Powder: -20°C for 3 years | In solvent: -80°C for 1 year
HJC0197 selectively blocks cAMP-induced Epac activation. HJC0197 is an effective exchange protein. Which straightly activated by cAMP (Epac) antagonist (IC50=5.9 μM for Epac2).
パッケージサイズ | 在庫状況 | 単価(税別) | |||
---|---|---|---|---|---|
サンプルについてお問い合わせ | |||||
1 mg | 在庫あり | ¥ 9,000 | |||
5 mg | 在庫あり | ¥ 19,500 | |||
10 mg | 在庫あり | ¥ 30,000 | |||
25 mg | 在庫あり | ¥ 52,500 | |||
50 mg | 在庫あり | ¥ 85,000 | |||
100 mg | 在庫あり | ¥ 126,000 | |||
1 mL * 10 mM (in DMSO) | 在庫あり | ¥ 22,500 |
説明 | HJC0197 selectively blocks cAMP-induced Epac activation. HJC0197 is an effective exchange protein. Which straightly activated by cAMP (Epac) antagonist (IC50=5.9 μM for Epac2). |
In vitro | In the presence of an equal concentration of cAMP, HJC0197 (25 μM) also inhibits Epac1-mediated Rap1-GDP exchange activity at 25 μM. |
分子量 | 339.45 |
分子式 | C19H21N3OS |
CAS No. | 1383539-73-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 25 mg/mL (73.65 mM)
You can also refer to dose conversion for different animals. 詳細
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HJC0197 1383539-73-8 GPCR/G Protein MAPK cAMP Ras cAMP-signaling activation GEF cellular inhibit HJC-0197 phosphorylation processes HJC 0197 Inhibitor inhibitor