Powder: -20°C for 3 years | In solvent: -80°C for 1 year
APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively.
説明 | APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119, respectively. |
ターゲット&IC50 | GPR119 (rat):33 nM (EC50), GPR119 (human):2.7 nM (EC50) |
別名 | APD 668 |
分子量 | 477.51 |
分子式 | C21H24FN5O5S |
CAS No. | 832714-46-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (94.24 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
APD668 832714-46-2 Endocrinology/Hormones GPCR/G Protein Membrane transporter/Ion channel Metabolism GPR P450 Potassium Channel Inhibitor CYPs diabetes Cytochrome P450 APD-668 GPR119 coupled G-protein steatohepatitis CYP2C9 G Protein-Coupled Receptor 119 APD 668 inhibit KcsA inhibitor