Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BAY-6035 is an inhibitor of SET and MYND domain-containing protein 3 (SMYD3). BAY-6035 has more than 100-fold selectivity over other histone methyltransferases.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 7,000 | |||
5 mg | 在庫あり | ¥ 18,500 | |||
10 mg | 在庫あり | ¥ 29,500 | |||
25 mg | 在庫あり | ¥ 60,500 | |||
50 mg | 在庫あり | ¥ 98,500 | |||
100 mg | 在庫あり | ¥ 147,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 20,500 |
説明 | BAY-6035 is an inhibitor of SET and MYND domain-containing protein 3 (SMYD3). BAY-6035 has more than 100-fold selectivity over other histone methyltransferases. |
ターゲット&IC50 | SMYD3:88 nM (IC50) |
In vitro | BAY-6035 inhibits methylation of MEKK2 peptide in a cell-free assay and in cells with IC50s of 88 and 70 nM, respectively[1]. |
分子量 | 396.48 |
分子式 | C22H28N4O3 |
CAS No. | 2247890-13-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (239.61 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BAY-6035 2247890-13-5 Chromatin/Epigenetic MAPK MEK Histone Methyltransferase BAY6035 inhibit MEKK2 BAY 6035 Inhibitor SMYD3 methylation inhibitor