Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 20,000 | |||
5 mg | 在庫あり | ¥ 49,000 | |||
10 mg | 在庫あり | ¥ 68,500 | |||
25 mg | 在庫あり | ¥ 106,500 | |||
50 mg | 在庫あり | ¥ 136,000 | |||
100 mg | 在庫あり | ¥ 181,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 54,000 |
説明 | Nevanimibe hydrochloride (PD-132301 hydrochloride) is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM). |
ターゲット&IC50 | ACAT1:EC50 of 9 nM |
In vitro | In H295R human adrenocortical carcinoma cells, Nevanimibe hydrochloride(ATR-101 hydrochloride) decreases the formation of cholesteryl esters and increases FC levels, demonstrating potent inhibition of ACAT1 activity. Caspase-3/7 levels and terminal deoxynucleotidyl transferase 2'-deoxyuridine 5'-triphosphate nick end labeled-positive cells are increased by ATR-101 treatment, indicating activation of apoptosis[2]. |
別名 | PD-132301 hydrochloride, ATR101 hydrochloride |
分子量 | 458.08 |
分子式 | C27H40ClN3O |
CAS No. | 133825-81-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 41.67 mg/mL (90.97 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Nevanimibe hydrochloride 133825-81-7 Apoptosis Metabolism Acyltransferase cancer O-acyltransferase ATR-101 Hydrochloride acyl-CoA:cholesterol acyltransferase PD 132301 Hydrochloride acyl-coenzyme PD-132301 Diglyceride acyltransferase orally adrenocortical A:cholesterol mono- acylglycerol acyltransferase inhibit ATR101 Hydrochloride PD132301 Hydrochloride ATR 101 Hydrochloride PD 132301 PD-132301 Hydrochloride Nevanimibe Hydrochloride Nevanimibe ATR 101 PD132301 ATR-101 Diacylglycerol acyltransferase active ATR101 Inhibitor PD-132301 hydrochloride ATR101 hydrochloride inhibitor