Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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10 mg | 在庫あり | ¥ 12,500 | |||
50 mg | 在庫あり | ¥ 17,500 | |||
100 mg | 在庫あり | ¥ 20,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 9,500 |
説明 | Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI). |
ターゲット&IC50 | DNA polymerase α:440 μM (IC50), DNA polymerase δ:>550 μM (IC50), HIV-1 RT:0.26 μM (IC50) |
In vitro | Delavirdine (mesylate) inhibits growth of clinical isolates of HIV-1 (ED50s = <0.005-0.69 μM). Delavirdine blocks replication of 25 primary HIV-1 isolates, including strains resistant to 3'-azido-2',3'-deoxythymidine (AZT) or 2',3'-dideoxyinosine, with a mean ED50 value of 0.066 μM. Delavirdine also inhibits growth of L. infantum promastigotes (IC50 = 26.1 μM)[1]. |
別名 | U 90152 (mesylate), BHAP-U 90152 (mesylate), Delavirdine (mesylate) |
分子量 | 552.67 |
分子式 | C23H32N6O6S2 |
CAS No. | 147221-93-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 40.3 mg/mL (72.92 mM)
You can also refer to dose conversion for different animals. 詳細
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Delavirdine mesylate 147221-93-0 Microbiology/Virology Proteases/Proteasome Reverse Transcriptase HIV Protease polymerase Inhibitor HIV U-90152 U 90152 (mesylate) DLV BHAP-U 90152 BHAP-U 90152 (mesylate) NNRTI inhibit AIDs HIV-1 RT U90152 Human immunodeficiency virus Delavirdine Delavirdine Mesylate U 90152 Delavirdine (mesylate) BHAP-U-90152 BHAP-U90152 inhibitor