Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
50 mg | 在庫あり | ¥ 45,500 | |||
100 mg | 在庫あり | ¥ 68,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 13,500 |
説明 | Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM. |
ターゲット&IC50 | HIV-1:0.41 nM |
In vitro | At low concentrations (0.0003-10?μmol/l) indinavir acts as a positive allosteric modulator (EC50?=?0.021?μmol/l), whereas at concentrations greater than 10?μmol/l (30-100?μmol/l) indinavir acts as an inhibitor of the α7-nicotinic acetylcholine receptor. |
別名 | L735524 sulfate, MK-639 sulfate |
分子量 | 711.87 |
分子式 | C36H49N5O8S |
CAS No. | 157810-81-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (140.48 mM)
You can also refer to dose conversion for different animals. 詳細
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Indinavir sulfate 157810-81-6 Microbiology/Virology Proteases/Proteasome HIV Protease SARS-CoV Inhibitor MK639 L-735524 Sulfate L 735524 Huh7 Matrix metalloproteinases L-735524 L735524 sulfate PBMC MK 639 MMP MK-639 Indinavir Sulfate SARS coronavirus Apoptosis hepatocarcinomas L735524 L735524 Sulfate Human immunodeficiency virus MK-639 Sulfate Indinavir inhibit MK-639 sulfate CD4 T cells MK639 Sulfate MK 639 Sulfate HIV L 735524 Sulfate inhibitor