|
T0865 |
Ranitidine Hydrochloride
|
AH19065 |
P450
,
Antibacterial
,
Histamine Receptor
|
|
Ranitidine Hydrochloride (AH19065) is a member of the class of histamine H2-receptor antagonists with antacid activity. Ranitidine is a competitive and reversible inhibitor of the action of histamine, released by enteroc... |
|
T3610 |
Ranitidine
|
HSDB 3925,Ranitidin |
P450
,
Antibacterial
,
Histamine Receptor
|
|
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors). It is used to treat gastrointestinal ulcers. |
|
T7524 |
Metiamide
|
SK&F 92058 |
Histamine Receptor
|
|
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist . |
|
T15195 |
Ebrotidine
|
FI3542 |
Histamine Receptor
|
|
Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a potent antisecretory activity and evidenced gastroprotection. |
|
T1575 |
Nizatidine
|
Axid,Acinon,Zanizal |
AChE
,
Histamine Receptor
|
|
Nizatidine (Acinon) is a competitive and reversible histamine H2-receptor antagonist with antacid activity. |
|
T0157 |
Roxatidine Acetate hydrochloride
|
HOE 760,Roxatidine Acetate HCl |
Histamine Receptor
|
|
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. It inhibits gastric acid secretion and ulcer formation. |
|
T31195 |
Dalcotidine
|
KU 1257,KU-1257 |
Histamine Receptor
|
|
Dalcotidine (KU 1257) is a novel histamine H2 receptor antagonist with histamine H9 receptor antagonistic activity and antisecretory effects.The Ki value for binding to guinea pig cerebral cortex was 0.040 The KB value f... |
|
T68056 |
Donetidine
|
|
Histamine Receptor
|
|
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders. |
|
T68122L |
Oxmetidine FA
|
Oxmetidine FA(72830-39-8 Free base) |
Histamine Receptor
|
|
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties. |
|
T22842 |
HTMT dimaleate
|
Histamine Trifluoromethyl Toluidide Dimaleate |
Histamine Receptor
|
|
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist. |
|
T68146 |
Sufotidine
|
AH 25352X,AH25352X,AH-25352X |
Histamine Receptor
|
|
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist. |
|
T68921 |
Impromidine hydrochloride
|
|
Histamine Receptor
|
|
Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies. |
|
T15005 |
CP-66948
|
|
Histamine Receptor
|
|
CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa. |
|
T68100 |
Mifentidine
|
DA 4577 |
Histamine Receptor
|
|
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers. |
|
T8599 |
Betazole dihydrochloride
|
Betazole hydrochloride |
Histamine Receptor
|
|
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor. |
|
T1627 |
Famotidine
|
MK-208 |
Histamine Receptor
|
|
Famotidine (MK-208) is a propanimidamide and histamine H2-receptor antagonist with antacid activity. As a competitive inhibitor of histamine H2-receptors located on the basolateral membrane of the parietal cell, famotidi... |
|
T11825 |
LCB-2853
|
|
PPAR
|
|
|
|
T22724 |
Dimaprit dihydrochloride
|
|
NOS
,
NO Synthase
,
Histamine Receptor
|
|
Dimaprit dihydrochloride is a selective histamine H2 receptor agonist. Dimaprit dihydrochloride also inhibits nNOS with an IC50 of 49 μM. It can stimulate gastric acid secretion. |
|
T10000 |
(±)-Tazifylline
|
|
Histamine Receptor
|
|
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor. Tazifylline shows much lower affinity for H2 receptors, α- and β-adrenoceptors, 5-hydroxytryptamine and muscarinic receptor subtypes. |
|
T68122 |
Oxmetidine
|
SKF 92994,Oxmetidina,Oxmetidinum |
Histamine Receptor
|
|
Oxmetidine (SKF 92994) is a novel H2 receptor antagonist that is cytotoxic. Oxmetidine inhibits transmembrane calcium flux in cardiac and vascular tissues and is used in the treatment of active duodenal ulcers. |
|
T2533 |
Alcaftadine
|
R89674,Lastacaft |
Histamine Receptor
|
|
Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis. |
|
T11324 |
FRG8701
|
|
Histamine Receptor
|
|
|
|
T13163 |
Tiotidine
|
ICI 125211 |
Others
|
|
|
|
T23565 |
Zolantidine dimaleate
|
|
Others
|
|
H2 receptor antagonist |
|
T22848 |
ICI 162,846
|
|
Others
|
|
histamine H2 receptor antagonist |
|
T70297 |
IY-80843
|
|
|
|
IY-80843 is an H2-receptor antagonist. |
|
T13382 |
Zaltidine
|
CP-57361 |
Others
|
|
Zaltidine is an antagonist of H2-receptor, and has the antisecretory action. |
|
T23942 |
DA 4626
|
DA4626,DA-4626 |
|
|
DA 4626 is H2-receptor antagonism. The compound which was investigated in a wider concentration range, behaved as simple competitive antagonists, yielding apparent KB values comparable with those estimated in conventiona... |
|
T23811 |
BMY-25368
|
BMY25368 |
|
|
BMY-25368 is a long-acting antagonist of the H2-receptor. |
|
T24162 |
Impromidine
|
Impromidina,Impromidinum |
|
|
Impromidine is a highly potent and specific agonist of the histamine H2 receptor. |
|
T71086 |
IT-066 HCl
|
|
|
|
IT-066 HCl is a histamine H2 receptor antagonist. |
|
T68747 |
Orf 17578
|
|
|
|
Orf 17578 is a histamine H2-receptor antagonist. |
|
T68479 |
Orf 17910
|
|
|
|
Orf 17910 is a histamine H2-receptor antagonist. |
|
T12228 |
Niperotidine
|
|
Histamine Receptor
|
|
Niperotidine is an antagonist of histamine H2-receptor. |
|
T28613 |
RP73870
|
RP 73870,RP-73870 |
|
|
RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity. |
|
T26039 |
Ramixotidine
|
|
|
|
Ramixotidine is a competitive antagonist of histamine H2-receptor. |
|
T10575 |
BMY-25271
|
|
Histamine Receptor
|
|
BMY-25271 is an antagonist of histamine H2 receptor. |
|
T23941 |
DA 4360
|
DA4360,DA-4360 |
|
|
DA 4360 is an H2-receptor antagonist. The compounds which were investigated in a wider concentration range, behaved as simple competitive antagonists, yielding apparent KB values comparable with those estimated in conven... |
|
T8439 |
Clobenpropit dihydrobromide
|
|
Apoptosis
,
Histamine Receptor
|
|
Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07) |
|
T71390 |
AY 29315
|
|
|
|
AY 29315 is a histamine H2-receptor antagonist with antisecretory and antiulcer activities. |
|
T23943 |
DA 4643
|
DA-4643,DA4643 |
|
|
DA 4643 is one of the histamine H2-receptor antagonists. Both mifentidine and DA 4643 interact with the histamine H2-receptor at the same site, utilizing in the binding process the same, or closely similar, receptor stru... |
|
T68704 |
Orf 17583
|
|
|
|
Orf 17583 is a histamine H2-receptor antagonist. |
|
T71529 |
NO 794
|
|
|
|
NO 794 is a histamine H2-receptor antagonist. |
|
T70709 |
FCE-27262
|
|
|
|
FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist. |
|
T15722 |
Lavoltidine
|
Loxtidine,AH-234844 |
Histamine Receptor
|
|
Lavoltidine is an orally active and irreversible histamine H2-receptor antagonist. Lavoltidine strongly suppresses gastric acid secretion and also induces hypergastrinemia. |
|
T71470 |
Famotidine hydrochloride
|
|
|
|
Famotidine hydrochloride is a competitive histamine H2-receptor antagonist. Its main pharmacodynamic effect is the inhibition of gastric secretion. |
|
T31743 |
Famotine hydrochloride
|
Famotine HCl,UK-2054 |
|
|
Famotine Hydrochloride is a histamine H2 receptor antagonist that suppresses acid production in the stomach and commonly treats peptic ulcer disease and gastroesophageal reflux disease. |
|
T71928 |
Nordimaprit dihydrochloride
|
|
|
|
Nordimaprit dihydrochloride is a metabolite of Dimaprit -- a histamine analog and selective H2 histamine receptor agonist. |
|
T35288 |
Z 300
|
Z-300,Z300 |
|
|
Z 300 is a histamine H2-receptor antagonist. Z 300 inhibits acid secretion and promotes gastric mucus metabolism in the corpus region. |
|
T70127 |
Famotine
|
|
|
|
Famotine is a histamine H2 receptor antagonist that inhibits stomach acid production. It is commonly used in the treatment of peptic ulcer disease and gastroesophageal reflux disease. |
