Powder: -20°C for 3 years | In solvent: -80°C for 1 year
3-Epiursolic acid may have antiinflammatory activity, it shows inhibition on Cathepsins L (catL), the IC50 value of 6.5 μM, cathepsins L (catL) and B play an important role in tumor progression and have been considered promising therapeutic targets in the development of novel anticancer agents.
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 21,000 | |||
5 mg | 在庫あり | ¥ 44,500 | |||
10 mg | 在庫あり | ¥ 76,500 | |||
25 mg | 在庫あり | お問い合わせ | |||
50 mg | 在庫あり | お問い合わせ | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 52,500 |
説明 | 3-Epiursolic acid may have antiinflammatory activity, it shows inhibition on Cathepsins L (catL), the IC50 value of 6.5 μM, cathepsins L (catL) and B play an important role in tumor progression and have been considered promising therapeutic targets in the development of novel anticancer agents. |
ターゲット&IC50 | Cathepsin L:19.5 μM (Ki), Cathepsin L:6.5 μM (IC50) |
In vitro | All three extracts were found to exhibit antiinflammatory activity with the chloroform extract being the most active. Chemical investigations of petroleum ether and chloroform extracts led to the isolation of beta-sitosterol, ursolic acid, oleanolic acid, 3-Epiursolic acid, 3-epioleanolic acid, and minor triterpenoids of derivatives of ursolic acid and oleanolic acids. Chromatographic purification of the methanol extract yielded two iridoid glucosides, verbenalin and hastatoside, a phenylpropanoid glycoside, verbascoside and beta-sitosterol-D-glucoside. |
植物由来 |
分子量 | 456.7 |
分子式 | C30H48O3 |
CAS No. | 989-30-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 45 mg/mL (98.53 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. 詳細
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3-Epiursolic acid 989-30-0 Immunology/Inflammation Proteases/Proteasome Cysteine Protease Immunology/Inflammation related inhibit Cathepsin 3 Epiursolic acid 3-Epiursolic Acid 3Epiursolic acid Inhibitor inhibitor