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Search Results for " cpa "

ターゲット

21

阻害剤

3

天然化合物

10

リコンビナントタンパク質

カタログ番号 製品名 別名 ターゲット
T10876 CPA inhibitor Carboxypeptidase inhibitor Carboxypeptidase
CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.
T16263 N6-Cyclopentyladenosine UK-80882,CPA Adenosine Receptor
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 recepto...
TP1560 C(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively.
T27138 Declopramide OXI-104,IMO-B,3-Chloroprocainamide Apoptosis
Declopramide (OXI-104) is a novel chemosensitizer with antitumor activity that induces apoptosis and can be used to study colorectal cancer and inflammatory bowel disease.
TP1473 Velmupressin c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively.
TP1205 Velmupressin acetate V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively.
T20701 MCPA NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone Others
MCPA(Krezone) is a highly effective phenoxy herbicide. Use of MCPA would have impacts on nearby water and soil resources.
T1025 Tranylcypromine (2-PCPA) hydrochloride Tranylcypromine (2-PCPA) HCl,SKF-385 HCl Histone Demethylase , MAO
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression.
T21519 CCPA 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE Adenosine Receptor
CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor
T22489 2'-MeCCPA 2-Chloro-N-cyclopentyl-2′-C-methyladenosine HCV Protease , Adenosine Receptor
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenylate cyclase activity with an IC value of 13.1 nM.2'-MeCCPA ...
T77567 BCPA Others
BCPA is a non-cytotoxic Pin1 modulator.BCPA modulates osteoclast activation and attenuates the reduction of Pin1 protein, thereby inhibiting RANKL-induced receptor activators of osteoclastogenesis.BCPA is used in the stu...
T60359 Cis-4-Br-2,5-F2-PCPA
cis-4-Br-2,5-F2-PCPA (S1024) inhibits LSD1 and LSD2 with Ki values of 94 nM and 8.4 μM, respectively. There is aberrant expression of LSD1 in cancer stem cells, cis-4-Br-2,5-F2-PCPA inhibits LSD1 cell proliferation and b...
T20948 MCPA-thioethyl HOK 7501,HOK7501,HOK-7501
MCPA-thioethyl is a biochemical.
T81054 T-1-MCPAB VEGFR
T-1-MCPAB, a VEGFR-2 inhibitor with an IC50 of 0.135 µM, effectively suppresses MCF7 cell migration and has applications in cancer research [1].
T41143 PCPA methyl ester hydrochloride 4-Chloro-DL-phenylalanine methyl ester hydrochloride 5-HT Receptor , Hydroxylase
pCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride) is an inhibitor of tryptophan hydroxylase inhibitor and 5-HT synthesis. pCPA methyl ester hydrochloride is permeable across the blood...
T82765 CcpA-IN-1 Antibiotic
CcpA-IN-1 is a Staphylococcus aureus antibiotic exhibiting significant bactericidal activity (MICs=460 nM) [1].
T74170 MOCPAC
MOCPAC is an HDAC1 specific substrate [1] .
T33228 MCPA-potassium
MCPA-potassium is a bioactive chemical.
T33227 MCPA-butyl Yamaclean M
MCPA-butyl is a biochemical.
T82684 Connexin mimetic peptide 40,37GAP26
Connexin mimetic peptide 40,37GAP26, a biologically active peptide, matches the GAP26 domain of the extracellular loop of major vascular connexins Cx37 and Cx40, referred to as 37,40Gap26 based on Cx homology. It has bee...
T71327 Paraxanthine-d6
Paraxanthine-d6 is intended for use as an internal standard for the quantification of paraxanthine by GC- or LC-MS. Paraxanthine is an active metabolite of caffeine. It is formed via N3-demethylation of caffeine by the c...

Compounds

CPA inhibitor
T10876
Synonym: Carboxypeptidase inhibitor
Target: Carboxypeptidase
N6-Cyclopentyladenosine
T16263
Synonym: UK-80882,CPA
Target: Adenosine Receptor
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
TP1560
Synonym:
Target:
Declopramide
T27138
Synonym: OXI-104,IMO-B,3-Chloroprocainamide
Target: Apoptosis
Velmupressin
TP1473
Synonym: c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2
Target:
Velmupressin acetate
TP1205
Synonym: V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate
Target:
MCPA
T20701
Synonym: NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone
Target: Others
Tranylcypromine (2-PCPA) hydrochloride
T1025
Synonym: Tranylcypromine (2-PCPA) HCl,SKF-385 HCl
Target: Histone Demethylase, MAO
CCPA
T21519
Synonym: 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE
Target: Adenosine Receptor
2'-MeCCPA
T22489
Synonym: 2-Chloro-N-cyclopentyl-2′-C-methyladenosine
Target: HCV Protease, Adenosine Receptor
BCPA
T77567
Synonym:
Target: Others
cis-4-Br-2,5-F2-PCPA
T60359
Synonym:
Target:
MCPA-thioethyl
T20948
Synonym: HOK 7501,HOK7501,HOK-7501
Target:
T-1-MCPAB
T81054
Synonym:
Target: VEGFR
pCPA methyl ester hydrochloride
T41143
Synonym: 4-Chloro-DL-phenylalanine methyl ester hydrochloride
Target: 5-HT Receptor, Hydroxylase
CcpA-IN-1
T82765
Synonym:
Target: Antibiotic
MOCPAC
T74170
Synonym:
Target:
MCPA-potassium
T33228
Synonym:
Target:
MCPA-butyl
T33227
Synonym: Yamaclean M
Target:
Connexin mimetic peptide 40,37GAP26
T82684
Synonym:
Target:
Paraxanthine-d6
T71327
Synonym:
Target:
カタログ番号 製品名 別名 ターゲット
T2895 Lupeol Fagarasterol,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol Apoptosis , Androgen Receptor , Akt
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
T15027 Cyclopiazonic acid Calcium Channel
Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A. flavus. Cyclopiazonic acid (CPA) is an endoplasmic reticulum calcium ATPase (Ca2+ATPase; SERCA)nanomolar inhibitor and a potent inducer of ce...
T8093 2-Benzylsuccinic acid DL-Benzylsuccinic acid Carboxypeptidase
2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.

Recombinant Proteins

カタログ番号 製品名 Species Expression System
TMPJ-00474 CPA1 Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxypeptidase A1 (CPA1) is secreted as a pancreatic peptidase that comes from the precursor form of inactive procarboxypeptidase. CPA1 comprises a signal peptide, a pro region and a mature chain, and can be activated ...
TMPY-01729 Carboxypeptidase A Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxypeptidase A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is P15085.
TMPY-01362 Carboxypeptidase A Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Carboxypeptidase A Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is Q7TPZ8.
TMPH-03260 Carboxypeptidase A1 Protein, Rat, Recombinant (His & Myc) Rat E. coli
Carboxypeptidase that catalyzes the release of a C-terminal amino acid, but has little or no action with -Asp, -Glu, -Arg, -Lys or -Pro. Catalyzes the conversion of leukotriene C4 to leukotriene F4 via the hydrolysis of ...
TMPH-01641 CPA3 Protein, Human, Recombinant (His) Human E. coli
CPA3 Protein, Human, Recombinant (His) is expressed in E. coli.
TMPJ-01184 CPA4 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Carboxypeptidase A4 (CPA4) is a member of the peptidase M14 family. CPA4 is metalloprotease that could be involved in the histone hyperacetylation pathway. CPA4 binds one zinc ion per subunit and could catalyze to releas...
TMPJ-00602 CPA2 Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxypeptidase A2 (CPA) is a secreted pancreatic procarboxy-peptidase that cleaves the C-terminal amide or ester bond of peptides that have a free C-terminal carboxyl group. The hydrolytic action of CPA2 was identified...
TMPY-00332 CPA2 Protein, Rat, Recombinant (His) Rat HEK293 Cells
CPA2 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.5 kDa and the accession number is A6IEG7.
TMPY-02664 Carboxypeptidase A2 Protein, Mouse, Recombinant (His) Mouse HEK293 Cells
Carboxypeptidase A2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.6 kDa and the accession number is Q504N0.
TMPY-00726 Carboxypeptidase A2 Protein, Human, Recombinant (His) Human HEK293 Cells
Carboxypeptidase A2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46 kDa and the accession number is P15085.