148, an antimicrobial peptide, effectively combats various multidrug-resistant bacteria in vitro and, in vivo, reduces skin colony-forming units (CFUs) in mouse models of A. baumannii or methicillin-resistant S. aur... |
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T74269 |
Antibacterial agent 83
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Others
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Antibacterial agent 83 (compound 17h) exhibits strong antibacterial efficacy against diverse strains of vancomycin-resistant Enterococcus faecalis (VRE) and methicillin-resistant Staphylococcus aureus (MRSA), significant... |
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T80414 |
ASP-1
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ASP-1 is a potent antistaphylococcal peptide, exhibiting minimum inhibitory concentrations (MICs) ranging from 2 μg/mL to 64 μg/mL against both S. aureus and methicillin-resistant S. aureus (MRSA) [1]. |
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T36706 |
Bottromycin A2
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Others
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Bottromycin A2is an antibiotic originally isolated fromStreptomyces.1It blocks the binding of aminoacyl-tRNA to the A site of the 50S ribosome, inhibiting protein synthesis.2Bottromycin A2is active against clinical isola... |
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T71266 |
Omadacycline HCl
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Others
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Omadacycline, also known as PTK 0796 and Amadacyclin, is a novel first-in-class aminomethylcycline with potent activity against important skin and pneumonia pathogens, including community-acquired methicillin-resistant S... |
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T38314 |
Parvodicin Complex
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Others
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Parvodicin complex is a mixture of closely related lipophilic glycopeptides originally isolated from A. parvosata. The parvodicin complex has activity against Gram-positive bacteria (MICs = 0.8-12.5 μg/ml) including meth... |
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T35487 |
Anacardic Acid Diene
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Others
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Anacardic acid diene is a polyunsaturated form of anacardic acid that has been found in cashew nut shell liquid. It has antibacterial activity against methicillin resistant S. aureus (MRSA) and S. mutans (MICs = 12.5 and... |
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T36598 |
Enopeptin A
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Others
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Enopeptin A, originally isolated from a culture broth of Streptomyces sp. RK-1051, is a depsipeptide antibiotic that contains two unusual amino acids (N-methylalanine and 4-methylproline) and features a pentaenone side c... |
