Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 約6-8 週間 | ¥ 45,000 |
5 mg | 約6-8 週間 | ¥ 100,500 |
10 mg | 約6-8 週間 | ¥ 148,500 |
25 mg | 約6-8 週間 | ¥ 226,500 |
50 mg | 約6-8 週間 | ¥ 317,000 |
1 mL * 10 mM (in DMSO) | 約6-8 週間 | ¥ 102,000 |
ターゲット&IC50 | 5-HT2 receptor:1.14 nM (ki), 5-HT2 receptor:5.8 nM (in rat cortical membrane) |
別名 | SR-46349 |
分子量 | 328.38 |
分子式 | C19H21FN2O2 |
CAS No. | 130579-75-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (152.26 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Eplivanserin 130579-75-8 GPCR/G Protein Neuroscience 5-HT Receptor 5-hydroxytryptamine Receptor Serotonin Receptor 5-HT2A SR46349 SR 46349 oral dopamine Inhibitor SR-46349 inhibit release inhibitor