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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T40997 | GLP-1R modulator C16 | GLP-1R modulator C16 | Glucagon Receptor |
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4. | |||
T40279 | GLP-1R modulator L7-028 | GLP-1R modulator L7-028 | cAMP , Glucagon Receptor |
GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling. | |||
T11409 | GLP-26 | HBV | |
GLP-26 disrupts the encapsidation of pre-genomic RNA, causes nucleocapsid disassembly and reduces cccDNA pools. GLP-26 is a HBV capsid assembly modulators (CAM), inhibits HBV DNA replication in Hep AD38 system (IC50=3 nM... | |||
T3984 | GLP-1(7-36), amide | MKC 253,Human GLP-1-(7-36)-amide,Glucagon-like Peptide 1 (7-36) amide,Glucagon-Like Peptide (GLP) I (7-36), amide, human,GLP-1(7-36),GLP-1-(7-36)-amide | Glucagon Receptor |
GLP-1(7-36), amide (MKC 253) is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays various antidiabetic effects by potentiating glucose-... | |||
T37890L | GLP-1(28-36)amide acetate | GLP-1(28-36)amide acetate(1225021-13-5 Free base) | Antioxidant , Glucagon Receptor |
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities. | |||
TP1376 | GLP-1(7-37) acetate(106612-94-6 free base) | GLP-1(7-37) acetate | Others , Glucagon Receptor |
Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion. | |||
T9579L | GLP-1 receptor agonist 9 citrate | GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base) | Glucagon Receptor |
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1. | |||
T37891L | GLP-1(32-36)amide acetate | GLP-1(32-36)amide acetate(1417302-71-6 Free base) | Others |
GLP-1(32-36)amide acetate is a pentapeptide and derived from the C terminus of the glucoregulatory hormone GLP-1. GLP-1(32-36)amide acetate could inhibit weight gain and modulate whole body glucose metabolism in diabetic... | |||
T15387 | GLP-1R Antagonist 1 | Glucagon Receptor | |
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM). | |||
TP2252 | GLP-1 (9-36) amide | Glucagon Receptor | |
antagonist at the human GLP-1 receptor | |||
T36579 | GLP-1R Agonist DMB | Glucagon Receptor | |
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor). | |||
T9579 | GLP-1 receptor agonist 9 | Glucagon Receptor | |
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist. | |||
T63909 | GLP-1R agonist 3 | Glucagon Receptor | |
GLP-1R agonist 3 is a thickened imidazole derivative compound that is a potent agonist of GLP-1R. GLP-1R agonist 3 has shown research potential in diabetes. | |||
T61483 | GLP-1R modulator C5 | Glucagon Receptor | |
GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes. | |||
TP2253 | GLP-2(rat) | GLP-2 (rat) | Others |
intestinal epithelium-specific growth factor | |||
T11408 | Orforglipron | LY3502970,GLP-1 receptor agonist 1 | Glucagon Receptor |
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1 diabetes in adults. | |||
TP1141 | GLP-1(7-36), amide acetate | GLP-1(7-36) Acetate,Human GLP-1-(7-36)-amide Acetate | |
GLP-1(7-36) Acetate is a major intestinal hormone that stimulates glucose-induced insulin secretion from β cells. | |||
TP1157 | GLP-2(1-33)(human) | GLP-2 (human),Glucagon-like peptide 2 (human) | |
GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium. | |||
T37891 | GLP-1(32-36)amide | ||
GLP-1(32-36)amide is a pentapeptide compound derived from the C terminus of the glucoregulatory hormone GLP-1. This compound has shown potential in inhibiting weight gain and regulating glucose metabolism in diabetic mic... | |||
T37890 | GLP-1(28-36)amide | ||
GLP-1(28-36)amide, a C-terminal nonapeptide derived from the cleavage of GLP-1 by neutral endopeptidase (NEP), is a significant product. It functions as an antioxidant and primarily targets the mitochondrion, where it ef... | |||
TP1306 | GLP-1(7-37) | ||
GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells. | |||
T37892 | GLP-1(7-36), amide TFA | ||
GLP-1(7-36), amide TFA is a prominent intestinal hormone known to stimulate glucose-induced insulin secretion from β cells[1]. | |||
TP1316 | GLP-1 moiety from Dulaglutide | ||
GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist. | |||
TP1487 | Glucagon-Like Peptide (GLP) II, human | ||
Glucagon-like peptide 2 (GLP-2) is a recently identified intestinal epithelium-specific growth factor that has been shown to reduce the severity of inflammatory disorders of the intestine in rodent models. Currently Gluc... | |||
T11407 | GLP-1 receptor agonist 2 | Others | |
GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist. | |||
T11404 | GLP-1 receptor agonist 3 | Others | |
GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively. | |||
T11405 | GLP-1 receptor agonist 4 | Others | |
GLP-1 receptor agonist 4 is a glucagon-like peptide-1 receptor (GLP-1R) agonist , has an EC50 of 64.5 nM. GLP-1 receptor agonist 4 can be used in the research for treatment of diabetes. | |||
T36380 | GLP-1 (1-36) amide (human, rat) (trifluoroacetate salt) | ||
GLP-1 amide is a peptide hormone cleaved from proglucagon in the pancreas.1,2 Mice lacking the glucagon receptor (Gcgr-/-) have approximately nine-fold higher levels of total GLP-1 amide, including GLP-1 (1-36) amide and... | |||
T78571 | Albiglutide fragment TFA | GLP-1-Gly8 TFA,GLP-1 (7-36) analog TFA | |
Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as a GLP-1 analog. It functions as a long-acting agonist of the ... | |||
T74609 | GLP-1R agonist 15 | ||
GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] . | |||
T64180 | GLP-1R agonist 1 | ||
GLP-1R agonist 1 is a thickened imidazole derivative compound and a potent agonist of GLP-1R. GLP-1R agonist 1 has potential for the study of diabetes. | |||
T74323 | GLP-1R agonist 4 | ||
GLP-1R agonist 4, a potent agonist of GLP-1R, shows promise for diabetes research[1]. Acting on the principle of glucagon-like peptide-1 (GLP-1), a hypoglycemic hormone secreted by L-cells in the lower gastrointestinal t... | |||
T64007 | GLP-1R agonist 10 | ||
GLP-1R agonist 10 is a GLP-1 agonist (EC50: 0.051 nM). | |||
T74610 | GLP-1R agonist 16 | ||
Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1]. | |||
T64191 | GLP-1R agonist 12 | ||
GLP-1R agonist 12 (Compound 123) is a GLP-1R agonist that can be used in the study of diabetes mellitus. | |||
T72686 | GLP-1R agonist 9 | ||
GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively. | |||
T74608 | GLP-1R agonist 14 | ||
GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1]. | |||
T63999 | GLP-1R agonist 8 | ||
GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 < 2 nM). | |||
T72611 | GLP-1R agonist 17 | ||
GLP-1R agonist 17 is a potent GLP-1 receptor agonist that demonstrates excellent efficacy in activating a GLP-1 receptor. It is primarily utilized in the research of cardiovascular metabolic diseases. | |||
T75823 | GLP-2(rat) TFA | ||
GLP-2(rat) TFA, an intestinal growth factor, promotes cell proliferation and prevents apoptosis. Additionally, it increases mucosal mass and function in the residual small intestine following massive small bowel resectio... | |||
T74132 | GLP-1 receptor agonist 8 | ||
GLP-1 receptor agonist 8, a potent agonist of GLP-1 R, holds potential for diabetes, obesity, and nonalcoholic fatty liver disease (NAFLD) research[1]. | |||
T82308 | GLP-2 (1-34) (human) | ||
GLP-2 (1-34) (human), a polypeptide secreted from the intestine shortly after eating, is utilized in research related to bone remodeling processes [1]. | |||
T82307 | Glp-His-Pro-Gly-NH2 | pGlu-His-Pro-Gly-NH2 | |
pGlu-His-Pro-Gly-NH2, also known as Glp-His-Pro-Gly-NH2, is a tetrapeptide that promotes the release of gonadotropin, luteinizing hormone (LH), and follicle-stimulating hormone (FSH) [1] [2]. | |||
T79348 | GLP-1 receptor agonist 13 | ||
Compound (S)-9, a GLP-1 receptor agonist, exhibits an EC50 of 76 nM for the glucagon GLP-1 receptor [1]. | |||
T64195 | GLP-1 receptor agonist 7 | ||
GLP-1 receptor agonist 7 is a potent glucagon-like peptide-1 (GLP-1) agonist and has shown research potential for GLP-1 related diseases, disorders and conditions, including diabetes. | |||
T75822 | GLP-1(9-36)amide TFA | ||
GLP-1(9-36)amide TFA, a predominant metabolite of glucagon-like peptide-1-(7-36)amide synthesized through dipeptidyl peptidase-4 (DPP-4) activity, functions as an antagonist to the human pancreatic GLP-1 receptor [1] [2]... | |||
T76192 | GLP-1(32-36)amide TFA | ||
GLP-1(32-36)amide TFA, originating from the C-terminal end of the glucoregulatory hormone GLP-1, is a pentapeptide that has demonstrated the ability to mitigate weight gain and regulate glucose metabolism throughout the ... | |||
T76191 | GLP-1(28-36)amide TFA | ||
GLP-1(28-36)amide TFA, a C-terminal nonapeptide derived from GLP-1 cleavage by neutral endopeptidase (NEP), acts as an antioxidant targeting mitochondria. It inhibits mitochondrial permeability transition (MPT), exhibiti... | |||
T64553 | GLP-1(7-37) TFA salt | ||
The truncated glucagon-like peptides GLP-1(7-37) is naturally occurring peptide product of the preproglucagon gene that are synthesized primarily in the intestine and acts as incretin that are released from the intestine... | |||
T80453 | GLP-1 (1-36) amide (human, rat) | Glucagon-like Peptide 1 (1-36) amide (human, rat) | |
GLP-1 (1-36) amide (human, rat) is a molecular variant of the GLP-1 (7-36) amide and has the capacity to stimulate [14C]aminopyrine accumulation in enzymatically dispersed, enriched rat parietal cells [1]. |
カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T3896 | Shanzhiside methyl ester | Glucagon Receptor | |
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 MAPK signaling. | |||
T19117 | 3-Deoxyglucosone | 3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose | GPX , Glucagon Receptor |
3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein amino groups to form advanced glycosylated end proteins (AGE... | |||
T37526 | 2-Oleoylglycerol | 2-Oleoyl Glycerol,2-OG,2-Monoolein | GPR |
2-Oleoylglycerol is a lipid found in palm kernel, sunflower seed and rice bran.2-Oleoylglycerol acts as a GPR119 agonist with neuroprotective effects and induces secretion of glucagon-like peptide 1 (GLP-1).2-Oleoylglyce... | |||
T40977 | Cinnamtannin A2 | ||
Cinnamtannin A2, a tetrameric procyanidin, enhances GLP-1 and insulin secretion in mice while also upregulating the expression of corticotrophin releasing hormone. Additionally, Cinnamtannin A2 exhibits antioxidant, anti... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPJ-00742 | GCG Protein, Human, Recombinant (His) | Human | Human Cells |
Glucagon is a secreted protein and belongs to the glucagon family. Glucagon can be cleved into 8 chains, playing an important role in initiating and maintaining hyperglycemic conditions in diabetes. Glucagon can regulate... | |||
TMPH-01385 | GLP1R Protein, Human, Recombinant (His) | Human | HEK293 |
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ... | |||
TMPH-01384 | GLP1R Protein, Human, Recombinant (E. coli, His) | Human | E. coli |
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ... | |||
TMPH-02676 | GLP1R Protein, Mouse, Recombinant (His & SUMO) | Mouse | E. coli |
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ... | |||
TMPH-03301 | GLP1R Protein, Rat, Recombinant (E. coli, His) | Rat | E. coli |
G-protein coupled receptor for glucagon-like peptide 1 (GLP-1). Ligand binding triggers activation of a signaling cascade that leads to the activation of adenylyl cyclase and increased intracellular cAMP levels. Plays a ... | |||
TMPY-06864 | GLP1R Protein, Human, Recombinant (His & Avi) | Human | HEK293 |
Glucagon-like peptide (GLP)-1 receptor is encoded by GLP1R. GLP1R plays a critical role in mediating the biological actions of GLP1 in mammals and fish. The neuronal GLP1Rs mediate body weight and anorectic effects of li... | |||
TMPH-00575 | GlpD Protein, E. coli, Recombinant (His) | E. coli | E. coli |
Conversion of glycerol 3-phosphate to dihydroxyacetone. Uses molecular oxygen or nitrate as electron acceptor. | |||
TMPH-03302 | GLP1R Protein, Rat, Recombinant (His) | Rat | Yeast |
GLP1R Protein, Rat, Recombinant (His) is expressed in Yeast. | |||
TMPH-01386 | GLP2R Protein, Human, Recombinant (His) | Human | HEK293 |
This is a receptor for glucagon-like peptide 2. The activity of this receptor is mediated by G proteins which activate adenylyl cyclase. | |||
TMPY-00779 | DPP4/CD26 Protein, Human, Recombinant | Human | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-00221 | DPP4/CD26 Protein, Mouse, Recombinant (hFc) | Mouse | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-00778 | DPP4/CD26 Protein, Human, Recombinant (hFc) | Human | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-00122 | DPP4/CD26 Protein, Human, Recombinant (His) | Human | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-04046 | DPP4/CD26 Protein, Cynomolgus, Recombinant | Cynomolgus | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-04251 | DPP4/CD26 Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-00074 | DPP4/CD26 Protein, Mouse, Recombinant (His) | Mouse | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPY-03952 | DPP4/CD26 Protein, Cynomolgus, Recombinant (hFc) | Cynomolgus | HEK293 |
Dipeptidyl peptidase-4 (DPP4) or adenosine deaminase complexing protein 2 (ADCP 2) or T-cell activation antigen CD26 is a serine exopeptidase belonging to the S9B protein family that cleaves X-proline dipeptides from the... | |||
TMPH-03208 | IL-6 Protein, Rabbit, Recombinant (His) | Rabbit | Yeast |
Cytokine with a wide variety of biological functions in immunity, tissue regeneration, and metabolism. Binds to IL6R, then the complex associates to the signaling subunit IL6ST/gp130 to trigger the intracellular IL6-sign... | |||
TMPH-03500 | IL-6 Protein, Sheep, Recombinant (GST) | Sheep | E. coli |
Cytokine with a wide variety of biological functions in immunity, tissue regeneration, and metabolism. Binds to IL6R, then the complex associates to the signaling subunit IL6ST/gp130 to trigger the intracellular IL6-sign... |
カタログ番号 | 製品名 | ||
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L9600 | Peptide Compound Library | 791 compounds | |
791 peptides can be used in peptide drug development and signaling transduction and mechanism study; |