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カタログ番号 | 製品名 | 別名 | ターゲット |
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T26887 | BOP | ||
BOP is anantagonist of alpha4beta1/alpha9beta1 integrins. BOP rapidly mobilizes long-term multi-lineage reconstituting hematopoietic stem cells (HSC). | |||
T41149 | BOP-JF549 | BOP-JF549 | |
BOP-JF549 is a fluorescent dual α9β1/α4β1 integrin inhibitor. Comprises BOP conjugated to Janelia Fluor® 549. Fluorogenic: fluoresces only once bound to integrins, enabling hassle-free no-wash experiments. Bright and pho... | |||
T41153 | BOP-JF646 | BOP-JF646 | |
BOP-JF646 is a fluorescent dual α9β1/α4β1 integrin inhibitor. Comprises BOP conjugated to Janelia Fluor®646. Fluorogenic: fluoresces only once bound to integrins, enabling hassle-free no-wash experiments. Bright and phot... | |||
T26888 | BOP sodium | BOP sodium salt | |
BOP sodium salt is an inhibitor of alpha9beta1 and alpha4beta1 integrin. | |||
T35585 | I-BOP | ||
I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP). I-BOP promotes cell proliferation by activating the PI3K pathway in vascular smooth muscle. | |||
T34905 | Totrombopag | SB559448,SB 559448,SB-559448,LGD-4665,Synonym 2,LGD 4665,LGD4665 | |
Totrombopag (SB559448) is a candidate compound for action on RSV polymerase. | |||
T12285 | Ebopiprant | OBE022,OBE-022 | Others |
TQ0223 | Lusutrombopag | S-888711,Mulpleta | Thrombin , Thrombopoietin Receptor |
Lusutrombopag (Mulpleta) is an orally bioavailable, small molecule thrombopoietin (TPO) receptor agonist for chronic liver disease (CLD) patients with thrombocytopenia prior to elective invasive surgery. | |||
T3187 | Fluoroclebopride | Dopamine Receptor | |
Fluoroclebopride is a dopamine (DA) D2 receptor ligand. | |||
T1058 | Carboplatin | NSC 241240,CBDCA,JM-8 | DNA Alkylator/Crosslinker , DNA/RNA Synthesis , Autophagy |
Carboplatin (JM-8) is a cisplatin derivative, a DNA synthesis inhibitor. Carboplatin binds to DNA, inhibits replication and transcription, and induces cell death. Carboplatin has antitumor activity. | |||
T7569 | Clebopride malate | Dopamine Receptor | |
Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting. | |||
T7417 | Avatrombopag | YM477,AKR-501,E5501 | Thrombin , Thrombopoietin Receptor |
Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiation and platelet production. | |||
T17018 | TCPOBOP | BCL | |
TCPOBOP is a constitutive androstane receptor agonist that induces robust hepatocyte proliferation and hepatomegaly. TCPOBOP decreases Fas-induced murine liver injury by altering Bcl-2 proteins. | |||
T6825 | Eltrombopag Olamine | Promacta Olamine,Revolade,Eltrombopag diethanolamine salt,SB497115,SB-497115GR | Thrombin |
Eltrombopag Olamine (Eltrombopag diethanolamine salt) is the orally active ethanolamine salt of eltrombopag, a small-molecule, nonpeptide thrombopoietin receptor agonist with megakaryopoiesis-stimulating activity. Eltrom... | |||
T13098 | TBOPP | Others | |
TBOPP is a selective DOCK1 inhibitor (IC50 : 8.4 μM), with anti-tumor activity for broader types of tumors. | |||
T2562 | Eltrombopag | SB-497115,SB-497115-GR | Thrombin |
Eltrombopag (SB-497115-GR), an orally active thrombopoietin receptor agonist with megakaryopoiesis stimulating activity, binds to and stimulates the platelet thrombopoietin receptor (TPO-R or CD110). | |||
T22285 | Carboprost | 15(S)-15-Methyl Prostaglandin F2α,15-Methyl-PGF2α | Prostaglandin Receptor |
Carboprost (15(S)-15-Methyl Prostaglandin F2α) is a synthetic prostaglandin analogue of PGF2α which has the effect of oxytocic. Carboprost is commonly used to restore uterine tone. | |||
T63356 | Bopindolol fumarate | ||
Bopindolol ((±)-Bopindolol) fumarate is an orally active β-adrenoceptor (ARs) antagonist with partial agonist activity that is non-selective for β1- and β2-ARs and has low affinity for the β3-AR subtype. Bopindolol fumar... | |||
T9451 | Bopindolol | ||
Bopindolol is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol is a prodrug of pindolol... | |||
T40654 | Avatrombopag hydrochloride | AKR-501 hydrochloride,YM477hydrochloride,E5501hydrochloride | |
Avatrombopag hydrochloride (AKR-501) is an orally active, nonpeptide agonist of the thrombopoietin (TPO) receptor with an EC 50 of 3.3 nM. It effectively mimics the biological activities of TPO, stimulating platelet prod... | |||
T68560 | Totrombopag choline | ||
Totrombopag, also known LGD-4665, GSK2285921 and SB559448, is an oral thromobopoietin receptor agonist, is being developed as a new generation small molecule thrombopoietin (TPO) mimetic. It is a highly selective and po... | |||
T34637 | Sibopirdine | X9121,EXP921 | |
Sibopirdine is a new type of cognitive enhancer and intelligence booster that has been studied as a cognitive enhancer for the treatment of Alzheimer's disease. | |||
T27536 | Hetrombopag olamine | ||
Hetrombopag olamine is a non-peptide thrombopoietin (TPO) receptor agonist with oral activity. | |||
T70000 | Ebopiprant HCl | ||
Ebopiprant, also known as OBE-022, is an Oral and Selective Prostaglandin F 2α Receptor Antagonist as an Effective and Safe Modality for the Treatment of Preterm Labor. OBE022 exhibits potent tocolytic effects on human ... | |||
T7569L | Clebopride | ||
Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic. | |||
T72265 | Eltrombopag methyl ester | ||
Eltrombopag Methyl Ester, a derivative of Eltrombopag, functions as a thrombopoietin (Tpo) receptor agonist to enhance platelet production and is employed in the study of certain thrombocytopenia variants. | |||
T62864 | Hetrombopag | ||
Hetrombopag is a potent agonist of the thrombopoietin receptor. Hetrombopag is well tolerated and has a controlled safety profile. hetrombopag has potential for studies in immune thrombocytopenia. | |||
T62865 | Rafutrombopag | ||
Rafutrombopag is a thrombopoietin (TPO) agonist. | |||
T68888 | Avatrombopag maleate | ||
Avatrombopag, also known as AKR-501, YM477, AS 1670542 or E5501, is a novel orally-active thrombopoietin (TPO) receptor agonist. AKR-501 specifically targeted the TPO receptor and stimulated megakaryocytopoiesis througho... | |||
T35871 | Bopindolol (malonate) | ||
Bopindolol is a non-selective β-adrenergic receptor antagonist. In vivo, bopindolol decreases heart rate and blood pressure and attenuates ischemia-induced myocardial acidosis in dogs. Formulations containing bopindolol ... | |||
T41152 | R-BC154 | R-BC154 | |
R-BC154 is a high affinity fluorescent α4β1/α9β1 inhibitor (Kdvalues are 12.7 and 38 nM, respectively); fluorescent version of BOP. Rapidly and preferentially mobilizes HSCs and progenitorsin vivo. Excitation maximum, 56... | |||
T36160 | 8-iso Prostaglandin E2 | 8-iso Prostaglandin E2 | |
8-iso PGE2 is one of several isoprostanes produced from arachidonic acid during lipid peroxidation. It is a potent renal vasoconstrictor in the rat. 8-iso PGE2 inhibits U-46619 or I-BOP-induced platelet aggregation with ... | |||
T80224 | Bid BH3 (80-99) | ||
Bid BH3 (80-99) is a biologically active peptide known as a pro-apoptotic member of the 'BH3-only' (BOPS) subset within the BCL-2 protein family, pivotal in apoptosis regulation. It notably interacts with Bcl-2, Bax, and... |
カタログ番号 | 製品名 | 別名 | ターゲット |
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T14865 | Carboprost tromethamine | Prostaglandin Receptor | |
Carboprost tromethamine, a synthetic 15-methyl analogue of prostaglandin F2α, effectively promotes uterine contractions and significantly reduces bleeding during and post-delivery. | |||
TN4394 | Kobophenol A | MMP , BCL , p38 MAPK , NF-κB , ROS , DNA/RNA Synthesis , CDK , JNK | |
Kobophenol A has antimicrobial, and anti-inflammatory activities, it might be a candidate for treatment of inflammatory bone diseases relevant to osteoblast cell death. Kobophenol A inhibits AChE activity in a dose-depen... |
カタログ番号 | 製品名 | Species | Expression System |
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TMPH-00785 | Bacteriorhodopsin Protein, Halobacterium halobium, Recombinant (His & Myc & SUMO) | Halobacterium halobium | E. coli |
Light-driven proton pump. | |||
TMPY-00939 | Thrombopoietin Protein, Mouse, Recombinant (His) | Mouse | HEK293 Cells |
Thrombopoietin Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37 kDa and the accession number is P40226-1. | |||
TMPY-01609 | Thrombopoietin Protein, Cynomolgus, Recombinant (His) | Cynomolgus | HEK293 Cells |
Thrombopoietin Protein, Cynomolgus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 36.8 kDa and the accession number is XP_005546625.1. | |||
TMPY-00157 | Ribophorin II Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Ribophorin II Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 84 kDa and the accession number is P04844-1. | |||
TMPY-00164 | Ribophorin II Protein, Human, Recombinant (His) | Human | HEK293 Cells |
Ribophorin II Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 58.4 kDa and the accession number is P04844-1. | |||
TMPY-04201 | Thrombopoietin Protein, Human, Recombinant (hFc) | Human | HEK293 Cells |
Thrombopoietin Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 45 kDa and the accession number is P40225-1. |