Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 30,500 | |||
5 mg | 在庫あり | ¥ 75,500 | |||
10 mg | 在庫あり | ¥ 129,500 | |||
25 mg | 在庫あり | ¥ 204,500 | |||
50 mg | 在庫あり | ¥ 282,500 | |||
100 mg | 在庫あり | ¥ 383,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 83,500 |
説明 | AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain. |
In vitro | AZD1940 demonstrates high binding affinity towards the CB1 and CB2 receptors in humans, rats, and mice, exhibiting full agonism at both receptor types across these species[1]. |
In vivo | After given orally to human, the mean maximum plasma concentration (Cmax) for AZD1940 800 mg was 9.3 nmol/L . The mean concentration over post-dose eight hours for AZD1940 was 236 nmol.h/L[1]. |
別名 | UNII-0J0035E9FT, AZD-1940, AZD 1940 |
分子量 | 413.52 |
分子式 | C20H29F2N3O2S |
CAS No. | 881413-29-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 90.0 mg/mL (217.6 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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AZD1940 881413-29-2 GPCR/G Protein Cannabinoid Receptor UNII-0J0035E9FT AZD-1940 AZD 1940 Inhibitor inhibitor inhibit