Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
5 mg | 在庫あり | ¥ 9,000 | |||
10 mg | 在庫あり | ¥ 15,000 | |||
25 mg | 在庫あり | ¥ 30,500 | |||
50 mg | 在庫あり | ¥ 58,000 | |||
100 mg | 在庫あり | ¥ 91,000 | |||
500 mg | 在庫あり | ¥ 213,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 10,000 |
説明 | LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM). |
ターゲット&IC50 | FAAH:12.4 nM |
In vitro | LY2183240 increases brain anandamide concentration and exerts antinociceptive effects in the formalin model of pain, anandamide uptake Following i.p. administration in rats. |
分子量 | 307.35 |
分子式 | C17H17N5O |
CAS No. | 874902-19-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (162.68 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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LY2183240 874902-19-9 Autophagy Metabolism Neuroscience FAAH Inhibitor brain uptake transport hydrolases Fatty acid amide hydrolase LY 2183240 serine LY-2183240 anandamide inhibit inhibitor