Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).
説明 | Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM). |
ターゲット&IC50 | D2 receptor:0.49 nM , 5-HT1A receptor:2.6 nM, D3 receptor:0.085 nM |
別名 | RGH-188 |
分子量 | 427.41 |
分子式 | C21H32Cl2N4O |
CAS No. | 839712-12-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Slightly soluble
You can also refer to dose conversion for different animals. 詳細
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Cariprazine 839712-12-8 GPCR/G Protein Neuroscience 5-HT Receptor Dopamine Receptor RGH188 Inhibitor Serotonin Receptor RGH 188 inhibit RGH-188 5-hydroxytryptamine Receptor inhibitor