Powder: -20°C for 3 years | In solvent: -80°C for 1 year
OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM).
説明 | OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM). OMDM-5 is a selective anandamide cellular uptake (ACU) inhibitor(Ki = 4.8 μM). |
ターゲット&IC50 | TRPV1:75 Nm(TRPV1), CB1:4.9 μM(Ki), ACU:4.8 μM(Ki) |
分子量 | 432.64 |
分子式 | C26H44N2O3 |
CAS No. | 616884-66-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 65 mg/ml (150.24 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
OMDM-5 616884-66-3 GPCR/G Protein Membrane transporter/Ion channel Metabolism Cannabinoid Receptor TRP/TRPV Channel Endogenous Metabolite fatty TRP Channel Transient receptor potential channels VR1 FAAH inhibit receptor Inhibitor CB1 vanilloid cells OMDM 5 type CB2 uptake RBL-2H3 acids OMDM5 cannabinoid inhibitor