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カタログ番号	製品名	別名	ターゲット
T7147	Valbenazine	NBI-98854	Monoamine Transporter
	Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.		Monoamine Transporter
T3280	Clodronate disodium tetrahydrate	clodronic acid disodium tetrahydrate,Disodium clodronate tetrahydrate,Clastoban,Clodronate disodium	IL Receptor , TNF
	Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.		IL Receptor , TNF
T7563	NBI-98782	(+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ	Monoamine Transporter
	NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)		Monoamine Transporter
T23409	FM4-64	SynaptoRedTM C2	Others
	FM4-64 (SynaptoRedTM C2) is a styryl dye that stains stably but does not fluoresce in aqueous solution.FM4-64 does not passively diffuse into the plasma membrane bilayer and must be actively transported across the membra...		Others
TP1429	VSV-G Peptide acetate(103425-05-4 free base)	VSV-G Peptide	Others
	VSV-G Peptide acetate(103425-05-4 free base) is a 11 amino acid peptide derived from the Vesicular Stomatitis viral glycoprotein.		Others
T13134	(+)-Tetrabenazine	(+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ	Monoamine Transporter
	(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1.		Monoamine Transporter
T22486	Vesamicol hydrochloride	(±)-AH5183 hydrochloride	AChR
	Vesamicol hydrochloride ((±)-AH5183 hydrochloride) is a acetylcholine transport inhibitor.		AChR
T7651	Rose Bengal sodium	Rose Bengal	Influenza Virus , Monoamine Transporter
	Rose Bengal sodium is a potent inhibitor of VGlut and vesicular monoamine transporter (VMAT) (Ki of 19 and 64 nM for VGlut andVMAT, respectively）		Influenza Virus , Monoamine Transporter
T3534	Tetrabenazine Racemate	Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE	Monoamine Transporter
	Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2). Tetrabenazine Racemate blocks neurotransmitter uptake into adrenergic storage vesicles and has been ...		Monoamine Transporter
T77549	Nurr1 agonist 2		Others
	Nurr1 agonist 2 is a Nurr1 agonist with an EC50 value of 0.07 μM. Nurr1 agonist 2 increases the mRNA expression of the Nurr1-regulated genes tyrosine hydroxylase (TH) and vesicular amino acid transporter 2 (VMAT2). Nurr1...		Others
T22781L	FFN 511 hydrochloride	FFN 511 hydrochloride(1004548-96-2 Free base)
	FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitters (FFNs) targeting neuronal vesicular monoamine transporter 2 (VMA T2).FFN 511 hydrochloride inhibits the binding of 5-hydroxytryptamine to VMA T2-containing ...
T0313	Evans blue	Direct Blue 53,C.I. 23860	GluR
	Evans blue (C.I. 23860) is an azo dye, inhibits L-glutamate uptake via the membrane-bound excitatory amino acid transporter (EAAT).		GluR
T36949	Niaprazine		5-HT Receptor , Adrenergic Receptor , Histamine Receptor
	Niaprazine is a histamine H1-receptor antagonist with marked sedative properties. Niaprazine has antihistamine and antiserotonin activities and can be used for sleep disorder research[1][2]. Niaprazine exhibits a low aff...		5-HT Receptor , Adrenergic Receptor , Histamine Receptor
T25750	Lobelane Hydrochloride
	Lobelane Hydrochloride is a vesicular monoamine transporter-2 (VMAT2) inhibitor.
T31791	FFN246 HCl	FFN 246,FFN246 hydrochloride,FFN246,FFN-246
	FFN246 is a fluorescent substrate for both the serotonin transporter and the vesicular monoamine transporter 2 (VMAT2).
T24941	VMAT2-IN-I HCl	VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride
	VMAT2-IN-I HCl is an inhibitor of vesicular monoamine transporter-2. It also has 15- fold greater affinity than GZ- 793A.
T31790	FFN200 dihydrochloride	FFN200 HCl,FFN200,FFN 200,FFN-200
	FFN200 is a vesicular monoamine transporter 2 (VMAT2) substrate that selectively traces monoamine exocytosis in both neuronal cell culture and brain tissue.
T70322	Valbenazine dihydrochloride
	Valbenazine dihydrochloride inhibits vesicular monoamine transporter 2 (VMAT2); used to treat tardive dyskinesia.
T12190	Trans (2,3)-Dihydrotetrabenazine	(2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine	Others
	Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).		Others
T22452	Valbenazine tosylate	NBI-98854	Monoamine Transporter
	Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).		Monoamine Transporter
T75768	VSV-G tag Peptide
	VSV-G Peptide is a 11 amino acid peptide derived from the Vesicular Stomatitis viral glycoprotein .
T39878	FFN270 hydrochloride	FFN270 hydrochloride
	FFN270 hydrochloride, a fluorescent tracer for norepinephrine and vesicular monoamine transporters, features dual resolved absorption/excitation peaks that vary with solvent pH (FFN270 ex: 320 nm or 365 nm, em: 475 nm). ...
T9300	DiPT
	DiPT is an agonist at the 5HT2A receptor and a partial agonist at the 5HT1A receptor, and inhibits the transport of 5-hydroxytryptamine transporter and vesicular monoamine transporter 2.
T78684	FFN246		5-HT Receptor
	FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and emission spectra at 392/427 nm, respectively. It serves to label...		5-HT Receptor
TP2191	VSV-G Peptide		Others
	VSV-G is a vesicular stomatitis virus G (VSV-G) protein fragment. VSV-G protein is commonly used in biomedical research to pseudotype retroviral and lentiviral vectors, conveying the ability to transduce a broad range of...		Others
T79758	BQZ-485		Apoptosis
	BQZ-485, a potent GDI2 inhibitor, interacts with Tyr245 to disrupt the native GDI2-Rab1A interaction. This disruption impedes vesicular transport from the endoplasmic reticulum (ER) to the Golgi apparatus, triggering sub...		Apoptosis
T36045	1a,1b-dihomo Prostaglandin E2	1a,1b-dihomo Prostaglandin E2
	1a,1b-dihomo Prostaglandin E2 (PGE2) is a rare polyunsaturated fatty acid first identified in extracts of sheep vesicular gland microsomes, known to contain COX, incubated with adrenic acid . 1a,1b-dihomo PGE2 has also b...
T36887	8(E),10(E),12(Z)-Octadecatrienoic Acid
	8(E),10(E),12(Z)-Octadecatrienoic acid is a conjugated polyunsaturated fatty acid (PUFA) that has been found inC. officinalisseed oil and has anticancer activity.1,2,3It inhibits the growth of Caco-2 cells when used at c...

Compounds

Valbenazine

T7147

Synonym: NBI-98854

Target: Monoamine Transporter

Clodronate disodium tetrahydrate

T3280

Synonym: clodronic acid disodium tetrahydrate,Disodium clodronate tetrahydrate,Clastoban,Clodronate disodium

Target: IL Receptor, TNF

NBI-98782

T7563

Synonym: (+)-α-Dihydrotetrabenazine,(+)-α-DHTBZ,(+)-DTBZ

Target: Monoamine Transporter

FM4-64

T23409

Synonym: SynaptoRedTM C2

Target: Others

VSV-G Peptide acetate(103425-05-4 free base)

TP1429

Synonym: VSV-G Peptide

Target: Others

(+)-Tetrabenazine

T13134

Synonym: (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ

Target: Monoamine Transporter

Vesamicol hydrochloride

T22486

Synonym: (±)-AH5183 hydrochloride

Target: Influenza Virus, Monoamine Transporter

Tetrabenazine Racemate

T3534

Synonym: Nitoman,Ro 1-9569 Racemate,Rubigen,TETRABENAZINE

Target: Monoamine Transporter

FFN 511 hydrochloride

T22781L

Synonym: FFN 511 hydrochloride(1004548-96-2 Free base)

Target:

Evans blue

T0313

Synonym: Direct Blue 53,C.I. 23860

Target: 5-HT Receptor, Adrenergic Receptor, Histamine Receptor

Lobelane Hydrochloride

Synonym: FFN 246,FFN246 hydrochloride,FFN246,FFN-246

Target:

VMAT2-IN-I HCl

T24941

Synonym: VMAT2 IN I Hydrochloride,VMAT2-IN-I Hydrochloride,VMAT2INI Hydrochloride

Target:

FFN200 dihydrochloride

T31790

Synonym: FFN200 HCl,FFN200,FFN 200,FFN-200

Target:

Valbenazine dihydrochloride

T70322

Synonym:

Target:

Trans (2,3)-Dihydrotetrabenazine

T12190

Synonym: (2R,3R,11bR)-rel-DHTBZ,(2R,3R,11bR)-rel-Dihydrotetrabenazine

Target: Monoamine Transporter

Synonym: FFN270 hydrochloride

Target: 5-HT Receptor

1a,1b-dihomo Prostaglandin E2

T36045

Synonym: 1a,1b-dihomo Prostaglandin E2

Target:

8(E),10(E),12(Z)-Octadecatrienoic Acid

T36887

Synonym:

Target:

カタログ番号	製品名	別名	ターゲット
T75570	Justicidin C
	Justicidin C, a lignan compound, exhibits potent antiviral properties, particularly against vesicular stomatitis virus, with minimal cytotoxicity observed in rabbit lung cells (RL-33) [1].

天然物製品

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPH-02004	RAB5C Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Protein transport. Probably involved in vesicular traffic. RAB5C Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 39.5 kDa and th...
TMPH-03381	Synaptoporin/SYNPR Protein, Rat, Recombinant (His)	Rat	E. coli
	Intrinsic membrane protein of small synaptic vesicles. Probable vesicular channel protein. Synaptoporin/SYNPR Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted mol...
TMPH-01254	DNM1 Protein, Human, Recombinant (His)	Human	E. coli
	Microtubule-associated force-producing protein involved in producing microtubule bundles and able to bind and hydrolyze GTP. Most probably involved in vesicular trafficking processes. Involved in receptor-mediated endocy...
TMPH-02127	SNX16 Protein, Human, Recombinant (His)	Human	E. coli
	May be involved in several stages of intracellular trafficking. Plays a role in protein transport from early to late endosomes. Plays a role in protein transport to the lysosome. Promotes degradation of EGFR after EGF si...
TMPH-01902	DDX60 Protein, Human, Recombinant (His)	Human	E. coli
	Positively regulates DDX58/RIG-I- and IFIH1/MDA5-dependent type I interferon and interferon inducible gene expression in response to viral infection. Binds ssRNA, dsRNA and dsDNA and can promote the binding of DDX58/RIG-...
TMPK-01234	LAMP5 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Lysosome-associated membrane protein 5 (LAMP5) is a mammalian ortholog of the Caenorhabditis elegans protein, UNC-46, which functions as a sorting factor to localize the vesicular GABA transporter UNC-47 to synaptic vesi...
TMPH-03399	VAMP2 Protein, Rat, Recombinant (His)	Rat	E. coli
	Involved in the targeting and/or fusion of transport vesicles to their target membrane. Major SNARE protein of synaptic vesicles which mediates fusion of synaptic vesicles to release neurotransmitters. Essential for fast...
TMPK-01233	LAMP5 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Lysosome-associated membrane protein 5 (LAMP5) is a mammalian ortholog of the Caenorhabditis elegans protein, UNC-46, which functions as a sorting factor to localize the vesicular GABA transporter UNC-47 to synaptic vesi...
TMPK-01161	LAMP5 Protein, Mouse, Recombinant (hFc)	Mouse	HEK293 Cells
	Lysosome-associated membrane protein 5 (LAMP5) is a mammalian ortholog of the Caenorhabditis elegans protein, UNC-46, which functions as a sorting factor to localize the vesicular GABA transporter UNC-47 to synaptic vesi...
TMPJ-00670	YKT6 Protein, Human, Recombinant (His)	Human	E. coli
	Synaptobrevin Homolog YKT6 (YKT6) is an enzyme that belongs to the Synaptobrevin family. YKT6 contains a longin domain and a v-SNARE coiled-coil homology domain. YKT6 is highly conserved from yeast to human and it can fu...
TMPY-03868	ARF5 Protein, Human, Recombinant (His)	Human	E. coli
	ARF5, also known as ADP-ribosylation factor 5, belongs to the small GTPase superfamily, Arf family. Members of this family stimulate the ADP-ribosyltransferase activity of cholera toxin and play a role in vesicular traff...
TMPY-03266	COL4A3BP Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	COL4A3BP is a member of the StarD2 subfamily. It contains a pleckstrin homology domain at its amino terminus and a START domain towards the end of the molecule. COL4A3BP has a lipid-binding domain that mediates intrac...
TMPK-00659	LAMP5 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	Lysosome-associated membrane protein 5 (LAMP5) is a mammalian ortholog of the Caenorhabditis elegans protein, UNC-46, which functions as a sorting factor to localize the vesicular GABA transporter UNC-47 to synaptic vesi...
TMPY-03796	ARF3 Protein, Human, Recombinant (His)	Human	E. coli
	ARF3, also known as ADP-ribosylation factor 3, belongs to the RAS superfamily. Members of this family include ARF1, ARF2, ARF3, ARF4, ARF5 and ARF6. ARF3 gene is a member of the human ARF gene family. These genes encode ...
TMPY-03854	TMED4 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	TMED4, also known as ERS25, belongs to the EMP24/GP25L family. TMED4 may play a role in the regulation of heat-shock response and apoptosis. It is involved in vesicular protein trafficking, mainly in the early secretory ...
TMPY-00342	TMED4 Protein, Human, Recombinant (mFc)	Human	HEK293 Cells
	TMED4, also known as ERS25, belongs to the EMP24/GP25L family. TMED4 may play a role in the regulation of heat-shock response and apoptosis. It is involved in vesicular protein trafficking, mainly in the early secretory ...
TMPJ-01311	EPT1 Protein, Human, Recombinant (GST)	Human	E. coli
	Ethanolaminephosphotransferase 1 (EPT1) is an enzyme that belongs to the CDP-Alcohol Phosphatidyltransferase Class-I Family. EPT1 is a Selenoprotein, which contains a Selenocysteine (Sec) residue at its active site. The ...
TMPY-06815	SYAP1 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Synapse-associated protein 1 (SYAP1), also known as PRO3113 and BSTA, belongs to the synapse-associated BSD domain family, featuring three α-helices and two conserved tryptophan and phenylalanine residues located at the ...
TMPH-03758	TSG101 Protein, Human, Recombinant (His & Myc & SUMO)	Human	E. coli
	Component of the ESCRT-I complex, a regulator of vesicular trafficking process. Binds to ubiquitinated cargo proteins and is required for the sorting of endocytic ubiquitinated cargos into multivesicular bodies (MVBs). M...
TMPY-03501	Optineurin Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	OPTN (Optineurin) is a Protein Coding gene. The Optineurin gene encodes the coiled-coil containing protein optineurin. Optineurin is a multifunctional adaptor protein intimately involved in various vesicular trafficking ...
TMPY-03616	NAPG Protein, Human, Recombinant (His)	Human	E. coli
	NAPG (NSF Attachment Protein Gamma, also known as gamma SNAP) is a Protein Coding gene. This gene encodes soluble NSF attachment protein gamma. The encoded protein mediates platelet exocytosis and controls the membrane f...
TMPY-02885	CD1B Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	CD1B contains 1 Ig-like (immunoglobulin-like) domain and belongs to the CD1 family. CD1 family members are transmembrane glycoproteins, which are structurally related to the major histocompatibility complex (MHC) protein...
TMPY-04422	Casein Kinase 1 gamma 2 Protein, Human, Recombinant (His)	Human	Baculovirus Insect Cells
	Casein kinase I gamma 2 isoform (CSNK1G2), a member of the large casein kinase I (CKI) subfamily, protein kinase superfamily. It may affect the development of brain, and associate with vesicular trafficking and neurotran...
TMPY-04566	CAMKV Protein, Human, Recombinant (His & GST)	Human	Baculovirus Insect Cells
	CaM kinase-like vesicle-associated protein, also known as CAMKV, is a peripheral membrane protein and Cytoplasmic vesicle membrane protein which belongs to theprotein kinase superfamily and CAMK Ser/Thr protein kinase...
TMPH-02855	PML Protein, Mouse, Recombinant (His & Myc)	Mouse	E. coli
	Functions via its association with PML-nuclear bodies (PML-NBs) in a wide range of important cellular processes, including tumor suppression, transcriptional regulation, apoptosis, senescence, DNA damage response, and vi...
TMPY-04455	PKC iota Protein, Human, Recombinant (GST)	Human	Baculovirus Insect Cells
	Protein kinase C iota type, also known as Atypical protein kinase C-lambda/iota, aPKC-lambda/iota and PRKCI, is a cytoplasm, membrane and nucleus protein which belongs to the protein kinase superfamily, AGC Ser/Thr prote...
TMPH-02873	RAB10 Protein, Mouse, Recombinant (His & SUMO)	Mouse	E. coli
	The small GTPases Rab are key regulators of intracellular membrane trafficking, from the formation of transport vesicles to their fusion with membranes. Rabs cycle between an inactive GDP-bound form and an active GTP-bou...
TMPH-01248	ADAR Protein, Human, Recombinant (His & SUMO)	Human	E. coli
	Catalyzes the hydrolytic deamination of adenosine to inosine in double-stranded RNA (dsRNA) referred to as A-to-I RNA editing. This may affect gene expression and function in a number of ways that include mRNA translatio...