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カタログ番号 | 製品名 | 別名 | ターゲット |
---|---|---|---|
T10876 | CPA inhibitor | Carboxypeptidase inhibitor | Carboxypeptidase |
CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM. | |||
T16263 | N6-Cyclopentyladenosine | UK-80882,CPA | Adenosine Receptor |
N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's of 2.3 nM, 790 nM, and 43 nM for human A1, A2A, and A3 recepto... | |||
TP1560 | C(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm | ||
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm a highly efficient, selective and short-acting peptide V2 receptor agonist (V2R), with EC50s of hV2R and rV2R being 0.25 and 0.05 nM, respectively. | |||
T27138 | Declopramide | OXI-104,IMO-B,3-Chloroprocainamide | Apoptosis |
Declopramide (OXI-104) is a novel chemosensitizer with antitumor activity that induces apoptosis and can be used to study colorectal cancer and inflammatory bowel disease. | |||
TP1473 | Velmupressin | c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 is a selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07nM and 0.02 nM for hV2R and rV2R, respectively. | |||
TP1205 | Velmupressin acetate | V2 receptor (V2R) agonist,c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate | |
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively. | |||
T20701 | MCPA | NSC-2351,Krezone,NSC2351,NSC 2351,U 46 M-Fluid,Raphone | Others |
MCPA(Krezone) is a highly effective phenoxy herbicide. Use of MCPA would have impacts on nearby water and soil resources. | |||
T1025 | Tranylcypromine (2-PCPA) hydrochloride | Tranylcypromine (2-PCPA) HCl,SKF-385 HCl | Histone Demethylase , MAO |
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and atypical depression. | |||
T21519 | CCPA | 2-chloro-N(6)cyclopentyladenosine,2-CHLORO-N-CYCLOPENTYLADENOSINE | Adenosine Receptor |
CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor | |||
T22489 | 2'-MeCCPA | 2-Chloro-N-cyclopentyl-2′-C-methyladenosine | HCV Protease , Adenosine Receptor |
2'-MeCCPA is a potent and highly selective A1 adenosine receptor (A1AR) agonist with a K-value of 1.8 nM for AR.2'-MeCCPA inhibits trichostatin-stimulated adenylate cyclase activity with an IC value of 13.1 nM.2'-MeCCPA ... | |||
T77567 | BCPA | Others | |
BCPA is a non-cytotoxic Pin1 modulator.BCPA modulates osteoclast activation and attenuates the reduction of Pin1 protein, thereby inhibiting RANKL-induced receptor activators of osteoclastogenesis.BCPA is used in the stu... | |||
T60359 | Cis-4-Br-2,5-F2-PCPA | ||
cis-4-Br-2,5-F2-PCPA (S1024) inhibits LSD1 and LSD2 with Ki values of 94 nM and 8.4 μM, respectively. There is aberrant expression of LSD1 in cancer stem cells, cis-4-Br-2,5-F2-PCPA inhibits LSD1 cell proliferation and b... | |||
T20948 | MCPA-thioethyl | HOK 7501,HOK7501,HOK-7501 | |
MCPA-thioethyl is a biochemical. | |||
T81054 | T-1-MCPAB | VEGFR | |
T-1-MCPAB, a VEGFR-2 inhibitor with an IC50 of 0.135 µM, effectively suppresses MCF7 cell migration and has applications in cancer research [1]. | |||
T41143 | PCPA methyl ester hydrochloride | 4-Chloro-DL-phenylalanine methyl ester hydrochloride | 5-HT Receptor , Hydroxylase |
pCPA methyl ester hydrochloride (4-Chloro-DL-phenylalanine methyl ester hydrochloride) is an inhibitor of tryptophan hydroxylase inhibitor and 5-HT synthesis. pCPA methyl ester hydrochloride is permeable across the blood... | |||
T82765 | CcpA-IN-1 | Antibiotic | |
CcpA-IN-1 is a Staphylococcus aureus antibiotic exhibiting significant bactericidal activity (MICs=460 nM) [1]. | |||
T74170 | MOCPAC | ||
MOCPAC is an HDAC1 specific substrate [1] . | |||
T33228 | MCPA-potassium | ||
MCPA-potassium is a bioactive chemical. | |||
T33227 | MCPA-butyl | Yamaclean M | |
MCPA-butyl is a biochemical. | |||
T82684 | Connexin mimetic peptide 40,37GAP26 | ||
Connexin mimetic peptide 40,37GAP26, a biologically active peptide, matches the GAP26 domain of the extracellular loop of major vascular connexins Cx37 and Cx40, referred to as 37,40Gap26 based on Cx homology. It has bee... | |||
T71327 | Paraxanthine-d6 | ||
Paraxanthine-d6 is intended for use as an internal standard for the quantification of paraxanthine by GC- or LC-MS. Paraxanthine is an active metabolite of caffeine. It is formed via N3-demethylation of caffeine by the c... |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T2895 | Lupeol | Fagarasterol,Monogynol B,Clerodol,(3β,13ξ)-Lup-20(29)-en-3-ol,Farganasterol | Apoptosis , Androgen Receptor , Akt |
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity. | |||
T15027 | Cyclopiazonic acid | Calcium Channel | |
Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A. flavus. Cyclopiazonic acid (CPA) is an endoplasmic reticulum calcium ATPase (Ca2+ATPase; SERCA)nanomolar inhibitor and a potent inducer of ce... | |||
T8093 | 2-Benzylsuccinic acid | DL-Benzylsuccinic acid | Carboxypeptidase |
2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite. |
カタログ番号 | 製品名 | Species | Expression System |
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TMPJ-00474 | CPA1 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A1 (CPA1) is secreted as a pancreatic peptidase that comes from the precursor form of inactive procarboxypeptidase. CPA1 comprises a signal peptide, a pro region and a mature chain, and can be activated ... | |||
TMPY-01729 | Carboxypeptidase A Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is P15085. | |||
TMPY-01362 | Carboxypeptidase A Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Carboxypeptidase A Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is Q7TPZ8. | |||
TMPH-03260 | Carboxypeptidase A1 Protein, Rat, Recombinant (His & Myc) | Rat | E. coli |
Carboxypeptidase that catalyzes the release of a C-terminal amino acid, but has little or no action with -Asp, -Glu, -Arg, -Lys or -Pro. Catalyzes the conversion of leukotriene C4 to leukotriene F4 via the hydrolysis of ... | |||
TMPH-01641 | CPA3 Protein, Human, Recombinant (His) | Human | E. coli |
CPA3 Protein, Human, Recombinant (His) is expressed in E. coli. | |||
TMPJ-01184 | CPA4 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Carboxypeptidase A4 (CPA4) is a member of the peptidase M14 family. CPA4 is metalloprotease that could be involved in the histone hyperacetylation pathway. CPA4 binds one zinc ion per subunit and could catalyze to releas... | |||
TMPJ-00602 | CPA2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A2 (CPA) is a secreted pancreatic procarboxy-peptidase that cleaves the C-terminal amide or ester bond of peptides that have a free C-terminal carboxyl group. The hydrolytic action of CPA2 was identified... | |||
TMPY-00332 | CPA2 Protein, Rat, Recombinant (His) | Rat | HEK293 Cells |
CPA2 Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.5 kDa and the accession number is A6IEG7. | |||
TMPY-02664 | Carboxypeptidase A2 Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Carboxypeptidase A2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.6 kDa and the accession number is Q504N0. | |||
TMPY-00726 | Carboxypeptidase A2 Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Carboxypeptidase A2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46 kDa and the accession number is P15085. |