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T37793 |
A2B receptor antagonist 2
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A2B receptor antagonist 2 |
Adenosine Receptor
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A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). |
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T10058 |
A2B receptor antagonist 1
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Adenosine Receptor
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A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist. |
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T77508 |
A2B receptor antagonist 2 hydrochloride
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Others
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A2B receptor antagonist 2 hydrochloride is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B). |
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T21389 |
Enprofylline
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Enprofilina,3-propylxanthine,3-n-Propylxanthine,Enprofyllinum |
Others
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Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sick... |
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T30696 |
Calonyctin A-2b
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DC-2b |
Others
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Calonyctin A-2b is one of two components of calonyctin A. |
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TMAZ-0236A |
Anti-GUCA2B Monoclonal Antibody-APC
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TMAZ-0236B |
Anti-GUCA2B Monoclonal Antibody-Biotin
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TMAZ-0236A6 |
Anti-GUCA2B Monoclonal Antibody-AF647
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TMAZ-0236P |
Anti-GUCA2B Monoclonal Antibody-PE
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TMAZ-0236 |
Anti-GUCA2B Monoclonal Antibody
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T23593 |
A2B57
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A 2 B 57,A-2-B-57 |
Others
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A2B57 is a selective SIRT2 inhibitor. |
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TMAZ-0236A5 |
Anti-GUCA2B Monoclonal Antibody-AF555
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TMAZ-0236A4 |
Anti-GUCA2B Monoclonal Antibody-AF488
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T8512 |
BAY-545
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Adenosine Receptor
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BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM). |
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T27629 |
ISAM-140
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ISAM140 |
Adenosine Receptor
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ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor. |
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T16136 |
MRS-1706
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Adenosine Receptor
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MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1, and A3 receptors respectively. MRS-1706 is an effective and selective adenosine A2B receptor inverse agonist. |
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T16140 |
MRS 1754
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Adenosine Receptor
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MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats. |
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T15418 |
GS-6201
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CVT-6883 |
Adenosine Receptor
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GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM. |
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T27800 |
LAS38096
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LAS 38096,LAS-38096 |
Adenosine Receptor
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LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient . |
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T14506 |
BAY 60-6583
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Others
,
Adenosine Receptor
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BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 receptors.BAY 60-6583 is cardioprotective in a model of myocardial... |
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T23201 |
PSB 1115
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Adenosine Receptor
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human A2B adenosine receptor antagonist |
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T9238 |
KI-7
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Adenosine Receptor
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KI-7 is an adenosine A2B receptor positive allosteric modulator. |
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T14944 |
CGS 15943
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PI3K
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Adenosine Receptor
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CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively. |
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T15715 |
LAS101057
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Adenosine Receptor
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LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma. |
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T23203 |
PSB-603
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PSB 603 |
Adenosine Receptor
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PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects. |
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T22234 |
Alloxazine
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Adenosine Receptor
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Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor. |
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T8613 |
1-Ethyl-6-aminouracil
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6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE |
Adenosine Receptor
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1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosine A2B receptors. |
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T6979 |
SCH 58261
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SCH58261 |
Adenosine Receptor
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SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a. |
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T2671 |
Regadenoson
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CVT-3146,Lexiscan |
Adenosine Receptor
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Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine re... |
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T22937 |
LUF 5834
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Others
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A2A and A2B adenosine receptor partial agonist |
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T26681 |
ATL802
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ATL 802,ATL-802 |
Others
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ATL802 is an adenosine A2B Receptor antagonist. |
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T23197 |
PSB 0788
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Others
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adenosine A2B receptor antagonist |
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T26680 |
ATL-801
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Others
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ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis. |
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T26621 |
AMP-579
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RPR100579,RPR 100579,AMP 579,RPR-100579 |
Others
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AMP-579 is an adenosine A1 receptor agonist. AMP-579 also acts as a A2b-adenosine receptor agonist in human 293 cells and rabbit hearts. |
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T84741 |
PSB-1115 potassium salt
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Others
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PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1]. |
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T62611 |
Adenosine receptor antagonist 2
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Others
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Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects. |
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T63856 |
M1069
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Others
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M1069 is a selective, orally active A2A/A2B diadenosine receptor antagonist that is more than 100-fold more selective than subtypes A1 and A3. M1069 antagonizes the immunosuppressive mechanisms induced by adenosine and e... |
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T69675 |
PSB-1901 free base
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Others
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PSB-1901 is a potent A2B Adenosine Receptor Antagonist with Picomolar Potency (Ki 0.0835 nM, KB 0.0598 nM, human A2BAR) with >10 000-fold selectivity versus all other AR subtypes. PSB-1901 was similarly potent and select... |
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T61850 |
Adenosine receptor inhibitor 1
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Others
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Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >100... |
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T83958 |
CELT-327
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Others
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CELT-327 is a potent, selective fluorescent hA2B/A3 adenosine receptor antagonist, exhibiting K_i values of 35.6 nM at A2B and 45.7 nM at A3 receptors. It efficiently labels HCT116 cells expressing A2B adenosine receptor... |
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T70421 |
VCP746
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Others
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VCP-746 is a potent adenosine A2B receptor agonist that stimulates anti-fibrotic signalling. VCP746 reduces hypertrophy in a rat neonatal cardiac myocyte model. VCP746 is a hybrid molecule consisting of an adenosine moie... |
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T62797 |
A2A receptor antagonist 3
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Others
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A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM). |
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T37669 |
CAY10498
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Others
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The A1, A2A, A2B, and A3 adenosine receptors (ARs) are ubiquitous G protein-coupled receptors. The four AR subtypes have been implicated in several areas of therapeutic interest such as stroke and other ischemic conditio... |
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T23202 |
PSB 36
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Others
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A1 adenosine receptor antagonist |
