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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T5117 | Hexaflumuron | Others | |
Hexaflumuron is a chitin synthesis inhibitor used to bait and eliminate termite colonies. Termites are unable to metabolize hexaflumuron and clearance is slow, resulting in up to 100% elimination. Hexaflumuron has also b... | |||
T20958 | Hexazinone | Others | |
Hexazinone is used as a broad spectrum herbicide. | |||
T8513 | Spastazoline | Others | |
Spastazoline is a potent and selective inhibitor of spastin(Human spastin with IC50 of 99 nM ). | |||
T14667 | BLT-1 | Others , HCV Protease | |
BLT-1 is a scavenger receptor BI (SR-BI)inhibitor. | |||
T10411 | AU1235 | Antibacterial | |
T8788 | Naptalam | Others | |
Naptalam is an herbicide.Naptalam is a dicarboxylic acid monoamide which results from addition of one equivalent of 1-naphthylamine to phthalic anhydride. It is a dicarboxylic acid monoamide, a carboxylic acid and a N-(1... | |||
T15802 | LY2183240 | FAAH , Autophagy | |
LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). LY2183240 is a novel and highly effective blocker of anandamide uptake (IC50 = 270 pM). | |||
T2298 | ML204 | TRP/TRPV Channel | |
ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels. | |||
T3171 | GSK137647A | GSK 137647 | GPR |
GSK137647A (GSK 137647) is a selective FFA4 agonist. | |||
T8616 | Fasentin | N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide | transporter |
Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1. | |||
T4405 | Ceftibuten dihydrate | Sch-39720 dihydrate | Antibacterial , Antibiotic |
Ceftibuten dihydrate (Sch-39720 dihydrate) is the dihydrate form of ceftibuten, and is a third-generation cephalosporin with antibacterial activity. | |||
T3088 | N-Ethylmaleimide | 1-Ethyl-1H-pyrrole-2,5-dione,Ethylmaleimide,NEM | Cysteine Protease , DUB |
N-Ethylmaleimide (NEM) is a sulfhydryl reagent that is widely used in experimental biochemical studies. | |||
T8936 | Proteinase K | proteinase K for tritirachium album,Protease K | Others |
Proteinase K (proteinase K for tritirachium album) is a nonspecific serine protease that is useful for general digestion of proteins. It is active in the presence of SDS or urea and over a wide range of pH (4-12), salt c... | |||
T3034 | Eprazinone dihydrochloride | Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl | Others , Neurokinin receptor |
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect. | |||
T22381 | Antimalarial agent 14 | 4-hydroxy-3-phenyl-naphthalene-1,2-dione,2-Hydroxy-3-phenyl-1,4-naphthoquinone | Others |
Antimalarial agent 14 (NSC-102533) is a bioactive chemical. | |||
T1244 | Celiprolol hydrochloride | Selecor,Selectrol | Adrenergic Receptor |
Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity. It is used in the management of ANGINA PECTORIS and HYPERTENSION. | |||
TP1849 | Transportan | ||
Transportan is a 27 amino acid-long peptide containing 12 functional amino acids from the amino terminus of the neuropeptide galanin and mastoparan in the carboxyl terminus, connected via a lysine. | |||
T81962 | Lactate transportor 1 | Monocarboxylate transporter | |
Lactate Transporter 1 (Compound 1) serves as an active lactate transporter within living cells and exerts cytotoxic effects, exhibiting IC50 values of 3.36 μM in HeLa, 3.27 μM in CAL27, 5.58 μM in MCF7, and 7.66 μM in MC... | |||
T6700 | Tenatoprazole | TU-199 | Proton pump |
Tenatoprazole (TU-199), a prodrug of the proton pump inhibitor (PPI) class, can inhibit proton transport (IC50: 3.2 μM). | |||
T22486 | Vesamicol hydrochloride | (±)-AH5183 hydrochloride | AChR |
Vesamicol hydrochloride ((±)-AH5183 hydrochloride) is a acetylcholine transport inhibitor. | |||
T11854 | Lipofermata | Others , Antibacterial | |
Lipofermata is a fatty acid transport protein (FATP) inhibitor that prevents lipid transport to melanoma cells and reduces melanoma growth and invasion. | |||
T20013 | Adamantanine | NSC 145160,NSC145160,NSC-145160 | Others |
Adamantanine (NSC-145160) is an amino acid transport inhibitor. | |||
T8940 | KUN56321 | 3H-Naphth[1,2-d]imidazole, 2-(4-bromophenyl)-3-phenyl- | Others |
KUN56321 (3H-Naphth[1,2-d]imidazole, 2-(4-bromophenyl)-3-phenyl-) is a luminescent agent. The application of KUN56321 comprises: coating the film of KUN56321 onto hole transport layer or electron transport layer of ITO g... | |||
T3445 | Importazole | Apoptosis , Others | |
Importazole is an inhibitor of the nuclear transport receptor importin-β. | |||
T19714 | Fenpyroximate | Others | |
Fenpyroximate is an acaricide and insecticide. It blocking the mitochondrial electron transport in complex I. | |||
T13134 | (+)-Tetrabenazine | (+)-TBZ,(3R,11bR)-Tetrabenazine,(3R,11bR)-TBZ | Monoamine Transporter |
(+)-Tetrabenazine ((3R,11bR)-Tetrabenazine) is a reversible vesicular monoamine transporter 2 (VMAT-2) inhibitor, inhibits transport by VMAT2 with 10-fold greater potency than transport by VMAT1. | |||
T77385 | Idactamab | INT-001 | |
Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2. | |||
T19060 | SPQ | Others | |
SPQ is used to measure membrane chloride transport mechanisms. | |||
T40515 | Metamitron | ||
Metamitron is a photosynthetic electron transport chain inhibitor and can be used as a chemical thinner. | |||
T9517 | Arprinocide | Others | |
Arprinocid is an inhibitor of hypoxanthine-guanine transport | |||
T34956 | Triplin | Others | |
Triplin is a chelator of copper ion. Triplin affects the transport of copper ions from ATX1 to RAN1. | |||
T20833 | Diflufenzopyr | SAN-835H,SAN835H,SAN 835H | Others |
Diflufenzopyr (SAN 835H), an auxin transport inhibitor, is semicarbazone-type. | |||
T10313 | AMXT-1501 tetrahydrochloride | Others | |
AMXT-1501 tetrahydrochloride is an inhibitor of polyamine transport. It blocks tumor growth in immunocompetent mice but not in athymic nude mice lacking T cells. | |||
T0502 | Zinc pyrithione | OM-1563 | Proton pump , Antibacterial , Antifungal |
Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump. | |||
T9897 | 7-Methoxy-1-naphthaleneacetic acid | Others | |
7-Methoxy-1-naphthaleneacetic acid is an inhibitor of auxin action in plants. 7-Methoxy-1-naphthaleneacetic acid inhibits polar auxin transport and tropic responses associated with asymmetric auxin distribution in Arabid... | |||
T40194 | MeAIB | α-(Methylamino)isobutyric acid | Others |
MeAIB is an N-acetyltransferase inhibitor that inhibits SNAT2-related signaling pathways. MeAIB is a specific substrate for amino acid transport system a (ATA1). Amino acid transport system a (ATA1) regulates the uptake ... | |||
T19783 | Dehydroabiethylamine | NSC-2955,NSC 2955,Dehydroabietylamine,NSC2955,Leelamine free base,Leelamine | P450 , PDK |
Dehydroabiethylamine (NSC-2955) is an inducer of hepatic CYP2B activity. Dehydroabiethylamine inhibits pyruvate dehydrogenase kinases (PDKs) and intracellular cholesterol transport with anti-tumor activity. | |||
T12038 | Migalastat hydrochloride | GR181413A hydrochloride,Migalastat HCl,GR181413A HCl | Others |
Migalastat hydrochloride (GR181413A) is an orally available, potent and competitive inhibitor of alpha-galactosidase A. It promotes the transport of alpha-galactosidase A to the lysosome and can be used in the study of F... | |||
T9372 | D-Histidine | Mitochondrial Metabolism | |
D-Histidine is an enantiomer of L-histidine. L-Histidine is an inhibitor of mitochondrial glutamine transport and also an essential amino acid for infants. | |||
T32873 | Maralixibat Chloride | SHP-625,SHP625,Livmarli,LUM001 chloride,Lopixibat chloride,Lopixibat,SHP625 chloride,SHP 625 | Potassium Channel |
Maralixibat Chloride (LUM001 chloride), an apical, sodium-dependent, bile acid transport inhibitor, prevents enterohepatic bile acid recirculation. | |||
T4172 | Methoxy-PMS | 1-Methoxyphenazine methosulfate,1-Methoxy PMS | Reactive Oxygen Species |
Methoxy-PMS (1-Methoxyphenazine methosulfate) is stable electron-transport mediator between NAD(P)H and tetrazolium dyes, can induce active oxygen formation. | |||
T77604 | WAY-326766 | CFTR | |
WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF). | |||
T16831 | (S)-SNAP5114 | Others , GABA Receptor | |
(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties. | |||
T2708 | SL327 | SL 327,SL-327 | MEK , DNA/RNA Synthesis |
SL327 is a selective inhibitor for MEK1/2 with IC50 of 0.18 μM/0.22 μM; able to transport through the blood-brain barrier. | |||
T8632 | Anthracene-9-carboxylic acid | Others | |
Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI. | |||
T17190 | U18666A | Others , HCV Protease | |
U18666A is a cell-permeable drug and is a cholesterol synthesis and transport inhibitor. It inhibits replication of Ebola virus, dengue virus, and human hepatitis C virus. | |||
T1768 | 7ACC2 | Mitochondrial Metabolism , Monocarboxylate transporter | |
7ACC2 is a new potent MCT inhibitor with IC50 of 11 nM for [14C]-lactate influx; new antitumor treatment targeting lactate transport in Y cells. | |||
T0719 | Tetrabenazine | Xenazine,Ro 1-9569 | Others , Dopamine Receptor , Monoamine Transporter |
Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrenergic storage vesicles and has been used as a high... | |||
T21483 | Tricaine methanesulfonate | MS-222 | Others |
Tricaine methanesulfonate (MS-222) (TMS) is an anesthetic. Many hatcheries and research studies use TMS to immobilize fish for marking or transport and to suppress sensory systems during invasive procedures. | |||
T2608 | CHIR-98014 | CHIR 98014,CT98014,CHIR98014 | FGFR , GSK-3 , Src , S6 Kinase |
CHIR-98014 (CT98014) is a selective GSK3 inhibitor; potentiate insulin activation of glucose transport and utilization in vitro and in vivo. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T9297 | Perseitol | Others | |
Perseitol is a sugar that is specific to avocado honey. Perseitol have recently been reported as candidate biomarkers for avocado intake. | |||
T8433 | HQNO | Mitochondrial Metabolism | |
HQNO is a natural product isolated from P. aeruginosa,and is a potent inhibitor of electron transport chain(Kd of 64 nM for complex III). It also is a potent mitochondrial NDH-2 inhibitorin many species. | |||
T21615 | Guanidinoethyl sulfonate | Taurocyamine | Chloride channel |
Guanidinoethyl sulfonate (Taurocyamine) is a competitive glycine receptor antagonist. | |||
T3S0156 | Atractyloside potassium salt | Atractyloside Dipotassium Salt | Others |
1. Atractyloside potassium salt (Atractyloside Dipotassium Salt) inhibits oxidative phosphorylation by blocking the transfer of adenosine nucleotides through the mitochondrial membrane. | |||
T5573 | Coenzyme Q9 | Ubiquinone Q9,Ubiquinone 9,CoQ9 | Apoptosis , Endogenous Metabolite |
Coenzyme Q9 (Ubiquinone 9) (CoQ9) is a normal constituent of human plasma. CoQ9 in human plasma may originate as a product of incomplete CoQ10 biosynthesis or from the diet. | |||
TN3150 | 6,8-Diprenylnaringenin | Senegalensin,Lonchocarpol A | BCRP , ABC |
T2911 | Stevioside | TLR | |
A natural, noncaloric sweetener with a potency 300 times more than that of regular sucrose. Exhibits transepithelial p-aminohippurate transport via organic anion transport system interference. | |||
T8170 | Carboxyatractyloside | Gummiferin,Carboxyatractyloside tripotassium salt | Others |
Carboxyatractyloside (Carboxyatractyloside tripotassium salt) is a natural product. It acts as an inhibitor of ADP/ATP carrier, inhibits mitochondrial ADP/ATP transport. | |||
T5300 | Ammonium formate | Formic acid ammonium salt | Others |
Ammonium formate (Formic acid ammonium salt) is the simplest carboxylic acid. Formate is an intermediate in normal metabolism. It is responsible for both metabolic acidosis and disrupting mitochondrial electron transport... | |||
T7975 | Rhodamine B | Rhodamine B,Tetraethylrhodamine,Brilliant Pink B,Basic Violet 1,Rhodamine O | Others |
Rhodamine B (Brilliant Pink B) is used as a tracer dye in water to determine the rate and direction of flow and transport. | |||
T21494 | Oligomycin | HIF | |
Oligomycin is an antifungal antibiotic that is an inhibitor of H+-ATP synthetase. The Oligomycin blocks oxidative phosphorylation and the electron transport chain. Oligomycin inhibited HIF-1alpha expression in hypoxic tu... | |||
T2S1120 | Ganoderenic acid B | P-gp | |
Ganoderenic acid B, a natural product derived from Ganoderma lucidum, can work by inhibiting the transport function of ABCB1 and enhancing the cytotoxicity of chemotherapy drugs against AbCB1-mediated multidrug resistant... | |||
T5068 | D-Glucuronic acid sodium salt monohydrate | Sodium D-glucuronate,D(+)-Glucuronic acid sodium salt monohydrate | Others , Endogenous Metabolite |
D-Glucuronic acid sodium salt monohydrate (Sodium D-glucuronate) is a carboxylic acid and highly soluble in water. In humans, glucuronic acid is often linked to toxic or poisonous substances to allow for subsequent elimi... | |||
T1045 | Trimipramine maleate | Surmontil maleate | Dopamine Receptor , 5-HT Receptor , Antibacterial , Adrenergic Receptor , Norepinephrine , Histamine Receptor |
Trimipramine maleate (Surmontil maleate) appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin and prolongs its action. Trimipramine Mal... | |||
TJS0928 | Calenduloside E | Silphioside F | Others |
Calenduloside E (Silphioside F) exhibits hypoglycemic activities by suppressing the transfer of glucose from the stomach to the small intestine and by inhibiting glucose transport at the brush border of the small intesti... | |||
T4927 | 4-Guanidinobutanoic acid | 4-GBA,4-Guanidinobutyric acid | Endogenous Metabolite |
4-Guanidinobutanoic acid (4-GBA) is an L-arginine metabolite that has been used in the intestinal transport tranport studies. It has been specifically use to human proton coupled amino acid transporters hPAT1. | |||
T3S0381 | Chrysophanol 8-O-glucoside | Serine Protease | |
Chrysophanol 8-O-glucoside and chrysophanol have mild cytotoxicity and anti-diabetic properties and can play metabolic roles in the insulin-stimulated glucose transport pathway | |||
T3S1775 | Tectochrysin | NSC 80687,Techtochrysine,Techtochrysin | NF-κB , STAT |
1. Tectochrysin (Techtochrysine) has antioxidant effect. 2. Tectochrysin is promising inhibitors for the reversal of ABCG2-mediated drug transport. 3. Tectochrysin leads to apoptotic cell death in NSC-LC cells through ac... | |||
T2970 | Rotenone | Rotenon,Paraderil,Barbasco,Rotocide,Dactinol | Apoptosis , Dehydrogenase , Mitochondrial Metabolism , p53 , Autophagy |
Rotenone (Rotocide) is a natural product and a botanical insecticide. Rotenone is a mitochondrial electron transport complex I inhibitor that promotes the production of reactive oxygen species in mitochondria and induces... | |||
TL0009 | Coniferin | Coniferoside,Abietin | Others , Antifungal |
Coniferin (Abietin) has ATP-dependent transport activity and has anti-oxidation effects. Coniferin has preferred substrates for the coniferin beta-glucosidase, the chromogenic coniferin analogue show the exclusive presen... | |||
T5291 | Malonic acid | Carboxyacetic Acid,1,3-Propanedioic Acid,Propanedioic Acid | Others |
Malonic acid (propanedioic acid) is the archetypal example of a competitive inhibitor: it acts against succinate dehydrogenase (complex II) in the respiratory electron transport chain. Malonic acid is found to be associa... | |||
T15245 | Erythromycin estolate | Phtalic anhydride,ilosone | Antibacterial |
Erythromycin estolate is a derivative of erythromycin, which belongs to the macrolide class of antibiotics and is often used to study a variety of bacterial infections. Erythromycin estolate has an inhibitory effect on b... | |||
T7285 | Ionomycin | Calcium Channel | |
Ionomycin is an calcium ionophore and an antibiotic that binds calcium ions (Ca2+). It is produced by the bacterium Streptomyces conglobatus.It is used in research to raise the intracellular calcium level (Ca2+) and as ... | |||
TJS0387 | Desoxyrhaponticin | Deoxyrhapontin,Deoxyrhaponticin | Apoptosis , Fatty Acid Synthase |
1. Desoxyrhaponticin (Deoxyrhaponticin) is an agent that is potentially effective in controlling postprandial hyperglycemia in diabetes, the in vivo antidiabetic action of this compound can be explained, in part at least... | |||
TN2496 | 1,4-Anthraquinone | Others | |
1,4-Anthraquinone is an anticancer drug that blocks nucleoside transport, inhibits macromolecule synthesis, induces DNA fragmentation, and decreases the growth and viability of L1210 leukemic cells in the same nanomolar ... | |||
T2924 | Phloretin | Dihydronaringenin,NSC 407292,RJC 02792 | SGLT , transporter , Endogenous Metabolite |
Phloretin (NSC-407292) is a well-known inhibitor of eukaryotic urea transporters, blocks VacA-mediated urea and ion transport. Phloretin is a dihydrochalcone, a type of natural phenols. It can be found in apple tree leav... | |||
T38805 | Euphol acetate | ||
Euphol acetate, a triterpene found in Euphorbia broteri, has demonstrated inhibitory effects on the hepatic transport proteins known as organic anion-transporting polypeptide 1/3 (OATP1B1/3). | |||
TN5114 | Taxinine | P-gp | |
Taxinine and Taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. | |||
TN4418 | Lasiodiplodin | ATPase , TNF | |
Lasiodiplodin may have potential anti-inflammatory activity, it shows moderate suppression effects on induced NO production. Lasiodiplodin inhibits electron transport chain. | |||
T38054 | Avenaciolide | ||
Avenaciolide is a water-insoluble fungal metabolite originally isolated from A. avenaceus. It inhibits glutamate transport in isolated rat liver mitochondria (Ki = 8 μM). | |||
T13490 | 25,26-Dihydroxyvitamin D3 | 25,26-Dihydroxycholecalciferol | Others |
25,26-Dihydroxyvitamin D3 is a metabolite of vitamin D3 with intestinal calcium transport activity. | |||
TN6565 | Maculosidin | ||
Maculosidine affect the PS I electron acceptors on leaf discs, it can inhibit ATP synthesis, basal, phosphorylating and uncoupled electron transport acting as Hill reaction inhibitors on spinach chloroplasts. | |||
T8303 | Cimicifugoside | Others | |
Cimicifugoside, a triterpenoid isolated from Cimicifuga simplex, is a novel specific nucleoside transport inhibitor. It also shows immunosuppressive activity. | |||
TN2301 | Vinleurosine | Others | |
Vinleurosine can partially inhibit the energy dependent transport of alpha-aminoisobutyric acid in Ehrlich ascites tumor cells. | |||
TN4749 | Pepluanin A | P-gp | |
Pepluanin A, shows a very high activity for a jatrophane diterpene, outperforming cyclosporin A by a factor of at least 2 in the inhibition of Pgp-mediated daunomycin transport. | |||
T17037 | Tenuazonic acid | Others | |
Tenuazonic acid is a putative nonhost-selective mycotoxin isolated from Alternaria alternate. Tenuazonic acid blocks electron transport beyond primary quinone acceptor (QA) by interacting with D1 protein and it is a broa... | |||
TN1387 | Angelol B | Others | |
The absorption and transport of angelol A and Angelol B are passive diffusion as the dominating process in Caco-2 cell monolayer model. | |||
T33342L | Methyl reserpate | NSC81464,NSC 81464,NSC-81464,Me reserpate | Norepinephrine |
Methyl reserpate (NSC 81464), a yohimbine-type alkaloid derived from the roots and leaves of Rauwolfia vomitoria, inhibits the transport of norepinephrine into chromophobe vesicles. | |||
TN5113 | Taxinine B | Others | |
Taxinine and taxinine B can inhibit the drug transport by P-glycoprotein in multidrug-resistant cells. Taxinine B shows stronger inhibitory effects than acetylsalicylic acid (ASA) on platelet aggregation induced by arach... | |||
T81158 | Siderin | ||
Siderin, a Photosystem II inhibitor, effectively impedes ATP synthesis and chloroplast electron transport in photosynthesis within isolated spinach chloroplasts and is utilized in research on plant photosynthesis [1]. | |||
T74293 | Allolithocholic acid | ||
Allolithocholic acid, a steroid acid present in normal serum and feces, aids in the excretion, absorption, and transport of fats and sterols within the intestine and liver [1]. | |||
T75699 | Coenzyme Q6 | ||
Coenzyme Q6 (Ubiquinone 30), an isoprenylated benzoquinone lipid, plays a pivotal role in respiratory electron transport and acts as a lipid antioxidant. Besides, it possesses antioxidant properties that inhibit the gene... | |||
T72172 | 4,6-O-Ethylidene-α-D-glucose | Ethylidene-glucose | |
4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucose transporter 1 (GLUT1), exhibiting a Ki of 12 mM against wild-type 2-... | |||
T75665 | 3-O-Methylellagic acid | ||
3-O-Methylellagic acid, a natural product isolated from Myrciaria cauliflora, exhibits anti-inflammatory and antibacterial activities. This compound not only inhibits glucose transport but also demonstrates a minimum inh... | |||
TN2945 | 3-Hydroxybakuchiol | ATPase , Caspase | |
3-Hydroxybakuchiol exerts cytotoxic and anti-proliferative effects on the TA3/Ha mouse mammary adenocarcinoma cell line and induces a decrease in the mitochondrial transmembrane potential, the activation of caspase-3, th... | |||
T82822 | Brassicanate A sulfoxide | ||
Brassicanate A sulfoxide, isolated from Brassica oleracea [1], exhibits herbicidal properties by inhibiting the biosynthesis of essential amino acids in plants. It operates by binding to key enzymes such as dihydroxyacid... | |||
T37810 | 6',7'-Epoxybergamottin | ||
6'7'-Epoxybergamottin is a furanocoumarin found in grapefruit. It is a potent inhibitor of the cytochrome P450 (CYP) isoform CYP3A4 with an IC50 value of 0.30 ppm in a cell-free assay, 0.33 μM in HL7 human liver cells, a... | |||
T36563 | (E)-Guggulsterone | ||
Bile acids are essential for solubilization and transport of dietary lipids, are the major products of cholesterol catabolism, and are physiological ligands for farnesoid X receptor (FXR), a nuclear receptor that regulat... |
カタログ番号 | 製品名 | Species | Expression System |
---|---|---|---|
TMPY-04861 | TMED1 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 Cells |
TMED1 Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46 kDa and the accession number is B2RRM5. | |||
TMPY-03119 | TMED1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TMED1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 20.6 kDa and the accession number is Q13445. | |||
TMPY-03108 | TMED1 Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
TMED1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 46.2 kDa and the accession number is Q13445. | |||
TMPY-03854 | TMED4 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
TMED4, also known as ERS25, belongs to the EMP24/GP25L family. TMED4 may play a role in the regulation of heat-shock response and apoptosis. It is involved in vesicular protein trafficking, mainly in the early secretory ... | |||
TMPY-00342 | TMED4 Protein, Human, Recombinant (mFc) | Human | HEK293 Cells |
TMED4, also known as ERS25, belongs to the EMP24/GP25L family. TMED4 may play a role in the regulation of heat-shock response and apoptosis. It is involved in vesicular protein trafficking, mainly in the early secretory ... | |||
TMPY-04072 | VTI1A Protein, Human, Recombinant (His) | Human | HEK293 Cells |
VTI1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 24.2 kDa and the accession number is Q96AJ9-2. | |||
TMPY-00526 | VTI1A Protein, Human, Recombinant (mFc) | Human | HEK293 Cells |
VTI1A Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 48.5 kDa and the accession number is Q96AJ9-2. | |||
TMPH-03432 | ACC1 Protein, S. cerevisiae, Recombinant (aa 2-581, His) | Saccharomyces cerevisiae | E. coli |
Carries out three functions: biotin carboxyl carrier protein, biotin carboxylase and carboxyltransferase. Involved in the synthesis of very-long-chain fatty acid synthesis which is required to maintain a functional nucle... | |||
TMPH-03431 | ACC1 Protein, S. cerevisiae, Recombinant (aa 217-775, His) | Saccharomyces cerevisiae | E. coli |
Carries out three functions: biotin carboxyl carrier protein, biotin carboxylase and carboxyltransferase. Involved in the synthesis of very-long-chain fatty acid synthesis which is required to maintain a functional nucle... | |||
TMPH-01136 | COG5 Protein, Human, Recombinant (His) | Human | E. coli |
COG5 Protein, Human, Recombinant (His) is expressed in E. coli. | |||
TMPJ-00999 | UBE2D1 Protein, Human, Recombinant (GST) | Human | E. coli |
Ubiquitin-conjugating enzyme E2 D1(UBE2D1)belongs to the ubiquitin-conjugating enzyme family. Ubiquitination involves at least three classes of enzymes: ubiquitin-activating enzymes, or E1s, ubiquitin-conjugating enzymes... | |||
TMPH-00206 | Pertactin autotransporter Protein, Bordetella pertussis, Recombinant (His & SUMO) | Bordetella pertussis | E. coli |
Agglutinogen that binds to eukaryotic cells; a process mediated by the R-G-D sequence. Pertactin may have a role in bacterial adhesion, and thus play a role in virulence. May contribute to the disease state of whooping c... | |||
TMPY-02956 | Apolipoprotein L/APOL1 Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
APOL1, also known as apolipoprotein L1, is a minor apoprotein component of HDL (High-density lipoprotein) or 'good cholesterol' which is synthesized in the liver and also in many other tissues, including pancreas, kidney... | |||
TMPY-03221 | Intrinsic Factor Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Gastric intrinsic factor, also known as GIF, belongs to the of the cobalamin transport protein family. It is a glycoprotein produced by the parietal cells of the stomach. Gastric intrinsic factor plays a key role in the ... | |||
TMPY-04329 | Vimentin Protein, Human, Recombinant (His) | Human | Baculovirus Insect Cells |
Vimentin is a type III intermediate filament (IF) protein found in various non-epithelial cells, especially mesenchymal cells. A vimentin monomer, has a central α-helical domain and carboxyl (tail) domains. Two monomers ... | |||
TMPH-02127 | SNX16 Protein, Human, Recombinant (His) | Human | E. coli |
May be involved in several stages of intracellular trafficking. Plays a role in protein transport from early to late endosomes. Plays a role in protein transport to the lysosome. Promotes degradation of EGFR after EGF si... | |||
TMPY-00490 | RAB6A Protein, Human, Recombinant (His) | Human | E. coli |
Rab6 is one of the most conserved Rab GTPaes throughout evolution and the most abundant Rab protein associated with the Golgi complex. The two ubiquitous Rab isoforms, Rab6A and Rab6A', that are generated by alternative ... | |||
TMPH-01300 | Stomatin/STOM Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Regulates ion channel activity and transmembrane ion transport. Regulates ASIC2 and ASIC3 channel activity. | |||
TMPH-02313 | RPGR Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Could be a guanine-nucleotide releasing factor. Plays a role in ciliogenesis. Probably regulates cilia formation by regulating actin stress filaments and cell contractility. Plays an important role in photoreceptor integ... | |||
TMPH-03641 | TroA Protein, Treponema pallidum, Recombinant (His & Myc) | Treponema pallidum | E. coli |
Part of an ATP-driven transport system TroABCD for zinc. Substrate-binding protein involved in the transport of zinc across the cytoplasmic membrane. TroA Protein, Treponema pallidum, Recombinant (His & Myc) is expressed... | |||
TMPH-02517 | APOD Protein, Mouse, Recombinant (His & Myc) | Mouse | E. coli |
APOD occurs in the macromolecular complex with lecithin-transport and binding of bilin. Appears to be able to transport a variety of ligands in a number of different contexts. APOD Protein, Mouse, Recombinant (His & Myc)... | |||
TMPH-00645 | Lactose permease Protein, E. coli, Recombinant (His) | E. coli | E. coli |
Responsible for transport of beta-galactosides into the cell, with the concomitant import of a proton (symport system). Can transport lactose, melibiose, lactulose or the analog methyl-1-thio-beta,D-galactopyranoside (TM... | |||
TMPH-03371 | Transferrin Protein, Rat, Recombinant (His & KSI) | Rat | E. coli |
Transferrins are iron binding transport proteins which can bind two Fe(3+) ions in association with the binding of an anion, usually bicarbonate. It is responsible for the transport of iron from sites of absorption and h... | |||
TMPH-02164 | Syntaxin-11 Protein, Human, Recombinant (GST) | Human | E. coli |
SNARE that acts to regulate protein transport between late endosomes and the trans-Golgi network. | |||
TMPH-01424 | GUCA2B Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Endogenous activator of intestinal guanylate cyclase. It stimulates this enzyme through the same receptor binding region as the heat-stable enterotoxins. May be a potent physiological regulator of intestinal fluid and el... | |||
TMPH-03589 | PsaA Protein, S. oralis, Recombinant (His & Myc) | Streptococcus oralis | E. coli |
Part of an ATP-driven transport system. PsaA Protein, S. oralis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 40.1 kDa and the accession... | |||
TMPH-01744 | NOX1 Protein, Human, Recombinant (His) | Human | E. coli |
NOH-1S is a voltage-gated proton channel that mediates the H(+) currents of resting phagocytes and other tissues. It participates in the regulation of cellular pH and is blocked by zinc. NOH-1L is a pyridine nucleotide-d... | |||
TMPH-02123 | SLC2A9 Protein, Human, Recombinant (His) | Human | E. coli |
Urate transporter, which may play a role in the urate reabsorption by proximal tubules. Does not transport glucose, fructose or galactose. | |||
TMPJ-00670 | YKT6 Protein, Human, Recombinant (His) | Human | E. coli |
Synaptobrevin Homolog YKT6 (YKT6) is an enzyme that belongs to the Synaptobrevin family. YKT6 contains a longin domain and a v-SNARE coiled-coil homology domain. YKT6 is highly conserved from yeast to human and it can fu... | |||
TMPH-03291 | FABP3 Protein, Rat, Recombinant (His & Myc) | Rat | HEK293 Cells |
FABP are thought to play a role in the intracellular transport of long-chain fatty acids and their acyl-CoA esters. | |||
TMPH-02873 | RAB10 Protein, Mouse, Recombinant (His & SUMO) | Mouse | E. coli |
The small GTPases Rab are key regulators of intracellular membrane trafficking, from the formation of transport vesicles to their fusion with membranes. Rabs cycle between an inactive GDP-bound form and an active GTP-bou... | |||
TMPH-02125 | SLCO2B1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
Mediates the Na(+)-independent transport of organic anions such as taurocholate, the prostaglandins PGD2, PGE1, PGE2, leukotriene C4, thromboxane B2 and iloprost. | |||
TMPH-03590 | PsaA Protein, S. pneumoniae (strain ATCC BAA-255/R6), Recombinant (His & Myc) | Streptococcus pneumoniae | E. coli |
Part of an ATP-driven transport system. PsaA Protein, S. pneumoniae (strain ATCC BAA-255/R6), Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight ... | |||
TMPY-03857 | MMGT1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
MMGT1 (Membrane Magnesium Transporter 1, also known as EMC5 and TMEM32) is a Protein Coding gene. 2 alternatively spliced human isoforms have been reported. The encoded protein belongs to the membrane magnesium transport... | |||
TMPH-01257 | Dystonin Protein, Human, Recombinant (His) | Human | P. pastoris (Yeast) |
Cytoskeletal linker protein. Acts as an integrator of intermediate filaments, actin and microtubule cytoskeleton networks. Required for anchoring either intermediate filaments to the actin cytoskeleton in neural and musc... | |||
TMPH-01256 | Dystonin Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Cytoskeletal linker protein. Acts as an integrator of intermediate filaments, actin and microtubule cytoskeleton networks. Required for anchoring either intermediate filaments to the actin cytoskeleton in neural and musc... | |||
TMPH-02004 | RAB5C Protein, Human, Recombinant (His & SUMO) | Human | E. coli |
Protein transport. Probably involved in vesicular traffic. RAB5C Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 39.5 kDa and th... | |||
TMPH-00707 | OppA Protein, E. coli, Recombinant (His & Myc) | E. coli | E. coli |
This protein is a component of the oligopeptide permease, a binding protein-dependent transport system, it binds peptides up to five amino acids long with high affinity. | |||
TMPH-00786 | BtuD Protein, Halobacterium salinarum, Recombinant (His) | Halobacterium salinarum | E. coli |
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system. | |||
TMPH-00787 | BtuD Protein, Halobacterium salinarum, Recombinant | Halobacterium salinarum | E. coli |
Required for corrinoid utilization. Probably part of the ABC transporter complex BtuCDF involved in cobalamin (vitamin B12) import. Probably responsible for energy coupling to the transport system. | |||
TMPH-03128 | TSPO Protein, Pig, Recombinant (His & Myc & SUMO) | Sus scrofa (Pig) | E. coli |
Promotes the transport of cholesterol across mitochondrial membranes and may play a role in lipid metabolism, but its precise physiological role is controversial. It is apparently not required for steroid hormone biosynt... | |||
TMPH-02573 | WISP3/CCN6 Protein, Mouse, Recombinant (His) | Mouse | E. coli |
Plays a role in mitochondrial electron transport and mitochondrial respiration. WISP3/CCN6 Protein, Mouse, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 4... | |||
TMPH-01592 | KIF18B Protein, Human, Recombinant (His & Myc) | Human | E. coli |
In complex with KIF2C, constitutes the major microtubule plus-end depolymerizing activity in mitotic cells. Its major role may be to transport KIF2C and/or MAPRE1 along microtubules. | |||
TMPH-02334 | RAB12 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
The small GTPases Rab are key regulators of intracellular membrane trafficking, from the formation of transport vesicles to their fusion with membranes. Rabs cycle between an inactive GDP-bound form and an active GTP-bou... | |||
TMPH-01009 | RHD Protein, Human, Recombinant (GST & His) | Human | E. coli |
May be part of an oligomeric complex which is likely to have a transport or channel function in the erythrocyte membrane. RHD Protein, Human, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis... | |||
TMPH-00831 | PMP2 Protein, Horse, Recombinant (His & SUMO) | Horse | E. coli |
May play a role in lipid transport protein in Schwann cells. May bind cholesterol. PMP2 Protein, Horse, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular we... | |||
TMPH-02122 | SLC2A1 Protein, Human, Recombinant (His & Myc) | Human | E. coli |
Facilitative glucose transporter, which is responsible for constitutive or basal glucose uptake. Has a very broad substrate specificity; can transport a wide range of aldoses including both pentoses and hexoses. Most imp... | |||
TMPH-03643 | TmpB Protein, Treponema phagedenis, Recombinant (His & Myc) | Treponema phagedenis | E. coli |
Tmp may serve as a porin or transport protein for large molecules. TmpB Protein, Treponema phagedenis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecula... | |||
TMPH-01434 | Hemoglobin subunit delta/HBD Protein, Human, Recombinant (GST & His) | Human | E. coli |
Involved in oxygen transport from the lung to the various peripheral tissues. Hemoglobin subunit delta/HBD Protein, Human, Recombinant (GST & His) is expressed in E. coli expression system with N-6xHis-GST tag. The predi... | |||
TMPH-03373 | SLC2A1 Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
Facilitative glucose transporter, which is responsible for constitutive or basal glucose uptake. Has a very broad substrate specificity; can transport a wide range of aldoses including both pentoses and hexoses. Most imp... | |||
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カタログ番号 | 製品名 | ||
---|---|---|---|
L7400 | Sodium Channel Blocker Library | 118 compounds | |
A unique collection of 118 sodium channel blockers and agonists for high throughput and high content screening; | |||
L9420 | Exosome Compound Library | 76 compounds | |
76 exosome-related compounds that can be used for high-throughput and high-content screening. |