Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM
パッケージサイズ | 在庫状況 | 単価(税別) | |||
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2 mg | 在庫あり | ¥ 7,000 | |||
5 mg | 在庫あり | ¥ 11,000 | |||
10 mg | 在庫あり | ¥ 18,500 | |||
25 mg | 在庫あり | ¥ 30,500 | |||
50 mg | 在庫あり | ¥ 45,000 | |||
100 mg | 在庫あり | ¥ 66,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 12,000 |
説明 | BRD9539 is an inhibitor of euchromatin histone methyltransferase 2 (EHMT2), also known as G9a, with an IC50 value of 6.3 μM |
ターゲット&IC50 | G9a:6.3 μM (IC50) |
In vitro | BRD9539 is selective for G9a and PRC2 over SU39H1 and NDMT1 up to a concentration of 40 μM. It is more potent than BRD4770 in enzyme assays but has no activity in cell-based assays when used at concentrations of 5 and 10 μM. |
分子量 | 399.44 |
分子式 | C24H21N3O3 |
CAS No. | 1374601-41-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 35 mg/mL (87.62 mM)
You can also refer to dose conversion for different animals. 詳細
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
BRD9539 1374601-41-8 Chromatin/Epigenetic Histone Methyltransferase chromatin BRD 9539 PRC2 G9a senescent inhibit H3K9 histones Inhibitor EHMT2 BRD-9539 inhibitor