Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 14,000 | |||
5 mg | 在庫あり | ¥ 34,000 | |||
10 mg | 在庫あり | ¥ 54,500 | |||
25 mg | 在庫あり | ¥ 109,500 | |||
50 mg | 在庫あり | ¥ 158,500 | |||
100 mg | 在庫あり | ¥ 225,500 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 37,500 |
説明 | Tonapofylline is an orally active and selective antagonist of the A1 adenosine receptor (Ki: 7.4 nM for human A1). Tonapofylline can be used in studies about heart failure. |
ターゲット&IC50 | A1 receptor (human):(ki)7.4 nM |
In vivo | Tonapofylline (1 mg/kg; p.o.) sustainably reduces the levels of post-Cisplatin serum creatinine and blood urea nitrogen and improves body weight recovery and significant attenuation of Cisplatin-induced (5.5 mg/kg) kidney pathology scores [3]. |
別名 | BG 9928 |
分子量 | 416.51 |
分子式 | C22H32N4O4 |
CAS No. | 340021-17-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 90 mg/mL (216.1 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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Tonapofylline 340021-17-2 GPCR/G Protein Neuroscience Adenosine Receptor BG-9928 BG 9928 BG9928 Inhibitor inhibitor inhibit