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T38565 |
Testosterone glucuronide
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Others
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Testosterone glucuronide is the major urinary metabolite of testosterone and is a potential urinary biomarker. |
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T37811 |
6-Chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt)
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Others
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6-Chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt) is a chromogenic substrate for β-glucuronidase. 6-Chloro-3-indolyl-β-D-Glucuronide (cyclohexylammonium salt) can be used in the histochemical analysis of β-glu... |
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T18887 |
4-Methylumbelliferyl-β-D-glucuronide hydrate
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MUG |
Others
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4-Methylumbelliferyl-β-D-glucuronide hydrate (MUG) is a fluorogenic substrat (λex=362 nm , λem=445 nm). |
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T125076 |
Hispidulin 7-glucuronide
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Hispidulin 7-glucuronide is a useful organic compound for research related to life sciences. The catalog number is T125076 and the CAS number is 31105-76-7. |
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T33284 |
Menthol glucuronide
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l-Menthyl glucuronide,l-Menthol glucuronide |
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Menthol glucuronide is a metabolite of L-(-)-Menthol, the natural form of Methanol. |
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T11253 |
Ezetimibe phenoxy glucuronide
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Ezetimibe β-D-glucuronide,Ezetimibe glucuronide |
Others
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Ezetimibe phenoxy glucuronide (Ezetimibe glucuronide) is the active metabolite of Ezetimibe. Antihyperlipoproteinemic activity. |
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T67690 |
PNPG-1
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4-Nitrophenyl β-D-glucuronide |
Others
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pNPG-1(4-Nitrophenyl β-D-glucuronide) is a glucuronide monosaccharide derivative that is a chromogenic substrate for β-glucosidase. |
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T80658 |
Quercetin 7-glucuronide
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Quercetin 7-O-β-glucuronide |
Drug Metabolite
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Quercetin 7-glucuronide (Quercetin 7-O-β-glucuronide), a Quercetin metabolite found in Madagascarian Uncarina species, has the capability to inhibit LDL oxidation [1]. |
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T11252 |
Ezetimibe phenoxy glucuronide-D4
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Ezetimibe β-D-glucuronide-D4,Ezetimibe glucuronide-D4 |
Others
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Ezetimibe phenoxy glucuronide-D4 (Ezetimibe glucuronide-D4) is the deuterium labeled Ezetimibe phenoxy glucuronide. |
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T37117 |
Etodolac Acyl Glucuronide
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Etodolac acyl glucuronide is a phase II metabolite of the non-steroidal anti-inflammatory drug (NSAID) and COX inhibitor etodolac .1It is formedviaglucuronidation of etodolac by the UDP-glucuronosyltransferase (UGT) isof... |
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T35440 |
(-)-Sitagliptin Carbamoyl Glucuronide
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(-)-Sitagliptin carbamoyl glucuronide is a minor phase II metabolite of the dipeptidyl peptidase 4 (DPP-4) inhibitor (-)-sitagliptin . (-)-Sitagliptin carbamoyl glucuronide is formed by N-carbamoyl glucuronidation and ha... |
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T71734 |
Muraglitazar glucuronide
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Muraglitazar glucuronide is a Peroxime Proliferator Activated (PPAR) Agonist that has glucose- and lipid-lowering activities. |
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T35621 |
Febuxostat Acyl Glucuronide
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Febuxostat acyl glucuronide is a metabolite of the xanthine oxidoreductase inhibitor febuxostat . Febuxostat acyl glucuronide is formed via glucuronidation of febuxostat by uridine diphosphate-glucuronosyltransferases (U... |
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T69267 |
Naproxen glucuronide
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Naproxen glucuronide is a nonsteroidal anti-inflammatory drug (NSAID) of the propionic acid class (the same class as ibuprofen) that relieves pain, fever, swelling, and stiffness. It is a nonselective COX inhibitor. |
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T37484 |
1-Salicylate Glucuronide
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1-Salicylate glucuronide is a metabolite of salicylic acid and aspirin .1It is formed from salicylic acid primarily by the UDP-glucuronosyltransferase (UGT) isoform UGT1A9 but also by a variety of other UGT isoforms and ... |
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T70560 |
Belinostat Glucuronide
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Belinostat Glucuronide is the major metabolite of Belinostat. Belinostat is a novel histone deacetylase 3 selective inhibitor that protects β cells from cytokine-induced apoptosis. |
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T35845 |
(R,S)-Carvedilol Glucuronide
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(R,S)-Carvedilol glucuronide is a racemic mixture of the carvedilol metabolites (R)-carvedilol glucuronide and (S)-carvedilol glucuronide. (R)-Carvedilol glucuronide is formed via glucuronidation of (R)-carvedilol by the... |
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T83873 |
Dabigatran Acyl-β-D-Glucuronide TFA
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Dabigatran β-1-O-Acyl Glucuronide |
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Dabigatran acyl-β-D-glucuronide, an active metabolite of the thrombin inhibitor dabigatran, is synthesized predominantly through the action of the UDP-glucuronosyltransferase isoform UGT2B15. This compound, at a concentr... |
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T37852 |
Chlorzoxazone N-Glucuronide
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Chlorzoxazone N-glucuronide is a phase II metabolite of the skeletal muscle relaxant chlorzoxazone . Chlorzoxazone N-glucuronide is formed via glucuronidation of chlorzoxazone by the UDP-glucuronosyltransferase (UGT) iso... |
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T71983 |
Zidovudine glucuronide
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Zidovudine glucuronide is an antiretroviral medication used to prevent and treat HIV/AIDS. It is of the nucleoside analog reverse-transcriptase inhibitor (NRTI) class. Zidovudine inhibits the enzyme (reverse transcriptas... |
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T11629 |
Ifenprodil glucuronide
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Others
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Ifenprodil glucuronide, a derivative of Ifenprodil, is a vasodilator and an inhibitor of platelet aggregation. In contrast to Ifenprodil, Ifenprodil glucuronide does not affect platelet aggregation nor arterial contracti... |
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T37378 |
Propofol β-D-Glucuronide
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Propofol β-D-glucuronide is a metabolite of propofol sulfate , a short-acting anesthetic agent. [1] [2] The metabolite is generated through the glucuronidation of propofol by uridine diphosphate glucuronosyltransferases.... |
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T12686 |
Raloxifene 4'-glucuronide
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Others
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Raloxifene 4'-glucuronide is a primary metabolite of Raloxifene. |
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T69838 |
NB-506 glucuronide
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NB-506 glucuronide is an indolocarbazole antitumor agent; a DNA topoisomerase I inhibitor. |
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T36128 |
Tolmetin β-D-Glucuronide
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Tolmetin β-D-Glucuronide has reactive properties with human serum albumin, allowing identification of the binding site and reaction mechanism by tandem mass spectrometry. |
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T36071 |
Silodosin Glucuronide (sodium salt)
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Silodosin glucuronide is an active metabolite of the α1A-adrenergic receptor antagonist silodosin . It is formed from silodosin by the UDP-glucuronosyltransferase (UGT) isoform UGT2B7. Silodosin glucuronide is toxic to r... |
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T36826 |
Acetaminophen Glucuronide (sodium salt)
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Acetaminophen glucuronide is an inactive metabolite of the analgesic and antipyretic agent acetaminophen . It is formed via glucuronidation of acetaminophen by the UDP-glucuronosyltransferase (UGT) isoforms UGT1A6, UGT1A... |
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T35952 |
All-trans Retinoyl β-D-Glucuronide
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all-trans Retinoyl β-D-glucuronide is a metabolite of all-trans retinoic acid formed by the UDP-glucuronosyltransferase (UGT) system. It is rapidly converted to all-trans retinoic acid following in vitro or in vivo admin... |
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T12688 |
Raloxifene 6-glucuronide
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Others
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Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8. |
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T35720 |
4’-hydroxy Atomoxetine Glucuronide (hydrate)
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4’-hydroxy Atomoxetine glucuronide is a metabolite of the norepinephrine transporter (NET) inhibitor atomoxetine .1It is formed from atomoxetine by glucuronidation of the intermediate metabolite 4-hydroxy atomoxetine.2
1... |
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T41022 |
β-D-glucuronide-pNP-carbonate
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β-D-glucuronide-pNP-carbonate is an ADC linker utilized in the synthesis of antibody-drug conjugates (ADCs). |
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T27121 |
Darexaban glucuronide
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YM 222714,YM222714,YM-222714 |
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Darexaban glucuronide is the major component in plasma after oral administration of darexaban to humans. Darexaban (YM150) is a direct inhibitor of factor Xa. |
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T36023 |
Formoterol O-β-D-Glucuronide
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Formoterol O-β-D-glucuronide is a metabolite of formoterol . |
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T35939 |
Dabigatran Acyl-β-D-Glucuronide
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Dabigatran acyl-β-D-glucuronide is a major active metabolite of the thrombin inhibitor dabigatran . The prodrug of dabigatran, dabigatran etexilate , is hydrolyzed by plasma esterases to form dabigatran, which is metabol... |
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T40557 |
Simvastatin Acyl-β-D-glucuronide
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Simvastatin Acyl-β-D-glucuronide, a metabolite formed from Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, showcasing a potent Ki of 0.2 nM. |
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T35865 |
Telmisartan Acyl-β-D-Glucuronide
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Telmisartan acyl-β-D-glucuronide is a major metabolite of the angiotensin II receptor antagonist telmisartan . It does not bind human serum albumin and is cleared from rat plasma with a clearance rate of 180 ml/min/kg fo... |
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T36794 |
Dolutegravir O-β-D-Glucuronide
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Dolutegravir O-β-D-glucuronide is a metabolite of the HIV integrase inhibitor dolutegravir .1It is formed from dolutegravir primarily by the UDP-glucuronosyltransferase (UGT) isoform UGT1A1in vivobut is also metabolized ... |
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T27167 |
Diclofenac Acyl Glucuronide
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Diclofenac Acyl Glucuronide is a major biliary metabolite of Diclofenac (GLXC-07892), a nonsteroidal antiinflammatory drug and COX inhibitor. |
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T37004 |
Estradiol 3-sulfate 17β-Glucuronide (potassium salt)
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Estradiol 3-sulfate is a sulfated form of the steroid hormone 17β-estradiol , and is common in fetal plasma and in the breast tissues of patients with mammary carcinoma. Sulfated estrogens, including estradiol 3-sulfate,... |
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T29009 |
Trifluoperazine N-Glucuronide
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Trifluoperazine N-Glucuronide is a metabolite of Trifluoperazine with antidepressant and antipsychotic activity. |
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T18231 |
MAC glucuronide linker-2
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Others
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MAC glucuronide linker-2 is an ADC linker employed in the synthesis of ADCs, offering cleavability [1]. |
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T18230 |
MAC glucuronide linker-1
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Others
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MAC glucuronide linker-1 is a nonclaevable ADC linker for antibody-drug-conjugations (ADCs). |
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T36518 |
Resveratrol-4'-O-D-Glucuronide
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Resveratrol-4'-O-D-Glucuronide has anti-fat accumulation properties, is metabolized by resveratrol, and can be used in metabolism-related studies. |
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T36917 |
Ethynyl Estradiol 3-β-D-Glucuronide (hydrate)
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Ethynyl estradiol 3-β-D-glucuronide is a metabolite of ethynyl estradiol that can be detected in urine.1,2It is used as a marker of estrogen contamination in fresh and saltwater.2
1.Hadd, H.E., Slikker, W., Jr., and Helt... |
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T35402 |
(±)-4-hydroxy Propranolol β-D-Glucuronide
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(±)-4-hydroxy Propranolol β-D-glucuronide is a metabolite of (±)-4-hydroxy propranolol , which is a metabolite of propranolol. The apparent half-life of (±)-4-hydroxy propranolol β-D-glucuronide is similar to propranolol... |
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T37251 |
Celecoxib Carboxylic Acid Acyl-β-D-Glucuronide
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Celecoxib carboxylic acid acyl-β-D-glucuronide is a phase II metabolite of celecoxib . Celecoxib is an anti-inflammatory compound from the diaryl heterocycle class that selectively inhibits cyclooxygenase-2 (COX-2; IC50s... |
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T37364 |
7-hydroxy Coumarin Glucuronide (sodium salt)
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7-hydroxy Coumarin glucuronide is a 7-hydroxy coumarin phase II metabolite that can be used as a standard for the analysis of 7-hydroxy coumarin metabolism. |
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T35619 |
Dapagliflozin-3-O-β-D-Glucuronide
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Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin . Dapagliflozin is a first generation selective sodium glucose cotransporter (SGLT) 2 inhibitor that blocks glucose transport.[1] Dapagliflozin is metab... |
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T36916 |
Estrone-3-Glucuronide (sodium salt hydrate)
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Estrone-3-Glucuronide is a metabolite of the primary premenopausal estrogen 17β-estradiol .1,2Urinary levels of estrone-3-Glucuronide peak approximately 36 hours prior to ovulation and have been used as a marker of ferti... |
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T37005 |
Estriol 3-β-D-Glucuronide (sodium salt)
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Estriol 3-β-D-glucuronide is a metabolite of estriol . It is formed from estriol by the UDP-glucuronosyltransferase (UGT) isoform UGT1A10. Estriol 3-β-D-glucuronide binds to basolateral and canalicular liver plasma membr... |
