Powder: -20°C for 3 years | In solvent: -80°C for 1 year
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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1 mg | 在庫あり | ¥ 18,500 | |||
5 mg | 在庫あり | ¥ 38,000 | |||
10 mg | 在庫あり | ¥ 54,000 | |||
25 mg | 在庫あり | ¥ 96,500 | |||
50 mg | 在庫あり | ¥ 137,500 | |||
100 mg | 在庫あり | ¥ 196,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 38,500 |
説明 | S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors. |
キナーゼ試験 | PI3K inhibition by LY294002 is determined in a radiometric assay using purified, recombinant enzymes with 1 μM ATP. The kinase reaction is carried out for 1 hour at room temperature (24oC) and is terminated by addition of PBS. IC50 values are subsequently determined using a sigmoidal dose-response curve fit (variable slope). CK2 and GSK3β (glycogen synthase kinase 3β) inhibition are established by kinase selectivity screening. LY294002 is tested against the Upstate panel of kinases in 10 μM ATP.[4] |
分子量 | 324.85 |
分子式 | C17H25ClN2O2 |
CAS No. | 1222097-72-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (76.96 mM)
You can also refer to dose conversion for different animals. 詳細
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S 38093 HCl 1222097-72-4 GPCR/G Protein Immunology/Inflammation Neuroscience Histamine Receptor Inhibitor inhibitor inhibit