T9 | TargetMol

カタログ番号	製品名	別名	ターゲット
T13246	UCT943		Parasite , PI4K
			Parasite , PI4K
T7302	CU-CPT9b	CU-CPT-9b,TLR8-specific antagonist 1	TLR
	CU-CPT9b (TLR8-specific antagonist 1) is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM). It inhibits activation of NF- B induced by the TLR8 agonist R-848 in TLR8-overexpressing HEK-Blue cells with an IC50 valu...		TLR
T14841	BVT948		Phosphatase , P450 , Histone Methyltransferase
	BVT948 is a protein tyrosine phosphatase (PTP) inhibitor. It can also inhibit several CYP450 isoforms and lysine methyltransferase SETD8 (KMT5A).		Phosphatase , P450 , Histone Methyltransferase
T5207	LIT927	LIT 927,LIT-927	CXCR
	LIT927 (LIT-927) is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to CXCR4).		CXCR
T3068	AT9283	J-504568	Apoptosis , FLT , JAK , Bcr-Abl , Aurora Kinase , Autophagy
	AT9283 (J-504568) is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora B and Abl(T315I).		Apoptosis , FLT , JAK , Bcr-Abl , Aurora Kinase , Autophagy
T4354	KPT9274	KPT-9274,KPT 9274,PAK4-IN-1	NAMPT , PAK
	KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.		NAMPT , PAK
T33616	NDT9520492	NDT 9520492,NDT-9520492
	NDT9520492 is a bioactive chemical.
T76593	(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)
	Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon), a gonadotropin-releasing hormone (GnRH) analog, effectively induces ovulation and/or spawning in farmed fish [1].
T69227	GT951
	GT951 is a EAAT2 activator.

Compounds

UCT943

T13246

Synonym:

Target: Parasite, PI4K

CU-CPT9b

T7302

Synonym: CU-CPT-9b,TLR8-specific antagonist 1

Target: Phosphatase, P450, Histone Methyltransferase

LIT927

T5207

Synonym: LIT 927,LIT-927

Target: Apoptosis, FLT, JAK, Bcr-Abl, Aurora Kinase, Autophagy

KPT9274

T4354

Synonym: KPT-9274,KPT 9274,PAK4-IN-1

Target: NAMPT, PAK

NDT9520492

T33616

Synonym: NDT 9520492,NDT-9520492

Target:

(Des-Gly10,D-Ala6,Pro-NHEt9)-LHRH (salmon)

カタログ番号	製品名	別名	ターゲット
T81052	T988C	(+)-T988C
	T988C, a heptacyclic epidithiodioxopiperazine (ETP) natural product, exhibits potent cytotoxicity against cultured P388 leukemia cells [1].

Recombinant Proteins

Species：

Expression System：

Tag：

カタログ番号	製品名	Species	Expression System
TMPY-05096	Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 103.6 kDa and the accession number is CAA25527.1.
TMPY-01873	Transferrin Receptor/TFRC Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is AAA61153.1.
TMPY-01897	PRSS3 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	Trypsin-3, also known as Trypsin III, brain trypsinogen, Serine protease 3 and PRSS3, is a secreted protein that belongs to the peptidase S1 family. Trypsin-3 / PRSS3 is expressed is in pancreas and brain. It contains on...
TMPY-05617	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated	Human	HEK293 Cells
	Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is P02786.
TMPK-00374	Transferrin R/CD71 Protein, Human, Recombinant (His & Avi)	Human	HEK293 Cells
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-00376	Transferrin R/CD71 Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-01261	Transferrin R/CD71 Protein, Cynomolgus, Recombinant (His)	Cynomolgus	HEK293 Cells
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPK-00375	Transferrin R/CD71 Protein, Human, Recombinant (His & Avi), Biotinylated	Human	HEK293 Cells
	The transferrin receptor (CD71) is known as a receptor for IgA1 on mesangial cells. The transcript and protein expression of glomerular CD71 was determined by real-time polymerase chain reaction and immunohistochemistry....
TMPJ-00378	Transferrin Receptor/TFRC Protein, Human, Recombinant (aa 101-760, His)	Human	HEK293 Cells
	Transferrin receptor protein 1 (TFRC) belongs to the peptidase M28 family that is synthesized as a 172 amino acid (aa). TFRC regulated by cellular iron levels through binding of the iron regulatory proteins, IRP1 and IRP...
TMPY-06287	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His & Avi), Biotinylated	SARS-CoV-2	Baculovirus Insect Cells
	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His & Avi), Biotinylated is expressed in Baculovirus insect cells with His and Avi tag. The predicted molecular weight is 136...
TMPY-06395	SARS-CoV-2 Spike S1 Protein (L5F & T95I & D253G & S477N & E484K & D614G, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (L5F & T95I & D253G & S477N & E484K & D614G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.39 kDa and the accession number is A0A6G7K2L4.
TMPY-02845	CST9L Protein, Human, Recombinant (hFc)	Human	HEK293 Cells
	Testatin is a member of the Cystatin family. Cystatins comprise genes that all show expression patterns that are strikingly restricted to reproductive tissue. Cystatins are a family of cysteine protease inhibitors with h...
TMPY-06444	SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (T19R & T95I & E156G & 157-158 deletion & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.23 kDa and the accession...
TMPY-06271	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His)	SARS-CoV-2	Baculovirus Insect Cells
	SARS-CoV-2 Spike S1+S2 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R & Q1071H, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134.51 kDa and the accession nu...
TMPY-06251	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.58 kDa and the accession number is A0A6G7K...
TMPY-06293	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His & Avi), Biotinylated	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (T95I & G142D & E154K & L452R & E484Q & D614G & P681R, His & Avi), Biotinylated is expressed in HEK293 mammalian cells with His and Avi tag. The predicted molecular weight is 78.39 kDa and the...
TMPY-06443	SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (T19R & T95I & G142D & Y145H & E156G & 157-158 deletion & A222V & L452R & T478K & D614G & P681R, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76....
TMPY-06421	SARS-CoV-2 Spike S1 Protein (T95I & Y144S & Y145N & R346K & E484K & N501Y & D614G & P681H, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 Protein (T95I & Y144S & Y145N & R346K & E484K & N501Y & D614G & P681H, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 76.36 kDa and the accession number is...
TMPY-06393	SARS-CoV-2 Spike S1+S2 Protein (L5F & T95I & D253G & S477N & E484K & D614G & A701V, His)	SARS-CoV-2	Baculovirus Insect Cells
	SARS-CoV-2 Spike S1+S2 Protein (L5F & T95I & D253G & S477N & E484K & D614G & A701V, His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 134.34 kDa and the accession number is A0A...
TMPY-06422	SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His)	SARS-CoV-2	HEK293 Cells
	SARS-CoV-2 Spike S1 NTD Protein (T19R & T95I & G142D & 156-157 deletion & R158G, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 34.10 kDa and the accession number is A0A6G7K2L...
TMPY-06647	CHST9 Protein, Human, Recombinant (His)	Human	HEK293 Cells
	CHST9 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 17.66 kDa and the accession number is NP_113610.2.