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Search Results for " Tripterygium "

2

阻害剤

26

天然化合物

カタログ番号 製品名 別名 ターゲット
T123808 Triptonoterpene
Triptonoterpene is a natural product found in Tripterygium wilfordii and Tripterygium doianum. Triptonoterpene is an abietane diterpenoid.
T26056 Regelinol
Regelinol is a new antitumor ursene-type triterpenoid isolated from Tripterygium regelii.
カタログ番号 製品名 別名 ターゲット
TN2141 Regelidine Others
Regelidine is a natural product from Tripterygium regelii.
T5S1058 Triptonide PG 492,NSC 165677 Apoptosis , Wnt/beta-catenin , Autophagy
1. Triptonide (PG 492) is effective in the treatment of autoimmune diseases and has potent antileukemic and antitumor activities. 2. Triptonide possesses anti-inflammatory activity, upregulate the expression of IL-37, an...
T3393 Triptophenolide Hypolide,(+)-Triptophenolide Androgen Receptor
Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.
T5S1054 Wilforgine Others
1. Wilforgine exhibits insecticidal activity of some degree.
T3382 Wilforlide A Abruslactone A,3-Epiabruslactone A,Regelide Tyrosinase
Wilforlide A (3-Epiabruslactone A) is a natural product, separated from the ethanolic extract of tripterygium wilfordii. High-dose wilforlide A has obvious anti-inflammatory effect, but has no significant immune suppress...
T3418 Demethylzeylasteral Demethylzeylasteral (T-96) Apoptosis , UGT
Demethylzeylasteral (T-96), isolated from Tripterygium wilfordii, has anti-inflammatory, immunosuppressive and anti-tumor activities. It inhibits the invasion of triple-negative breast cancer by blocking the TGF-β signal...
T26055 Regelin Regelin C
Regelin is an antitumor ursene-type triterpenoid isolated from Tripterygium regelii.
TN5185 Triptonodiol Others
Triptonodiol is a natural product from Tripterygium wilfordii Hook.f.
T80941 Triptonoterpene Me ether
Triptonoterpene Me ether (compound 5), a rosinane-type diterpenoid, is derived from the traditional Chinese medicinal plant, Tripterygium wilfordii Hook. f [1].
TN5960 Polpunonic acid Maytenonic acid,Maytenoic acid
Polpunonic acid is a natural product from Tripterygium wilfordii Hook.f.
TN5255 Wilforol A Others
Wilforol A is a natural product from Tripterygium wilfordii Hook. f.
T80940 Triptonoterpenol
Triptonoterpenol (Compound 6) is a secondary metabolite derived from Tripterygium wilfordii [1].
T83434 1b-Benzoyl-8a-cinnamoyl-4a,5a-dihydroxydihydroagarofuran
1b-Benzoyl-8a-cinnamoyl-4a,5a-dihydroxydihydroagarofuran is a sesquiterpenoid isolated from the root bark of Tripterygium hypoglaucum, characterized by the presence of both a benzoyl and a cinnamoyl group [1].
T40252 Peritassine A
Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties.
T80942 Triptonoditerpenic acid
Triptonoditerpenic acid is an aromatic pimarane diterpenoid that can be isolated from Tripterygium wilfordii. It exhibits cytotoxicity against HepG2, Hep3B, and Bcap37 cell lines, with IC50 values of 42.53 μM, 29.74 μM, ...
TN5188 Triptoquinonide Others
Triptoquinonide is a natural product from Tripterygium wilfordii.
T13936 Triptotriterpenic acid A Maytenfolic acid,Abrusgenic acid Others
Triptotriterpenic acid A is a natural product isolate from Tripterygium wilfordii.
TMA0925 Wilforlide A acetate Others
Wilforlide A (T1) serves as a quality control standard of Tripterygium Glycosides that be listed in Drug Standard of Ministry of Public Health of the People's Republic of China. T1 has anti-inflammatory effects.
TN2283 Tripterifordin HIV Protease
Tripterifordin shows anti-HIV replication activity in H9 lymphocyte cells with an EC50 of 1 microgram/ml.
T80938 Triptotriterpenic acid C
Triptotriterpenic acid C, an ursolic-type compound, can be isolated from the total glycosides extracted from the root of Tripterygium wilfordii Hook.f [1].
T27174 Dihydrocelastrol DHCE. (-)-Triptohypol C,Triptohypol C
Dihydrocelastrol is synthesized by hydrogenation of celastrol, a treterpene isolated from Chinese medicinal plant Tripterygium regelii. Dihydrocelastrol could inhibit cell proliferation and promote apoptosis through casp...
T2179 Triptolide PG490,NSC 163062 Apoptosis , Mdm2 , HSP , NF-κB
Triptolide (PG490) belongs to the tricyclic diterpenoid group of natural products and is an inhibitor of NF-κB activation. Triptolide exhibits immunosuppressive, anti-rheumatic, anti-inflammatory, anti-proliferative and ...
TN1987 Neotriptophenolide Others
Neotriptophenolide is a natural product
T80939 Triptoquinone H
Triptoquinone H, a natural product derived from the traditional Chinese medicinal plant Tripterygium hypoglaucu, exhibits potent cytotoxic, immunomodulatory, and anti-inflammatory properties. It is utilized in research c...
T6S1049 Wilforine ATPase
Wilforine is a sesquiterpene pyridine alkaloid; important bioactive compound in T. wilfordii plants, and is effective in treating idiopathic pulmonary fibrosis. Wilforine has anti-inflammatory effect, which might be medi...
T4S1050 Pristimerin Celastrol methyl ester NF-κB , Antibacterial
1. Pristimerin (Celastrol methyl ester) has anticancer activity , treatment with Pristimerin may be a potential strategy for the suppression of hypoxia-induced metastasis through the reversal of hypoxia-induced stem cell...

天然物製品

Regelidine
TN2141
Synonym:
Target: Others
Triptonide
T5S1058
Synonym: PG 492,NSC 165677
Target: Apoptosis, Wnt/beta-catenin, Autophagy
Triptophenolide
T3393
Synonym: Hypolide,(+)-Triptophenolide
Target: Androgen Receptor
Wilforgine
T5S1054
Synonym:
Target: Others
Wilforlide A
T3382
Synonym: Abruslactone A,3-Epiabruslactone A,Regelide
Target: Tyrosinase
Demethylzeylasteral
T3418
Synonym: Demethylzeylasteral (T-96)
Target: Apoptosis, UGT
Regelin
T26055
Synonym: Regelin C
Target:
Triptonodiol
TN5185
Synonym:
Target: Others
Triptonoterpene Me ether
T80941
Synonym:
Target:
Polpunonic acid
TN5960
Synonym: Maytenonic acid,Maytenoic acid
Target:
Wilforol A
TN5255
Synonym:
Target: Others
Triptonoterpenol
T80940
Synonym:
Target:
1b-Benzoyl-8a-cinnamoyl-4a,5a-dihydroxydihydroagarofuran
T83434
Synonym:
Target:
Peritassine A
T40252
Synonym:
Target:
Triptonoditerpenic acid
T80942
Synonym:
Target:
Triptoquinonide
TN5188
Synonym:
Target: Others
Triptotriterpenic acid A
T13936
Synonym: Maytenfolic acid,Abrusgenic acid
Target: Others
Wilforlide A acetate
TMA0925
Synonym:
Target: Others
Tripterifordin
TN2283
Synonym:
Target: HIV Protease
Triptotriterpenic acid C
T80938
Synonym:
Target:
Dihydrocelastrol
T27174
Synonym: DHCE. (-)-Triptohypol C,Triptohypol C
Target:
Triptolide
T2179
Synonym: PG490,NSC 163062
Target: Apoptosis, Mdm2, HSP, NF-κB
Neotriptophenolide
TN1987
Synonym:
Target: Others
Triptoquinone H
T80939
Synonym:
Target:
Wilforine
T6S1049
Synonym:
Target: ATPase
Pristimerin
T4S1050
Synonym: Celastrol methyl ester
Target: NF-κB, Antibacterial