Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively.
説明 | Almorexant (ACT 078573) is a potent and competitive dual orexin 1 receptor (OX1)/orexin 2 receptor (OX2) antagonist with Ki values of 1.3 and 0.17 nM for OX1 and OX2, respectively. |
ターゲット&IC50 | OX2:0.17 nM(ki), OX1:1.3 nM(ki) |
別名 | ACT 078573 |
分子量 | 512.56 |
分子式 | C29H31F3N2O3 |
CAS No. | 871224-64-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (87.79 mM)
You can also refer to dose conversion for different animals. 詳細
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Almorexant 871224-64-5 GPCR/G Protein Neuroscience OX Receptor pancreatic cancer Orexin Receptor (OX Receptor) Pancreatic ductal adenocarcinoma Cataplexy HCRT Receptor Inhibitor ACT078573 Apoptosis GPCR orexin Hypocretin Receptor Ca2+ channels narcolepsy Caspase HPAF-II cells ACT-078573 AsPC-1 cells Calcium Channel Ca channels hypocretin ACT 078573 inhibit PDAC inhibitor