Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Tetrahydrocannabivarin (CRM) is a neutral cannabis receptor subtype (CB1) receptor antagonist, it can increases neural responding to rewarding and aversive stimuli, this effect profile suggests therapeutic activity in obesity, perhaps with a lowered risk of depressive side effects. Tetrahydrocannabivarin exhibits anticonvulsant effects in a piriform cortical brain slice model of epileptiform activity.
パッケージサイズ | 在庫状況 | 単価(税別) |
---|---|---|
1 mg | 在庫あり | ¥ 268,500 |
5 mg | 在庫あり | ¥ 539,500 |
10 mg | 在庫あり | ¥ 727,500 |
25 mg | 在庫あり | ¥ 1,076,500 |
50 mg | 在庫あり | ¥ 1,457,500 |
100 mg | 在庫あり | ¥ 1,969,500 |
説明 | Tetrahydrocannabivarin (CRM) is a neutral cannabis receptor subtype (CB1) receptor antagonist, it can increases neural responding to rewarding and aversive stimuli, this effect profile suggests therapeutic activity in obesity, perhaps with a lowered risk of depressive side effects. Tetrahydrocannabivarin exhibits anticonvulsant effects in a piriform cortical brain slice model of epileptiform activity. |
In vitro | At 3-1000 nanomol (nM), THCV did not prevent electrically induced contractions of mouse isolated vas deferens; though, the amount of THCV in this range formed dextral shifts in the log concentration-response curves of WIN and anandamide for electrically evoked contractions. These changes were not convoyed by a reduction in the maximal effect of any agonist. Nevertheless, at 3 millimolar (mM), THCV did lessen the contractile reaction of the vas deferens in a CB1 receptor antagonist (SR141716)-independent way. Moreover, THCV looks like SR141716 antagonist, which at high quantities also cooperates with non-CB1 targets.[1]. |
植物由来 |
別名 | THCV, delta9-Tetrahydrocannabivarin, CRM, Tetrahydrocannavarin |
分子量 | 286.41 |
分子式 | C19H26O2 |
CAS No. | 31262-37-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: Slightly soluble
You can also refer to dose conversion for different animals. 詳細
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Tetrahydrocannabivarin 31262-37-0 GPCR/G Protein Cannabinoid Receptor THCV O-4394 inhibit THC-V Inhibitor O4394 delta9-Tetrahydrocannabivarin CRM O 4394 Tetrahydrocannavarin inhibitor